Catalytic Asymmetric Addition Reactions of Carbonyls. A Common Catalytic Approach
Jørgensen, Karl Anker, Johannsen, Mogens, Yao, Sulan, Audrain, Hélène, Thorhauge, Jacob
Published in Accounts of chemical research (20.07.1999)
Published in Accounts of chemical research (20.07.1999)
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Journal Article
New Catalysts for the Asymmetric Hydrosilylation of Ketones Discovered by Mass Spectrometry Screening
Yao, Sulan, Meng, Jun-Cai, Siuzdak, Gary, Finn, M. G
Published in Journal of organic chemistry (04.04.2003)
Published in Journal of organic chemistry (04.04.2003)
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Journal Article
Synthesis and biological activity of new 5- O-sugar modified ketolide and 2-fluoro-ketolide antibiotics
Liang, Chang-Hsing, Yao, Sulan, Chiu, Yu-Hung, Leung, Po Yee, Robert, Nicole, Seddon, Jaime, Sears, Pam, Hwang, Chan-Kou, Ichikawa, Yoshi, Romero, Alex
Published in Bioorganic & medicinal chemistry letters (01.03.2005)
Published in Bioorganic & medicinal chemistry letters (01.03.2005)
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Journal Article
Structure–activity relationships of bivalent aminoglycosides and evaluation of their microbiological activities
Liang, Chang-Hsing, Romero, Alex, Rabuka, David, Sgarbi, Paulo W.M., Marby, Kenneth A., Duffield, Jonathan, Yao, Sulan, Cheng, Mayling L., Ichikawa, Yoshi, Sears, Pamela, Hu, Changyong, Hwang, San-Bao, Shue, Youe-Kong, Sucheck, Steven J.
Published in Bioorganic & medicinal chemistry letters (15.04.2005)
Published in Bioorganic & medicinal chemistry letters (15.04.2005)
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Journal Article
Use of a racemic derivatizing agent for measurement of enantiomeric excess by circular dichroism spectroscopy
Hattori, Tetsutaro, Minato, Yuji, Yao, Sulan, Finn, M.G, Miyano, Sotaro
Published in Tetrahedron letters (05.11.2001)
Published in Tetrahedron letters (05.11.2001)
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Journal Article
ARX788, a Site-specific Anti-HER2 Antibody–Drug Conjugate, Demonstrates Potent and Selective Activity in HER2-low and T-DM1–resistant Breast and Gastric Cancers
Skidmore, Lillian, Sakamuri, Sukumar, Knudsen, Nick A., Hewet, Amha Gebre, Milutinovic, Snezana, Barkho, Wisam, Biroc, Sandra Lyn, Kirtley, Jessica, Marsden, Robin, Storey, Kristine, Lopez, Ianina, Yu, Wayne, Fang, Shiao-Yan, Yao, Sulan, Gu, Yi, Tian, Feng
Published in Molecular cancer therapeutics (01.09.2020)
Published in Molecular cancer therapeutics (01.09.2020)
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Journal Article
Nonclinical Development of Next-generation Site-specific HER2-targeting Antibody–drug Conjugate (ARX788) for Breast Cancer Treatment
Nagaraja Shastri, Prathap, Zhu, Jingjing, Skidmore, Lillian, Liang, Xuejun, Ji, Yanping, Gu, Yi, Tian, Feng, Yao, Sulan, Xia, Gang
Published in Molecular cancer therapeutics (01.09.2020)
Published in Molecular cancer therapeutics (01.09.2020)
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Journal Article
Glyco-optimization of aminoglycosides: new aminoglycosides as novel anti-infective agents
SULAN YAO, SGARBI, Paulo W. M, ICHIKAWA, Yoshi, SEARS, Pamela, SUCHECK, Steven J, MARBY, Kenneth A, RABUKA, David, O'HARE, Sean M, CHENG, Mayling L, BAIRI, Mrunali, CHANGYONG HU, HWANG, San-Bao, HWANG, Chan-Kou
Published in Bioorganic & medicinal chemistry letters (16.07.2004)
Published in Bioorganic & medicinal chemistry letters (16.07.2004)
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Abstract PS10-57: A randomized, multicenter, open-label phase II/III study of ARX788 vs Lapatinib and Capecitabine in patients with HER2-positive locally advanced or metastatic breast cancer (ZMC-ARX788-211)
Hu, Xichun, Zhang, Jian, Wang, Leiping, Xia, Gang, Ji, Yanping, Xiong, Gaozhun, Liang, Xuejun, Yao, Sulan, Tian, Feng
Published in Cancer research (Chicago, Ill.) (15.02.2021)
Published in Cancer research (Chicago, Ill.) (15.02.2021)
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Journal Article
Safety and unique pharmacokinetic profile of ARX788, a site-specific ADC, in heavily pretreated patients with HER2-overexpresing solid tumors: Results from two phase 1 clinical trials
Hurvitz, Sara A., Park, Haeseong, Frentzas, Sophia, Shannon, Catherine M., Cuff, Katharine, Eek, Richard Wilhelm, Budd, George Thomas, McCartney, Amelia, O'Shaughnessy, Joyce, Lu, Janice M., Zhang, Jian, Ji, Dongmei, Shen, Weina, Li, Matt, Yan, Jinchun, Xia, Gang, Ji, Yanping, Yao, Sulan, Xiong, Gaozhun, Hu, Xichun
Published in Journal of clinical oncology (20.05.2021)
Published in Journal of clinical oncology (20.05.2021)
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Abstract CT211: A phase 1 dose-escalation and dose-expansion study to evaluate the safety, pharmacokinetics, and anti- tumor activity of ARX517 in subjects with advanced solid tumors resistant or refractory to standard therapies (APEX-01 trial, NCT04662580)
Pachynski, Russell K., Nordquist, Luke, Schweizer, Michael T., Shen, John, Adra, Nabil, Bilen, Mehmet A., Reichert, Zachery R., Aggarwal, Rahul, Siddiqui, Bilal A., Li, Matt, Xu, Dong, Huhn, Richard, L'Heureux, Darryl Z., Yan, Jinchun, Buechler, Ying, Yao, Sulan, Simitzi, John, Shi, Wenge, Zhang, Shawn, Tagawa, Scott T.
Published in Cancer research (Chicago, Ill.) (15.06.2022)
Published in Cancer research (Chicago, Ill.) (15.06.2022)
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Journal Article
Study on silica supported CuCrMo nitrobenzene hydrogenation catalysts
Fang, Xiangming, Yao, Sulan, Qing, Zhong, Li, Fengyi
Published in Applied catalysis. A, General (01.11.1997)
Published in Applied catalysis. A, General (01.11.1997)
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Journal Article
Catalytic Enantioselective Aza Diels-Alder Reactions of Imino Dienophiles
Yao, Sulan, Johannsen, Mogens, Hazell, Rita G., Jørgensen, Karl Anker
Published in Angewandte Chemie (International ed.) (04.12.1998)
Published in Angewandte Chemie (International ed.) (04.12.1998)
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Journal Article
Catalytic Approach for the Formation of Optically Active Allyl α-Amino Acids by Addition of Allylic Metal Compounds to α-Imino Esters
Fang, Xiangming, Johannsen, Mogens, Yao, Sulan, Gathergood, Nicholas, Hazell, Rita G, Jørgensen, Karl Anker
Published in Journal of organic chemistry (25.06.1999)
Published in Journal of organic chemistry (25.06.1999)
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Journal Article
An efficient entry to new sugar modified ketolide antibiotics
Romero, Alex, Liang, Chang-Hsing, Chiu, Yu-Hung, Yao, Sulan, Duffield, Jonathan, Sucheck, Steven J., Marby, Ken, Rabuka, David, Leung, Po Yee, Shue, Youe-Kong, Ichikawa, Yoshi, Hwang, Chan-Kou
Published in Tetrahedron letters (28.02.2005)
Published in Tetrahedron letters (28.02.2005)
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