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El‐Kouhen, O, Lehto, S G, Pan, J B, Chang, R, Baker, S J, Zhong, C, Hollingsworth, P R, Mikusa, J P, Cronin, E A, Chu, K L, McGaraughty, S P, Uchic, M E, Miller, L N, Rodell, N M, Patel, M, Bhatia, P, Mezler, M, Kolasa, T, Zheng, G Z, Fox, G B, Stewart, A O, Decker, M W, Moreland, R B, Brioni, J D, Honore, P
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Published in British journal of pharmacology (01.11.2006)
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Discovery of 4-Amino-5-(3-bromophenyl)-7-(6-morpholino-pyridin- 3-yl)pyrido[2,3-d]pyrimidine, an Orally Active, Non-Nucleoside Adenosine Kinase Inhibitor
Lee, Chih-Hung, Jiang, Meiqun, Cowart, Marlon, Gfesser, Greg, Perner, Richard, Kim, Ki Hwan, Gu, Yu Gui, Williams, Michael, Jarvis, Michael F, Kowaluk, Elizabeth A, Stewart, Andrew O, Bhagwat, Shripad S
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Published in Journal of medicinal chemistry (21.06.2001)
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Symmetrical Bis(heteroarylmethoxyphenyl)alkylcarboxylic Acids as Inhibitors of Leukotriene Biosynthesis
Kolasa, Teodozyj, Gunn, David E, Bhatia, Pramila, Basha, Anwer, Craig, Richard A, Stewart, Andrew O, Bouska, Jennifer B, Harris, Richard R, Hulkower, Keren I, Malo, Peter E, Bell, Randy L, Carter, George W, Brooks, Clint D. W
Published in Journal of medicinal chemistry (24.08.2000)
Published in Journal of medicinal chemistry (24.08.2000)
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Selective Inhibition of ICAM-1 and E-Selectin Expression in Human Endothelial Cells. 2. Aryl Modifications of 4-(Aryloxy)thieno[2,3-c]pyridines with Fine-Tuning at C-2 Carbamides
Zhu, Gui-Dong, Arendsen, David L, Gunawardana, Indrani W, Boyd, Steven A, Stewart, Andrew O, Fry, Dennis G, Cool, Barbara L, Kifle, Lemma, Schaefer, Verlyn, Meuth, Joseph, Marsh, Kennan C, Kempf-Grote, Anita J, Kilgannon, Patrick, Gallatin, W. Michael, Okasinski, Gregory F
Published in Journal of medicinal chemistry (11.10.2001)
Published in Journal of medicinal chemistry (11.10.2001)
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Heteroarylmethoxyphenylalkoxyiminoalkylcarboxylic Acids as Leukotriene Biosynthesis Inhibitors
Kolasa, Teodozyj, Gunn, David E, Bhatia, Pramila, Woods, Keith W, Gane, Todd, Stewart, Andrew O, Bouska, Jennifer B, Harris, Richard R, Hulkower, Keren I, Malo, Peter E, Bell, Randy L, Carter, George W, Brooks, Clint D. W
Published in Journal of medicinal chemistry (24.02.2000)
Published in Journal of medicinal chemistry (24.02.2000)
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Optimization of the potency and duration of action of N-hydroxyurea 5-lipoxygenase inhibitors
Bell, R L, Bouska, J B, Malo, P E, Lanni, C, Harris, R R, Otis, E R, Stewart, A O, Brooks, D W, Carter, G W
Published in The Journal of pharmacology and experimental therapeutics (01.02.1995)
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Published in The Journal of pharmacology and experimental therapeutics (01.02.1995)
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(R)-(+)-N-[3-[5-[(4-FLUOROPHENYL)METHYL]-2-THIENYL]-1-METHYL-2-PROPYNYL]-N-HYDROXYUREA (ABT-761), A 2ND-GENERATION 5-LIPOXYGENASE INHIBITOR
BROOKS, CDW, STEWART, AO, BASHA, A, BHATIA, P, RATAJCZYK, JD, MARTIN, JG, CRAIG, RA, KOLASA, T, BOUSKA, JB, LANNI, C, HARRIS, RR, MALO, PE, CARTER, GW, BELL, RL
Published in Journal of medicinal chemistry (24.11.1995)
Published in Journal of medicinal chemistry (24.11.1995)
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Hydroxamic acid inhibitors of 5-lipoxygenase: quantitative structure-activity relationships
Summers, James B, Kim, Ki H, Mazdiyasni, Hormoz, Holms, James H, Ratajczyk, James D, Stewart, Andrew O, Dyer, Richard D, Carter, George W
Published in Journal of medicinal chemistry (01.03.1990)
Published in Journal of medicinal chemistry (01.03.1990)
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Design of inhibitors of leukotriene biosynthesis and their therapeutic potential
Brooks, C. D. W., Stewart, A. O., Kolasa, Teodozyj, Basha, A., Bhatia, Pramila, Ratajczyk, J. D., Craig, R. A., Gunn, David, Harris, R. R., Bouska, J. B., Malo, P. E., Bell, R. L., Carter, G. W.
Published in Pure and applied chemistry (28.02.1998)
Published in Pure and applied chemistry (28.02.1998)
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Preclinical and clinical activity of zileuton and A-78773
Bell, R L, Lanni, C, Malo, P E, Brooks, D W, Stewart, A O, Hansen, R, Rubin, P, Carter, G W
Published in Annals of the New York Academy of Sciences (01.11.1993)
Published in Annals of the New York Academy of Sciences (01.11.1993)
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Structure-activity analysis of a class of orally active hydroxamic acid inhibitors of leukotriene biosynthesis
Summers, James B, Gunn, Bruce P, Martin, Jonathan G, Martin, Michael B, Mazdiyasni, Hormoz, Stewart, Andrew O, Young, Patrick R, Bouska, Jennifer B, Goetze, Andrew M
Published in Journal of medicinal chemistry (01.10.1988)
Published in Journal of medicinal chemistry (01.10.1988)
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Orally active hydroxamic acid inhibitors of leukotriene biosynthesis
Summers, James B, Gunn, Bruce P, Martin, Jonathan G, Mazdiyasni, Hormoz, Stewart, Andrew O, Young, Patrick R, Goetze, Andrew M, Bouska, Jennifer B, Dyer, Richard D
Published in Journal of medicinal chemistry (01.01.1988)
Published in Journal of medicinal chemistry (01.01.1988)
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Second generation leukotriene biosynthesis inhibitors
Basha, A., Brooks, D. W., Stewart, A. O., Bell, R. L., Carter, G. W.
Published in Pure and applied chemistry (01.01.1994)
Published in Pure and applied chemistry (01.01.1994)
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Structure–activity studies of 5-substituted pyridopyrimidines as adenosine kinase inhibitors
Cowart, Marlon, Lee, Chih-Hung, Gfesser, Gregory A., Bayburt, Erol K., Bhagwat, Shripad S., Stewart, Andrew O., Yu, Haixia, Kohlhaas, Kathy L., McGaraughty, Steve, Wismer, Carol T., Mikusa, Joseph, Zhu, Chang, Alexander, Karen M., Jarvis, Michael F., Kowaluk, Elizabeth A.
Published in Bioorganic & medicinal chemistry letters (08.01.2001)
Published in Bioorganic & medicinal chemistry letters (08.01.2001)
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Pyridopyrimidine analogues as novel adenosine kinase inhibitors
Zheng, Guo Zhu, Lee, Chih-Hung, Pratt, John K, Perner, Richard J, Jiang, Mei Qun, Gomtsyan, Arthur, Matulenko, Mark A, Mao, Yui, Koenig, John R, Kim, Ki H, Muchmore, Steve, Yu, Haixia, Kohlhaas, Kathy, Alexander, Karen M, McGaraughty, Steve, Chu, Katharine L, Wismer, Carol T, Mikusa, Joseph, Jarvis, Michael F, Marsh, Kennan, Kowaluk, Elizabeth A, Bhagwat, Shripad S, Stewart, Andrew O
Published in Bioorganic & medicinal chemistry letters (20.08.2001)
Published in Bioorganic & medicinal chemistry letters (20.08.2001)
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Structure−Activity Relationships of N-Hydroxyurea 5-Lipoxygenase Inhibitors
Stewart, Andrew O, Bhatia, Pramila A, Martin, Jonathan G, Summers, James B, Rodriques, Karen E, Martin, Michael B, Holms, James H, Moore, Jimmie L, Craig, Richard A, Kolasa, Teodozyj, Ratajczyk, James D, Mazdiyasni, Hormoz, Kerdesky, Francis A. J, DeNinno, Shari L, Maki, Robert G, Bouska, Jennifer B, Young, Patrick R, Lanni, Carmine, Bell, Randy L, Carter, George W, Brooks, Clint D. W
Published in Journal of medicinal chemistry (20.06.1997)
Published in Journal of medicinal chemistry (20.06.1997)
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C-Glycosidation of pyridyl thioglycosides
Stewart, Andrew O, Williams, Robert M
Published in Journal of the American Chemical Society (01.07.1985)
Published in Journal of the American Chemical Society (01.07.1985)
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