Optimized Catalytic Enantioselective Aryl Transfer Process Gives Access to mGlu2 Receptor Potentiators
Magnus, Nicholas A, Anzeveno, Peter B, Coffey, D. Scott, Hay, David A, Laurila, Michael E, Schkeryantz, Jeffrey M, Shaw, Bruce W, Staszak, Michael A
Published in Organic process research & development (01.05.2007)
Published in Organic process research & development (01.05.2007)
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Discovery of Cathepsin S Inhibitor LY3000328 for the Treatment of Abdominal Aortic Aneurysm
Jadhav, Prabhakar K, Schiffler, Matthew A, Gavardinas, Kostas, Kim, Euibong J, Matthews, Donald P, Staszak, Michael A, Coffey, D. Scott, Shaw, Bruce W, Cassidy, Kenneth C, Brier, Richard A, Zhang, Yuke, Christie, Robert M, Matter, William F, Qing, Keyun, Durbin, Jim D, Wang, Yong, Deng, Gary G
Published in ACS medicinal chemistry letters (09.10.2014)
Published in ACS medicinal chemistry letters (09.10.2014)
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Diastereomeric Salt Resolution Based Synthesis of LY503430, an AMPA (α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid) Potentiator
Magnus, Nicholas A, Aikins, James A, Cronin, Jason S, Diseroad, William D, Hargis, Amy D, LeTourneau, Michael E, Parker, Bruce E, Reutzel-Edens, Susan M, Schafer, John P, Staszak, Michael A, Stephenson, Gregory A, Tameze, Shella L, Zollars, Lisa M. H
Published in Organic process research & development (01.09.2005)
Published in Organic process research & development (01.09.2005)
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Green N-Methylation of Electron Deficient Pyrroles with Dimethylcarbonate
Laurila, Michael L, Magnus, Nicholas A, Staszak, Michael A
Published in Organic process research & development (20.11.2009)
Published in Organic process research & development (20.11.2009)
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The Development of Practical Synthetic Routes to a CB2 Agonist: Efficient Construction of a Densely Substituted Purine Core
DeBaillie, Amy C, Jones, Chauncey D, Laurila, Michael E, Magnus, Nicholas A, Staszak, Michael A
Published in Organic process research & development (15.02.2013)
Published in Organic process research & development (15.02.2013)
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Synthesis of 4-Cyano Pyrroles via Mild Knorr Reactions with β-Ketonitriles
Magnus, Nicholas A, Staszak, Michael A, Udodong, Uko E, Wepsiec, James P
Published in Organic process research & development (15.09.2006)
Published in Organic process research & development (15.09.2006)
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Nucleosidic Phosphoramidite Synthesis via Phosphitylation: Activator Selection and Process Development
Xie, Chaoyu, Staszak, Michael A, Quatroche, John T, Sturgill, Christa D, Khau, Vien V, Martinelli, Michael J
Published in Organic process research & development (01.11.2005)
Published in Organic process research & development (01.11.2005)
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A Convergent Kilogram-Scale Synthesis of the PPARα Agonist LY518674: Discovery of a Novel Acid-Mediated Triazolone Synthesis
Braden, Timothy M, Coffey, D. Scott, Doecke, Christopher W, LeTourneau, Michael E, Martinelli, Michael J, Meyer, Christopher L, Miller, Richard D, Pawlak, Joseph M, Pedersen, Steven W, Schmid, Christopher R, Shaw, Bruce W, Staszak, Michael A, Vicenzi, Jeffrey T
Published in Organic process research & development (01.05.2007)
Published in Organic process research & development (01.05.2007)
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Reaction of cryptophycin 52 with thiols
Martinelli, Michael J, Vaidyanathan, Rajappa, Khau, Vien Van, Staszak, Michael A
Published in Tetrahedron letters (29.04.2002)
Published in Tetrahedron letters (29.04.2002)
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Journal Article
Reductive Alkylation of Glycopeptide Antibiotics: Synthesis and Antibacterial Activity
COOPER, ROBIN D. G., SNYDER, NANCY J., ZWEIFEL, MARK J., STASZAK, MICHAEL A., WILKIE, STEPHEN C., NICAS, THALIA I., MULLEN, DEBORAH L., BUTLER, THOMAS F., RODRIGUEZ, MICHAEL J., HUFF, BRET E., THOMPSON, RICHARD C.
Published in Journal of antibiotics (1996)
Published in Journal of antibiotics (1996)
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Enantioselective Syntheses of 1-Carbacephalosporins from Chemoenzymically Derived β-Hydroxy-α-Amino Acids: Applications to the Total Synthesis of Carbacephem Antibiotic Loracarbef
Jackson, Billy G, Pedersen, Steve W, Fisher, Jack W, Misner, Jerry W, Gardner, John P, Staszak, Michael A, Doecke, Christopher, Rizzo, John, Aikins, James, Farkas, Eugene, Trinkle, Kristina L, Vicenzi, Jeffrey, Reinhard, Matt, Kroeff, Eugene P, Higginbotham, Chris A, Gazak, R.J, Zhang, Tony Y
Published in Tetrahedron (28.07.2000)
Published in Tetrahedron (28.07.2000)
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The Development of Practical Synthetic Routes to a CB 2 Agonist: Efficient Construction of a Densely Substituted Purine Core
DeBaillie, Amy C., Jones, Chauncey D., Laurila, Michael E., Magnus, Nicholas A., Staszak, Michael A.
Published in Organic process research & development (15.02.2013)
Published in Organic process research & development (15.02.2013)
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Strategies for the synthesis of N-(azacycloalkyl)bisindolylmaleimides: selective inhibitors of PKCβ
Faul, Margaret M., Grutsch, John L., Kobierski, Michael E., Kopach, Michael E., Krumrich, Christine A., Staszak, Michael A., Udodong, Uko, Vicenzi, Jeffrey T., Sullivan, Kevin A.
Published in Tetrahedron (01.09.2003)
Published in Tetrahedron (01.09.2003)
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Protection, metalation, and electrophilic substitution of 5-methyl tetrazole
Huff, Bret E., LeTourneau, Michael E., Staszak, Michael A., Ward, Jeffrey A.
Published in Tetrahedron letters (20.05.1996)
Published in Tetrahedron letters (20.05.1996)
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Synthesis of 2′,3′-dideoxy-3′-hydroxymethylcytidine; a unique antiviral nucleoside
Faul, Margaret M., Huff, Bret E., Dunlap, Steven E., Frank, Scott A., Fritz, James E., Kaldor, Stephen W., LeTourneau, Michael E., Staszak, Michael A., Ward, Jeffrey A., Werner, John A., Winneroski, Leonard L.
Published in Tetrahedron (16.06.1997)
Published in Tetrahedron (16.06.1997)
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Practical and Enantiospecific Synthesis of LY303870, a Novel NK-1 Antagonist
Hipskind, Philip A, Howbert, J. Jeffry, Cho, Stephen, Cronin, Jason S, Fort, Stuart L, Ginah, Francis O, Hansen, Guy J, Huff, Bret E, Lobb, Karen L
Published in Journal of organic chemistry (01.10.1995)
Published in Journal of organic chemistry (01.10.1995)
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