Atropisomeric 4‑Phenyl‑4H‑1,2,4-triazoles as Selective Glycine Transporter 1 Inhibitors
Sugane, Takashi, Tobe, Takahiko, Hamaguchi, Wataru, Shimada, Itsuro, Maeno, Kyoichi, Miyata, Junji, Suzuki, Takeshi, Kimizuka, Tetsuya, Sakamoto, Shuichi, Tsukamoto, Shin-ichi
Published in Journal of medicinal chemistry (25.07.2013)
Published in Journal of medicinal chemistry (25.07.2013)
Get full text
Journal Article
Consequence of Hapten Stereochemistry: An Efficacious Methamphetamine Vaccine
Olson, Margaret E, Sugane, Takashi, Zhou, Bin, Janda, Kim D
Published in Journal of the American Chemical Society (11.09.2019)
Published in Journal of the American Chemical Society (11.09.2019)
Get full text
Journal Article
Catch and Anchor Approach To Combat Both Toxicity and Longevity of Botulinum Toxin A
Lin, Lucy, Olson, Margaret E, Sugane, Takashi, Turner, Lewis D, Tararina, Margarita A, Nielsen, Alexander L, Kurbanov, Elbek K, Pellett, Sabine, Johnson, Eric A, Cohen, Seth M, Allen, Karen N, Janda, Kim D
Published in Journal of medicinal chemistry (08.10.2020)
Published in Journal of medicinal chemistry (08.10.2020)
Get full text
Journal Article
Covalent inhibition of botulinum neurotoxin A – Exploration of warhead reactivity and function using a bifunctional approach
Turner, Lewis D., Nielsen, Alexander L., Lin, Lucy, Pellett, Sabine, Sugane, Takashi, Olson, Margaret E., Janda, Kim D.
Published in Toxicon (Oxford) (01.01.2021)
Published in Toxicon (Oxford) (01.01.2021)
Get full text
Journal Article
Atropisomeric 4-Phenyl-4 H -1,2,4-triazoles as Selective Glycine Transporter 1 Inhibitors
Sugane, Takashi, Tobe, Takahiko, Hamaguchi, Wataru, Shimada, Itsuro, Maeno, Kyoichi, Miyata, Junji, Suzuki, Takeshi, Kimizuka, Tetsuya, Sakamoto, Shuichi, Tsukamoto, Shin-ichi
Published in Journal of medicinal chemistry (25.07.2013)
Published in Journal of medicinal chemistry (25.07.2013)
Get full text
Journal Article
Irreversible inhibition of BoNT/A protease: proximity-driven reactivity contingent upon a bifunctional approach
Turner, Lewis D, Nielsen, Alexander L, Lin, Lucy, Pellett, Sabine, Sugane, Takashi, Olson, Margaret E, Johnson, Eric A, Janda, Kim D
Published in MedChemComm (23.06.2021)
Published in MedChemComm (23.06.2021)
Get full text
Journal Article
Synthesis and Biological Evaluation of 3-Biphenyl-4-yl-4-phenyl-4 H -1,2,4-triazoles as Novel Glycine Transporter 1 Inhibitors
Sugane, Takashi, Tobe, Takahiko, Hamaguchi, Wataru, Shimada, Itsuro, Maeno, Kyoichi, Miyata, Junji, Suzuki, Takeshi, Kimizuka, Tetsuya, Kohara, Atsuyuki, Morita, Takuma, Doihara, Hitoshi, Saita, Kyouko, Aota, Masaki, Furutani, Masako, Shimada, Yoshiaki, Hamada, Noritaka, Sakamoto, Shuichi, Tsukamoto, Shin-ichi
Published in Journal of medicinal chemistry (13.01.2011)
Published in Journal of medicinal chemistry (13.01.2011)
Get full text
Journal Article
Synthesis and Biological Evaluation of 3-Biphenyl-4-yl-4-phenyl-4H-1,2,4-triazoles as Novel Glycine Transporter 1 Inhibitors
Sugane, Takashi, Tobe, Takahiko, Hamaguchi, Wataru, Shimada, Itsuro, Maeno, Kyoichi, Miyata, Junji, Suzuki, Takeshi, Kimizuka, Tetsuya, Kohara, Atsuyuki, Morita, Takuma, Doihara, Hitoshi, Saita, Kyouko, Aota, Masaki, Furutani, Masako, Shimada, Yoshiaki, Hamada, Noritaka, Sakamoto, Shuichi, Tsukamoto, Shin-ichi
Published in Journal of medicinal chemistry (13.01.2011)
Published in Journal of medicinal chemistry (13.01.2011)
Get full text
Journal Article
PIPERAZINE DERIVATIVE
MORITOMO, Hiroyuki, SUGANE, Takashi, YAMASHITA, Daisuke, HOSOGAI, Naomi, ASAI, Norio
Year of Publication 25.01.2018
Get full text
Year of Publication 25.01.2018
Patent
A versatile and efficient method for the synthesis of benz[a]azulenic enones starting from readily available o-(2-furyl)cycloheptatrienylbenzenes
Sasabe, M, Houda, Y, Takagi, H, Sugane, T, Bo, Yamamura, K
Published in Perkin 1 : an international journal of organic and bio-organic chemistry (01.01.2000)
Published in Perkin 1 : an international journal of organic and bio-organic chemistry (01.01.2000)
Get full text
Journal Article
Practical and efficient synthesis of the (R)-atropisomer of a 4-phenyl 1,2,4-triazole derivative as a selective GlyT1 inhibitor
Sugane, Takashi, Hamada, Noritaka, Tobe, Takahiko, Hamaguchi, Wataru, Shimada, Itsuro, Maeno, Kyoichi, Miyata, Junji, Suzuki, Takeshi, Kimizuka, Tetsuya, Sakamoto, Shuichi, Tsukamoto, Shin-ichi
Published in Tetrahedron: asymmetry (15.12.2012)
Published in Tetrahedron: asymmetry (15.12.2012)
Get full text
Journal Article
Synthesis and biological evaluation of (4H-1,2,4-triazol-4-yl)isoquinoline derivatives as selective glycine transporter 1 inhibitors
Sugane, Takashi, Tobe, Takahiko, Hamaguchi, Wataru, Shimada, Itsuro, Maeno, Kyoichi, Miyata, Junji, Suzuki, Takeshi, Kimizuka, Tetsuya, Morita, Takuma, Sakamoto, Shuichi, Tsukamoto, Shin-ichi
Published in Bioorganic & medicinal chemistry (01.01.2012)
Published in Bioorganic & medicinal chemistry (01.01.2012)
Get full text
Journal Article
피페라진 유도체
HOSOGAI NAOMI, TANABE DAISUKE, MIHARA HISASHI, MORITOMO HIROYUKI, YAMASHITA DAISUKE, YONETOKU YASUHIRO, OSODA KAZUHIKO, ASAI NORIO, SUGANE TAKASHI, MAENO KYOICHI, SUGASAWA KEIZO, SHIMIZU TAKAFUMI, MAKINO TAKUYA
Year of Publication 30.03.2018
Get full text
Year of Publication 30.03.2018
Patent
PIPERAZINE DERIVATIVE
SUGASAWA, Keizo, MAENO, Kyoichi, MIHARA, Hisashi, MAKINO, Takuya, OSODA, Kazuhiko, MORITOMO, Hiroyuki, HOSOGAI, Naomi, ASAI, Norio, YONETOKU, Yasuhiro, SHIMIZU, Takafumi, SUGANE, Takashi, YAMASHITA, Daisuke, TANABE, Daisuke
Year of Publication 09.02.2017
Get full text
Year of Publication 09.02.2017
Patent
CARBAMATE COMPOUND OR SALT THEREOF
SOMEYA AKIYOSHI, MUNAKATA RYOSUKE, SUGANE TAKASHI, AOKI SATOSHI, HIGAKI MASAHIDE, ISHII TAKAHIRO
Year of Publication 11.08.2011
Get full text
Year of Publication 11.08.2011
Patent
ANTAGONIST FOR MUTATED ANDROGEN RECEPTOR
FURUTANI TAKASHI, TANIGUCHI NOBUAKI, SUGANE TAKASHI, YAMADA TOMOHIRO, WATANABE KAZUSHI, HIRANO MASAAKI, KONAGAI SATOSHI, TAKEDA MASAYOSHI, KONDOH YUTAKA, KAKEFUDA AKIO, IDEYAMA YUKITAKA, KUROMITSU SADAO
Year of Publication 23.12.2013
Get full text
Year of Publication 23.12.2013
Patent
AZOLE COMPOUND
MUNAKATA RYOSUKE, SAMIZU KIYOHIRO, SUGANE TAKASHI, AOKI SATOSHI, KAWANO NORIYUKI, ISHII TAKAHIRO, OKA HIROMASA
Year of Publication 14.04.2011
Get full text
Year of Publication 14.04.2011
Patent
CARBAMATE COMPOUND OR SALT THEREOF
AOKI, SATOSHI, HIGAKI, MASAHIDE, SOMEYA, AKIYOSHI, MUNAKATA, RYOSUKE, ISHII, TAKAHIRO, SUGANE, TAKASHI
Year of Publication 14.05.2010
Get full text
Year of Publication 14.05.2010
Patent
AZOLE COMPOUND
KAWANO, NORIYUKI, SUGANE, TAKASHI, ISHII, TAKAHIRO, AOKI, SATOSHI, MUNAKATA, RYOSUKE, SAMIZU, KIYOHIRO, OKA, HIROMASA
Year of Publication 21.01.2010
Get full text
Year of Publication 21.01.2010
Patent
ANTAGONIST FOR MUTATED ANDROGEN RECEPTOR
KAKEFUDA, AKIO, WATANABE, KAZUSHI, HIRANO, MASAAKI, KONDOH, YUTAKA, KONAGAI, SATOSHI, TANIGUCHI, NOBUAKI, IDEYAMA, YUKITAKA, FURUTANI, TAKASHI, KUROMITSU, SADAO, TAKEDA, MASAYOSHI, YAMADA, TOMOHIRO, SUGANE, TAKASHI
Year of Publication 26.04.2012
Get full text
Year of Publication 26.04.2012
Patent