Pre-clinical and translational pharmacology of a human interleukin-22 IgG fusion protein for potential treatment of infectious or inflammatory diseases
Stefanich, Eric G., Rae, Julie, Sukumaran, Siddharth, Lutman, Jeff, Lekkerkerker, Annemarie, Ouyang, Wenjun, Wang, Xiaoting, Lee, Donna, Danilenko, Dimitry M., Diehl, Lauri, Loyet, Kelly M., Herman, Ann
Published in Biochemical pharmacology (01.06.2018)
Published in Biochemical pharmacology (01.06.2018)
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Journal Article
Production, characterization and pharmacokinetic properties of antibodies with N-linked Mannose-5 glycans
Yu, Marcella, Brown, Darren, Reed, Chae, Chung, Shan, Lutman, Jeff, Stefanich, Eric, Wong, Anne, Stephan, Jean-Philippe, Bayer, Robert
Published in mAbs (01.07.2012)
Published in mAbs (01.07.2012)
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Journal Article
Automated Affinity Capture and On-Tip Digestion to Accurately Quantitate in Vivo Deamidation of Therapeutic Antibodies
Tran, John C, Tran, Daniel, Hilderbrand, Amy, Andersen, Nisana, Huang, Tao, Reif, Karin, Hotzel, Isidro, Stefanich, Eric G, Liu, Yichin, Wang, Jianyong
Published in Analytical chemistry (Washington) (06.12.2016)
Published in Analytical chemistry (Washington) (06.12.2016)
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Journal Article
Utilizing PK and PD Biomarkers to Guide the First-in-Human Starting Dose Selection of MTBT1466A: A Novel Humanized Monoclonal Anti-TGFβ3 Antibody for the Treatment of Fibrotic Diseases
Yadav, Rajbharan, Sukumaran, Siddharth, Lutman, Jeff, Mitra, Mayur S., Halpern, Wendy, Sun, Tianhe, Setiadi, A. Francesca, Neighbors, Margaret, Sheng, X. Rebecca, Yip, Victor, Shen, Ben-Quan, Liu, Chang, Han, Lyrialle, Ovacik, Ayse Meric, Wu, Yan, Glickstein, Sara, Kunder, Rebecca, Arron, Joseph R., Pan, Lin, Kamath, Amrita V., Stefanich, Eric G.
Published in Journal of pharmaceutical sciences (01.11.2023)
Published in Journal of pharmaceutical sciences (01.11.2023)
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Journal Article
Translational PK/PD and the first-in-human dose selection of a PD1/IL15: an engineered recombinant targeted cytokine for cancer immunotherapy
Yadav, Rajbharan, Schubbert, Suzanne, Holder, Patrick G, Chiang, Eugene Y, Kiabi, Nargess, Bogaert, Liz, Leung, Irene, Rashid, Rumana, Avery, Kendra N, Bonzon, Christine, Desjarlais, John R, Sanjabi, Shomyseh, Sharma, Amy, Lepherd, Michelle, Shelton, Amy, Chan, Pam, Liu, Yanqiu, Joslyn, Louis, Hosseini, Iraj, Stefanich, Eric G, Kamath, Amrita V, Bernett, Matthew J, Shivva, Vittal
Published in Frontiers in pharmacology (03.06.2024)
Published in Frontiers in pharmacology (03.06.2024)
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Journal Article
Equilibrative Nucleoside Transporter 3 Deficiency Perturbs Lysosome Function and Macrophage Homeostasis
Hsu, Chia-Lin, Lin, Weiyu, Seshasayee, Dhaya, Chen, Yung-Hsiang, Ding, Xiao, Lin, Zhonghua, Suto, Eric, Huang, Zhiyu, Lee, Wyne P., Park, Hyunjoo, Xu, Min, Sun, Mei, Rangell, Linda, Lutman, Jeff L., Ulufatu, Sheila, Stefanich, Eric, Chalouni, Cecile, Sagolla, Meredith, Diehl, Lauri, Fielder, Paul, Dean, Brian, Balazs, Mercedesz, Martin, Flavius
Published in Science (American Association for the Advancement of Science) (06.01.2012)
Published in Science (American Association for the Advancement of Science) (06.01.2012)
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Journal Article
A Preclinical Population Pharmacokinetic Model for Anti‐CD20/CD3 T‐Cell‐Dependent Bispecific Antibodies
Ferl, Gregory Z., Reyes, Arthur, Sun, Liping L., Cheu, Melissa, Oldendorp, Amy, Ramanujan, Saroja, Stefanich, Eric G.
Published in Clinical and translational science (01.05.2018)
Published in Clinical and translational science (01.05.2018)
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Journal Article
An integrated approach for characterizing immunogenic responses toward a bispecific antibody
Cohen, Sivan, Chung, Shan, Spiess, Christoph, Lundin, Victor, Stefanich, Eric, Laing, Steven T, Clark, Vanessa, Brumm, Jochen, Zhou, Ying, Huang, Catherine, Guerrero, Joyce, Myneni, Srividya, Yadav, Rajbharan, Siradze, Ketevan, Peng, Kun
Published in mAbs (01.01.2021)
Published in mAbs (01.01.2021)
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Journal Article
Nonclinical Pharmacokinetics and Pharmacodynamics Characterization of Anti-CD79b/CD3 T Cell-Dependent Bispecific Antibody Using a Surrogate Molecule: A Potential Therapeutic Agent for B Cell Malignancies
Yadav, Rajbharan, Sukumaran, Siddharth, Zabka, Tanja S, Li, Jinze, Oldendorp, Amy, Morrow, Gary, Reyes, Arthur, Cheu, Melissa, Li, Jessica, Wallin, Jeffrey J, Tsai, Siao, Sun, Laura, Wang, Peiyin, Ellerman, Diego, Spiess, Christoph, Polson, Andy, Stefanich, Eric G, Kamath, Amrita V, Ovacik, Meric A
Published in Pharmaceutics (30.04.2022)
Published in Pharmaceutics (30.04.2022)
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Journal Article
Therapeutic Antibody-Induced Vascular Toxicity Due to Off-Target Activation of Nitric Oxide in Cynomolgus Monkeys
Pai, Rama, Ma, Ning, Connor, Anu V, Danilenko, Dimitry M, Tarrant, Jacqueline M, Salvail, Dany, Wong, Lisa, Hartley, Dylan P, Misner, Dinah, Stefanich, Eric, Wu, Yan, Chen, Yongmei, Wang, Hong, Dambach, Donna M
Published in Toxicological sciences (01.06.2016)
Published in Toxicological sciences (01.06.2016)
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Journal Article
Nonclinical safety assessment of a human interleukin‐22FC IG fusion protein demonstrates in vitro to in vivo and cross‐species translatability
Lee, Donna W., Zhong, Shelly, Pai, Rama, Rae, Julie, Sukumaran, Siddharth, Stefanich, Eric G., Lutman, Jeff, Doudement, Estelle, Wang, Xiaoting, Harder, Brandon, Lekkerkerker, Annemarie, Herman, Ann, Ouyang, Wenjun, Danilenko, Dimitry M.
Published in Pharmacology research & perspectives (01.12.2018)
Published in Pharmacology research & perspectives (01.12.2018)
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Journal Article
Effect of antigen binding affinity and effector function on the pharmacokinetics and pharmacodynamics of anti-IgE monoclonal antibodies
Mortensen, Deborah L., Prabhu, Saileta, Stefanich, Eric G., Kadkhodayan-Fischer, Saloumeh, Gelzleichter, Thomas R., Baker, Dana, Jiang, Jenny, Wallace, Kristin, Iyer, Suhasini, Fielder, Paul J., Putnam, Wendy S.
Published in mAbs (01.11.2012)
Published in mAbs (01.11.2012)
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Journal Article
Functional consequences of the macrophage stimulating protein 689C inflammatory bowel disease risk allele
Kauder, Steven E, Santell, Lydia, Mai, Elaine, Wright, Lilyan Y, Luis, Elizabeth, N'Diaye, Elsa N, Lutman, Jeff, Ratti, Navneet, Sa, Susan M, Maun, Henry R, Stefanich, Eric, Gonzalez, Lino C, Graham, Robert R, Diehl, Lauri, Faubion, Jr, William A, Keir, Mary E, Young, Judy, Chaudhuri, Amitabha, Lazarus, Robert A, Egen, Jackson G
Published in PloS one (23.12.2013)
Published in PloS one (23.12.2013)
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Journal Article
Nonclinical safety assessment of a human interleukin‐22 FC IG fusion protein demonstrates in vitro to in vivo and cross‐species translatability
Lee, Donna W., Zhong, Shelly, Pai, Rama, Rae, Julie, Sukumaran, Siddharth, Stefanich, Eric G., Lutman, Jeff, Doudement, Estelle, Wang, Xiaoting, Harder, Brandon, Lekkerkerker, Annemarie, Herman, Ann, Ouyang, Wenjun, Danilenko, Dimitry M.
Published in Pharmacology research & perspectives (01.12.2018)
Published in Pharmacology research & perspectives (01.12.2018)
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Journal Article
Evidence for an Asialoglycoprotein Receptor on Nonparenchymal Cells for O-Linked Glycoproteins
Stefanich, Eric G, Ren, Song, Danilenko, Dimitry M, Lim, Amy, Song, An, Iyer, Suhasini, Fielder, Paul J
Published in The Journal of pharmacology and experimental therapeutics (01.11.2008)
Published in The Journal of pharmacology and experimental therapeutics (01.11.2008)
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Journal Article
Randomized Phase I Healthy Volunteer Study of UTTR1147A (IL-22Fc): A Potential Therapy for Epithelial Injury
Rothenberg, Michael E, Wang, Yehong, Lekkerkerker, Annemarie, Danilenko, Dimitry M, Maciuca, Romeo, Erickson, Rich, Herman, Ann, Stefanich, Eric, Lu, Timothy T
Published in Clinical pharmacology and therapeutics (01.01.2019)
Published in Clinical pharmacology and therapeutics (01.01.2019)
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Journal Article
Role of the Distal Half of the c-Mpl Intracellular Domain in Control of Platelet Production by Thrombopoietin In Vivo
Luoh, Shiuh-Ming, Stefanich, Eric, Solar, Gregg, Steinmetz, Hope, Lipari, Terry, Pestina, Tamara I., Jackson, Carl W., de Sauvage, Frederic J.
Published in Molecular and Cellular Biology (01.01.2000)
Published in Molecular and Cellular Biology (01.01.2000)
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Journal Article
Anti-CD20/CD3 T cell-dependent bispecific antibody for the treatment of B cell malignancies
Sun, Liping L, Ellerman, Diego, Mathieu, Mary, Hristopoulos, Maria, Chen, Xiaocheng, Li, Yijin, Yan, Xiaojie, Clark, Robyn, Reyes, Arthur, Stefanich, Eric, Mai, Elaine, Young, Judy, Johnson, Clarissa, Huseni, Mahrukh, Wang, Xinhua, Chen, Yvonne, Wang, Peiyin, Wang, Hong, Dybdal, Noel, Chu, Yu-Waye, Chiorazzi, Nicholas, Scheer, Justin M, Junttila, Teemu, Totpal, Klara, Dennis, Mark S, Ebens, Allen J
Published in Science translational medicine (13.05.2015)
Published in Science translational medicine (13.05.2015)
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Journal Article
Sialic Acid Mediated Endothelial and Hepatic Uptake: A Mechanism based Mathematic Model Elucidating the Complex Pharmacokinetics and Pharmacodynamics of Efmarodocokin Alfa, a Variably Glycosylated Fusion Protein
Tao, Xun, Sukumaran, Siddharth, Sperinde, Gizette, Liu, Chang, Beardsley, Michelle Irwin, Day, Peter, Kalo, Matt, Ayewoh, Ebehiremen, Cai, Hao, Wang, Yehong, Jun, Inyoung, Hirst, Kyle, Nguyen, Van, Chung, Shan, Lee, Donna, Lekkerkerker, Annemarie, Stefanich, Eric
Published in Journal of pharmaceutical sciences (01.07.2024)
Published in Journal of pharmaceutical sciences (01.07.2024)
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