BCX-1812 (RWJ-270201): Discovery of a Novel, Highly Potent, Orally Active, and Selective Influenza Neuraminidase Inhibitor through Structure-Based Drug Design
Babu, Y. Sudhakar, Chand, Pooran, Bantia, Shanta, Kotian, Pravin, Dehghani, Ali, El-Kattan, Yahya, Lin, Tsu-Hsing, Hutchison, Tracy L, Elliott, Arthur J, Parker, Cynthia D, Ananth, Sandya L, Horn, LaShun L, Laver, Graeme W, Montgomery, John A
Published in Journal of medicinal chemistry (21.09.2000)
Published in Journal of medicinal chemistry (21.09.2000)
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Design, parallel synthesis, and crystal structures of biphenyl antithrombotics as selective inhibitors of tissue factor FVIIa complex. Part 1: Exploration of S2 pocket pharmacophores
Kotian, Pravin L., Krishnan, Raman, Rowland, Scott, El-Kattan, Yahya, Saini, Surendra K., Upshaw, Ramanda, Bantia, Shanta, Arnold, Shane, Sudhakar Babu, Y., Chand, Pooran
Published in Bioorganic & medicinal chemistry (01.06.2009)
Published in Bioorganic & medicinal chemistry (01.06.2009)
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Journal Article
Syntheses and Neuraminidase Inhibitory Activity of Multisubstituted Cyclopentane Amide Derivatives
Chand, Pooran, Babu, Y. Sudhakar, Bantia, Shanta, Rowland, Scott, Dehghani, Ali, Kotian, Pravin L, Hutchison, Tracy L, Ali, Shoukath, Brouillette, Wayne, El-Kattan, Yahya, Lin, Tsu-Hsing
Published in Journal of medicinal chemistry (08.04.2004)
Published in Journal of medicinal chemistry (08.04.2004)
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Journal Article
Intramuscularly administered neuraminidase inhibitor peramivir is effective against lethal H5N1 influenza virus in mice
Boltz, David A., Ilyushina, Natalia A., Arnold, C. Shane, Babu, Y. Sudhakar, Webster, Robert G., Govorkova, Elena A.
Published in Antiviral research (01.11.2008)
Published in Antiviral research (01.11.2008)
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Journal Article
Application of Crystallographic and Modeling Methods in the Design of Purine Nucleoside Phosphorylase Inhibitors
RZMOVL, S. E, SUDHAKAR BABU, Y, BUGG, C. E, ERION, M. D, GUIDA, W. C, MONTGOMERY, J. A, SECRIST, J. A
Published in Proceedings of the National Academy of Sciences - PNAS (15.12.1991)
Published in Proceedings of the National Academy of Sciences - PNAS (15.12.1991)
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Journal Article
Systematic Structure-Based Design and Stereoselective Synthesis of Novel Multisubstituted Cyclopentane Derivatives with Potent Antiinfluenza Activity
Chand, Pooran, Kotian, Pravin L, Dehghani, Ali, El-Kattan, Yahya, Lin, Tsu-Hsing, Hutchison, Tracy L, Babu, Y. Sudhakar, Bantia, Shanta, Elliott, Arthur J, Montgomery, John A
Published in Journal of medicinal chemistry (06.12.2001)
Published in Journal of medicinal chemistry (06.12.2001)
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Journal Article
Structure of calmodulin refined at 2.2 Å resolution
Babu, Y.Sudhakar, Bugg, Charles E., Cook, William J.
Published in Journal of molecular biology (05.11.1988)
Published in Journal of molecular biology (05.11.1988)
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Journal Article
The antithrombotic and anti-inflammatory effects of BCX-3607, a small molecule tissue factor/factor VIIa inhibitor
Arnold, C. Shane, Parker, Cynthia, Upshaw, Ramanda, Prydz, Hans, Chand, Pooran, Kotian, Pravin, Bantia, Shanta, Babu, Y. Sudhakar
Published in Thrombosis research (2006)
Published in Thrombosis research (2006)
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Journal Article
Three-dimensional structure of calmodulin
Babu, Y S, Sack, J S, Greenhough, T J, Bugg, C E, Means, A R, Cook, W J
Published in Nature (London) (02.05.1985)
Published in Nature (London) (02.05.1985)
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Journal Article
Structure-based design of inhibitors of purine nucleoside phosphorylase. 1. 9-(Arylmethyl) derivatives of 9-deazaguanine
Montgomery, John A., Niwas, Shri, Rose, Jerry D., Secrist, John A., Babu, Y. Sudhakar, Bugg, Charles E., Erion, Mark D., Guida, Wayne C., Ealick, Steven E.
Published in Journal of medicinal chemistry (1993)
Published in Journal of medicinal chemistry (1993)
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Journal Article
Structure-based design of inhibitors of purine nucleoside phosphorylase. 2. 9-Alicyclic and 9-heteroalicyclic derivatives of 9-deazaguanine
Secrist, John A, Niwas, Shri, Rose, Jerry D, Babu, Y. Sudhakar, Bugg, Charles E, Erion, Mark D, Guida, Wayne C, Ealick, Steven E, Montgomery, John A
Published in Journal of medicinal chemistry (01.06.1993)
Published in Journal of medicinal chemistry (01.06.1993)
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Journal Article
Three-dimensional structure of a sarcoplasmic calcium-binding protein from Nereis diversicolor
Cook, W J, Ealick, S E, Babu, Y S, Cox, J A, Vijay-Kumar, S
Published in The Journal of biological chemistry (05.01.1991)
Published in The Journal of biological chemistry (05.01.1991)
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Journal Article
Structure-based design of inhibitors of purine nucleoside phosphorylase. 3. 9-Arylmethyl derivatives of 9-deazaguanine substituted on the arylmethyl group
Erion, Mark D, Niwas, Shri, Rose, Jerry D, Ananthan, Subramaniam, Allen, Mark, Secrist, John A, Babu, Y. Sudhakar, Bugg, Charles E, Guida, Wayne C
Published in Journal of medicinal chemistry (01.11.1993)
Published in Journal of medicinal chemistry (01.11.1993)
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Journal Article
Corrigendum to “Design, parallel synthesis, and crystal structures of biphenyl antithrombotics as selective inhibitors of tissue factor FVIIa complex. Part 1: Exploration of S2 pocket pharmacophores” [Bioorg. Med. Chem. 17 (2009) 3934]
Kotian, Pravin L., Krishnan, Raman, Rowland, Scott, El-Kattan, Yahya, Saini, Surendra K., Upshaw, Ramanda, Bantia, Shanta, Arnold, Shane, Babu, Y. Sudhakar, Chand, Pooran
Published in Bioorganic & medicinal chemistry (2010)
Published in Bioorganic & medicinal chemistry (2010)
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Journal Article
Purification, crystallization and preliminary crystallographic analysis of porcine aldose reductase
El-Kabbani, Ossama, Narayana, Sthanam V.L., Babu, Y.Sudhakar, Moore, Karen M., Flynn, T.G., Petrash, J.M., Westbrook, Edwin M., DeLucas, Lawrence J., Bugg, Charles E.
Published in Journal of molecular biology (20.04.1991)
Published in Journal of molecular biology (20.04.1991)
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Journal Article
Intramuscular Administration of Neuraminidase Inhibitor Peramivir Promotes Survival Against Lethal H5N1 Influenza Infection in Mice
Boltz, David A., Ilyushina, Natalia A., Arnold, C. Shane, Babu, Y. Sudhakar, Webster, Robert G., Govorkova, Elena A.
Published in Antiviral research (01.06.2007)
Published in Antiviral research (01.06.2007)
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Journal Article
Three-dimensional structure of human erythrocytic purine nucleoside phosphorylase at 3.2 A resolution
S E Ealick, S A Rule, D C Carter, T J Greenhough, Y S Babu, W J Cook, J Habash, J R Helliwell, J D Stoeckler, R E Parks, Jr
Published in The Journal of biological chemistry (25.01.1990)
Published in The Journal of biological chemistry (25.01.1990)
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