1,4-Dihydroindeno[1,2- c]pyrazoles as potent checkpoint kinase 1 inhibitors: Extended exploration on phenyl ring substitutions and preliminary ADME/PK studies
Tong, Yunsong, Claiborne, Akiyo, Pyzytulinska, Magdalena, Tao, Zhi-Fu, Stewart, Kent D., Kovar, Peter, Chen, Zehan, Credo, Robert B., Guan, Ran, Merta, Philip J., Zhang, Haiying, Bouska, Jennifer, Everitt, Elizabeth A., Murry, Bernard P., Hickman, Dean, Stratton, Tim J., Wu, Jian, Rosenberg, Saul H., Sham, Hing L., Sowin, Thomas J., Lin, Nan-horng
Published in Bioorganic & medicinal chemistry letters (01.07.2007)
Published in Bioorganic & medicinal chemistry letters (01.07.2007)
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Journal Article
L,4 -dihydroindeno[1,2 -c ]pyrazoles as potent checkpoint kinase 1 inhibitors : Extended exploration on phenyl ring substitutions and preliminary ADME/PK studies
YUNSONG TONG, CLAIBORNE, Akiyo, HAIYING ZHANG, BOUSKA, Jennifer, EVERITT, Elizabeth A, MURRY, Bernard P, HICKMAN, Dean, STRATTON, Tim J, JIAN WU, ROSENBERG, Saul H, SHAM, Hing L, SOWIN, Thomas J, PYZYTULINSKA, Magdalena, LIN, Nan-Horng, TAO, Zhi-Fu, STEWART, Kent D, KOVAR, Peter, ZEHAN CHEN, CREDO, Robert B, RAN GUAN, MERTA, Philip J
Published in Bioorganic & medicinal chemistry letters (2007)
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Published in Bioorganic & medicinal chemistry letters (2007)
Journal Article