Structure of the full-length glucagon class B G-protein-coupled receptor
Zhang, Haonan, Qiao, Anna, Yang, Dehua, Yang, Linlin, Dai, Antao, de Graaf, Chris, Reedtz-Runge, Steffen, Dharmarajan, Venkatasubramanian, Zhang, Hui, Han, Gye Won, Grant, Thomas D., Sierra, Raymond G., Weierstall, Uwe, Nelson, Garrett, Liu, Wei, Wu, Yanhong, Ma, Limin, Cai, Xiaoqing, Lin, Guangyao, Wu, Xiaoai, Geng, Zhi, Dong, Yuhui, Song, Gaojie, Griffin, Patrick R., Lau, Jesper, Cherezov, Vadim, Yang, Huaiyu, Hanson, Michael A., Stevens, Raymond C., Zhao, Qiang, Jiang, Hualiang, Wang, Ming-Wei, Wu, Beili
Published in Nature (London) (08.06.2017)
Published in Nature (London) (08.06.2017)
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Journal Article
High-Resolution Crystal Structure of an Engineered Human β₂-Adrenergic G Protein-Coupled Receptor
Cherezov, Vadim, Rosenbaum, Daniel M, Hanson, Michael A, Rasmussen, Søren G.F, Thian, Foon Sun, Kobilka, Tong Sun, Choi, Hee-Jung, Kuhn, Peter, Weis, William I, Kobilka, Brian K, Stevens, Raymond C
Published in Science (American Association for the Advancement of Science) (23.11.2007)
Published in Science (American Association for the Advancement of Science) (23.11.2007)
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Journal Article
Structural basis of ligand binding modes at the neuropeptide Y Y1 receptor
Yang, Zhenlin, Han, Shuo, Keller, Max, Kaiser, Anette, Bender, Brian J., Bosse, Mathias, Burkert, Kerstin, Kögler, Lisa M., Wifling, David, Bernhardt, Guenther, Plank, Nicole, Littmann, Timo, Schmidt, Peter, Yi, Cuiying, Li, Beibei, Ye, Sheng, Zhang, Rongguang, Xu, Bo, Larhammar, Dan, Stevens, Raymond C., Huster, Daniel, Meiler, Jens, Zhao, Qiang, Beck-Sickinger, Annette G., Buschauer, Armin, Wu, Beili
Published in Nature (London) (01.04.2018)
Published in Nature (London) (01.04.2018)
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Journal Article
An electrostatic mechanism for Ca2+-mediated regulation of gap junction channels
Bennett, Brad C., Purdy, Michael D., Baker, Kent A., Acharya, Chayan, McIntire, William E., Stevens, Raymond C., Zhang, Qinghai, Harris, Andrew L., Abagyan, Ruben, Yeager, Mark
Published in Nature communications (12.01.2016)
Published in Nature communications (12.01.2016)
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Journal Article
Structural Basis for Apelin Control of the Human Apelin Receptor
Ma, Yingli, Yue, Yang, Ma, Yanbin, Zhang, Qing, Zhou, Qingtong, Song, Yunpeng, Shen, Yuqing, Li, Xun, Ma, Xiaochuan, Li, Chao, Hanson, Michael A., Han, Gye Won, Sickmier, E. Allen, Swaminath, Gayathri, Zhao, Suwen, Stevens, Raymond C., Hu, Liaoyuan A., Zhong, Wenge, Zhang, Mingqiang, Xu, Fei
Published in Structure (London) (06.06.2017)
Published in Structure (London) (06.06.2017)
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Journal Article
Computational design of thermostabilizing point mutations for G protein-coupled receptors
Popov, Petr, Peng, Yao, Shen, Ling, Stevens, Raymond C, Cherezov, Vadim, Liu, Zhi-Jie, Katritch, Vsevolod
Published in eLife (21.06.2018)
Published in eLife (21.06.2018)
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Journal Article
NMR structure and dynamics of the agonist dynorphin peptide bound to the human kappa opioid receptor
O’Connor, Casey, White, Kate L., Doncescu, Nathalie, Didenko, Tatiana, Roth, Bryan L., Czaplicki, Georges, Stevens, Raymond C., Wüthrich, Kurt, Milon, Alain
Published in Proceedings of the National Academy of Sciences - PNAS (22.09.2015)
Published in Proceedings of the National Academy of Sciences - PNAS (22.09.2015)
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Journal Article
De Novo Structural Pattern Mining in Cellular Electron Cryotomograms
Xu, Min, Singla, Jitin, Tocheva, Elitza I., Chang, Yi-Wei, Stevens, Raymond C., Jensen, Grant J., Alber, Frank
Published in Structure (London) (02.04.2019)
Published in Structure (London) (02.04.2019)
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Journal Article
Single-molecule view of basal activity and activation mechanisms of the G protein-coupled receptor β₂AR
Lamichhane, Rajan, Liu, Jeffrey J., Pljevaljcic, Goran, White, Kate L., van der Schans, Edwin, Katritch, Vsevolod, Stevens, Raymond C., Wüthrich, Kurt, Millar, David P.
Published in Proceedings of the National Academy of Sciences - PNAS (17.11.2015)
Published in Proceedings of the National Academy of Sciences - PNAS (17.11.2015)
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Journal Article
Nucleotides Acting at P2Y Receptors: Connecting Structure and Function
Jacobson, Kenneth A, Paoletta, Silvia, Katritch, Vsevolod, Wu, Beili, Gao, Zhan-Guo, Zhao, Qiang, Stevens, Raymond C, Kiselev, Evgeny
Published in Molecular pharmacology (01.08.2015)
Published in Molecular pharmacology (01.08.2015)
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Journal Article
Constitutive phospholipid scramblase activity of a G protein-coupled receptor
Goren, Michael A., Morizumi, Takefumi, Menon, Indu, Joseph, Jeremiah S., Dittman, Jeremy S., Cherezov, Vadim, Stevens, Raymond C., Ernst, Oliver P., Menon, Anant K.
Published in Nature communications (08.10.2014)
Published in Nature communications (08.10.2014)
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Journal Article
Structural basis for signal recognition and transduction by platelet-activating-factor receptor
Cao, Can, Tan, Qiuxiang, Xu, Chanjuan, He, Lingli, Yang, Linlin, Zhou, Ye, Zhou, Yiwei, Qiao, Anna, Lu, Minmin, Yi, Cuiying, Han, Gye Won, Wang, Xianping, Li, Xuemei, Yang, Huaiyu, Rao, Zihe, Jiang, Hualiang, Zhao, Yongfang, Liu, Jianfeng, Stevens, Raymond C., Zhao, Qiang, Zhang, Xuejun C., Wu, Beili
Published in Nature structural & molecular biology (01.06.2018)
Published in Nature structural & molecular biology (01.06.2018)
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Journal Article
Crystal structure of the Frizzled 4 receptor in a ligand-free state
Yang, Shifan, Wu, Yiran, Xu, Ting-Hai, de Waal, Parker W., He, Yuanzheng, Pu, Mengchen, Chen, Yuxiang, DeBruine, Zachary J., Zhang, Bingjie, Zaidi, Saheem A., Popov, Petr, Guo, Yu, Han, Gye Won, Lu, Yang, Suino-Powell, Kelly, Dong, Shaowei, Harikumar, Kaleeckal G., Miller, Laurence J., Katritch, Vsevolod, Xu, H. Eric, Shui, Wenqing, Stevens, Raymond C., Melcher, Karsten, Zhao, Suwen, Xu, Fei
Published in Nature (London) (01.08.2018)
Published in Nature (London) (01.08.2018)
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Journal Article
Crystal structure of a multi-domain human smoothened receptor in complex with a super stabilizing ligand
Zhang, Xianjun, Zhao, Fei, Wu, Yiran, Yang, Jun, Han, Gye Won, Zhao, Suwen, Ishchenko, Andrii, Ye, Lintao, Lin, Xi, Ding, Kang, Dharmarajan, Venkatasubramanian, Griffin, Patrick R., Gati, Cornelius, Nelson, Garrett, Hunter, Mark S., Hanson, Michael A., Cherezov, Vadim, Stevens, Raymond C., Tan, Wenfu, Tao, Houchao, Xu, Fei
Published in Nature communications (17.05.2017)
Published in Nature communications (17.05.2017)
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Journal Article
In situ structure of actin remodeling during glucose-stimulated insulin secretion using cryo-electron tomography
Li, Weimin, Li, Angdi, Yu, Bing, Zhang, Xiaoxiao, Liu, Xiaoyan, White, Kate L., Stevens, Raymond C., Baumeister, Wolfgang, Sali, Andrej, Jasnin, Marion, Sun, Liping
Published in Nature communications (12.02.2024)
Published in Nature communications (12.02.2024)
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Journal Article
Structure-Based Discovery of Novel Chemotypes for Adenosine A2A Receptor Antagonists
Katritch, Vsevolod, Jaakola, Veli-Pekka, Lane, J. Robert, Lin, Judy, IJzerman, Adriaan P, Yeager, Mark, Kufareva, Irina, Stevens, Raymond C, Abagyan, Ruben
Published in Journal of medicinal chemistry (25.02.2010)
Published in Journal of medicinal chemistry (25.02.2010)
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Journal Article
Conjunctive encoding of exploratory intentions and spatial information in the hippocampus
Zeng, Yi-Fan, Yang, Ke-Xin, Cui, Yilong, Zhu, Xiao-Na, Li, Rui, Zhang, Hanqing, Wu, Dong Chuan, Stevens, Raymond C., Hu, Ji, Zhou, Ning
Published in Nature communications (15.04.2024)
Published in Nature communications (15.04.2024)
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Journal Article
Structure-Based Discovery of New Antagonist and Biased Agonist Chemotypes for the Kappa Opioid Receptor
Zheng, Zhong, Huang, Xi-Ping, Mangano, Thomas J, Zou, Rodger, Chen, Xin, Zaidi, Saheem A, Roth, Bryan L, Stevens, Raymond C, Katritch, Vsevolod
Published in Journal of medicinal chemistry (13.04.2017)
Published in Journal of medicinal chemistry (13.04.2017)
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Journal Article
The Importance of Ligand-Receptor Conformational Pairs in Stabilization: Spotlight on the N/OFQ G Protein-Coupled Receptor
Miller, Rebecca L., Thompson, Aaron A., Trapella, Claudio, Guerrini, Remo, Malfacini, Davide, Patel, Nilkanth, Han, Gye Won, Cherezov, Vadim, Caló, Girolamo, Katritch, Vsevolod, Stevens, Raymond C.
Published in Structure (London) (01.12.2015)
Published in Structure (London) (01.12.2015)
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Journal Article
The Role of a Sodium Ion Binding Site in the Allosteric Modulation of the A2A Adenosine G Protein-Coupled Receptor
Gutiérrez-de-Terán, Hugo, Massink, Arnault, Rodríguez, David, Liu, Wei, Han, Gye Won, Joseph, Jeremiah S., Katritch, Ilia, Heitman, Laura H., Xia, Lizi, IJzerman, Adriaan P., Cherezov, Vadim, Katritch, Vsevolod, Stevens, Raymond C.
Published in Structure (London) (03.12.2013)
Published in Structure (London) (03.12.2013)
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Journal Article