Novel 6-aminofuro[3,2-c]pyridines as potent, orally efficacious inhibitors of cMET and RON kinases
Steinig, Arno G., Li, An-Hu, Wang, Jing, Chen, Xin, Dong, Hanqing, Ferraro, Caterina, Jin, Meizhong, Kadalbajoo, Mridula, Kleinberg, Andrew, Stolz, Kathryn M., Tavares-Greco, Paula A., Wang, Ti, Albertella, Mark R., Peng, Yue, Crew, Linda, Kahler, Jennifer, Kan, Julie, Schulz, Ryan, Cooke, Andy, Bittner, Mark, Turton, Roy W., Franklin, Maryland, Gokhale, Prafulla, Landfair, Darla, Mantis, Christine, Workman, Jen, Wild, Robert, Pachter, Jonathan, Epstein, David, Mulvihill, Mark J.
Published in Bioorganic & medicinal chemistry letters (01.08.2013)
Published in Bioorganic & medicinal chemistry letters (01.08.2013)
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A highly effective one-pot synthesis of quinolines from o-nitroarylcarbaldehydes
Li, An-Hu, Ahmed, Eilaf, Chen, Xin, Cox, Matthew, Crew, Andrew P., Dong, Han-Qing, Jin, Meizhong, Ma, Lifu, Panicker, Bijoy, Siu, Kam W., Steinig, Arno G., Stolz, Kathryn M., Tavares, Paula A. R., Volk, Brian, Weng, Qinghua, Werner, Doug, Mulvihill, Mark J.
Published in Organic & biomolecular chemistry (01.01.2007)
Published in Organic & biomolecular chemistry (01.01.2007)
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Novel 2-phenylquinolin-7-yl-derived imidazo[1,5- a]pyrazines as potent insulin-like growth factor-I receptor (IGF-IR) inhibitors
Mulvihill, Mark J., Ji, Qun-Sheng, Coate, Heather R., Cooke, Andrew, Dong, Hanqing, Feng, Lixin, Foreman, Kenneth, Rosenfeld-Franklin, Maryland, Honda, Ayako, Mak, Gilda, Mulvihill, Kristen M., Nigro, Anthony I., O’Connor, Matthew, Pirrit, Caroline, Steinig, Arno G., Siu, Kam, Stolz, Kathryn M., Sun, Yingchuan, Tavares, Paula A.R., Yao, Yan, Gibson, Neil W.
Published in Bioorganic & medicinal chemistry (01.02.2008)
Published in Bioorganic & medicinal chemistry (01.02.2008)
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1,3-Disubstituted-imidazo[1,5- a]pyrazines as insulin-like growth-factor-I receptor (IGF-IR) inhibitors
Mulvihill, Mark J., Ji, Qun-Sheng, Werner, Doug, Beck, Patricia, Cesario, Cara, Cooke, Andrew, Cox, Matthew, Crew, Andrew, Dong, Hanqing, Feng, Lixin, Foreman, K.W., Mak, Gilda, Nigro, Anthony, O’Connor, Matthew, Saroglou, Lydia, Stolz, Kathryn M., Sujka, Izabela, Volk, Brian, Weng, Qinghua, Wilkes, Robin
Published in Bioorganic & medicinal chemistry letters (15.02.2007)
Published in Bioorganic & medicinal chemistry letters (15.02.2007)
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Discovery of an Orally Efficacious Imidazo[5,1-f][1,2,4]triazine Dual Inhibitor of IGF-1R and IR
Jin, Meizhong, Gokhale, Prafulla C, Cooke, Andy, Foreman, Kenneth, Buck, Elizabeth, May, Earl W, Feng, Lixin, Bittner, Mark A, Kadalbajoo, Mridula, Landfair, Darla, Siu, Kam W, Stolz, Kathryn M, Werner, Douglas S, Laufer, Radoslaw S, Li, An-Hu, Dong, Hanqing, Steinig, Arno G, Kleinberg, Andrew, Yao, Yan, Pachter, Jonathan A, Wild, Robert, Mulvihill, Mark J
Published in ACS medicinal chemistry letters (09.12.2010)
Published in ACS medicinal chemistry letters (09.12.2010)
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Abstract 3900: Discovery of FQIT: An imidazo[5,1- f ][1,2,4]triazine derived dual IGF-1R/IR inhibitor
Jin, Meizhong, Gokhale, Prafulla, Cooke, Andy, Foreman, Kenneth, Buck, Elizabeth, May, Earl, Feng, Lixing, Bittner, Mark, Kadalbajoo, Mridula, Landfair, Darla, Siu, Kam, Stolz, Kathryn, Werner, Douglas, Laufer, Radoslaw, Li, An-Hu, Dong, Hanqing, Steinig, Arno, Kleinberg, Andrew, Yao, Yan, Pachter, Jonathan, Wild, Robert, Mulvihill, Mark
Published in Cancer research (Chicago, Ill.) (15.04.2012)
Published in Cancer research (Chicago, Ill.) (15.04.2012)
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AMINO PYRIMIDINE ANTICANCER COMPOUNDS
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Year of Publication 12.04.2012
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Year of Publication 12.04.2012
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Abstract 2915: Discovery and characterization of OSI-296, a dual inhibitor of cMET and RON kinases
Steinig, Arno G., Li, An-Hu, Wang, Jing, Kleinberg, Andrew, Dong, Hanqing, Wang, Ti, Gavagan, Kathryn M. Stolz, Jin, Meizhong, Tavares-Greco, Paula, Peng, Yue, Kahler, Jen, Castaldo, Linda, McCormack, Siobhan, Kan, Julie, Albertella, Mark, Cooke, Andy, Turton, Roy, Bittner, Mark, Franklin, Maryland, Landfair, Darla, Gokhale, Prafulla, Wild, Robert, Pachter, Jonathan, Epstein, David, Mulvihill, Mark J.
Published in Cancer research (Chicago, Ill.) (15.04.2012)
Published in Cancer research (Chicago, Ill.) (15.04.2012)
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AMINO PYRIMIDINE ANTICANCER COMPOUNDS
CHILUKURI RAMESH, SHERMAN DAN, LI AN-HU, FOREMAN KENNETH, ZAHLER ROBERT, CHEN XIN, DONG HANQING, VOLK BRIAN, APPARI RAMA DEVI, GUPTA RAMESH C, STOLZ KATHRYN M, FERRARO CATERINA, CREW ANDREW P
Year of Publication 30.03.2018
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Year of Publication 30.03.2018
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AMINO PYRIMIDINE ANTICANCER COMPOUNDS
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Year of Publication 20.12.2017
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Year of Publication 20.12.2017
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Year of Publication 04.08.2015
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Year of Publication 19.03.2013
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AMINO PYRIMIDINE ANTICANCER COMPOUNDS
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Year of Publication 31.10.2012
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Amino pyrimidine anticancer compounds
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Year of Publication 03.11.2011
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AMINO PYRIMIDINE ANTICANCER COMPOUNDS
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Year of Publication 09.06.2011
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AMINO PYRIMIDINE ANTICANCER COMPOUNDS
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Year of Publication 21.04.2011
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Year of Publication 21.04.2011
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