The Chemistry Behind ADCs
Kostova, Vesela, Désos, Patrice, Starck, Jérôme-Benoît, Kotschy, Andras
Published in Pharmaceuticals (Basel, Switzerland) (07.05.2021)
Published in Pharmaceuticals (Basel, Switzerland) (07.05.2021)
Get full text
Journal Article
S55746 is a novel orally active BCL-2 selective and potent inhibitor that impairs hematological tumor growth
Casara, Patrick, Davidson, James, Claperon, Audrey, Le Toumelin-Braizat, Gaëtane, Vogler, Meike, Bruno, Alain, Chanrion, Maïa, Lysiak-Auvity, Gaëlle, Le Diguarher, Thierry, Starck, Jérôme-Benoît, Chen, Ijen, Whitehead, Neil, Graham, Christopher, Matassova, Natalia, Dokurno, Pawel, Pedder, Christopher, Wang, Youzhen, Qiu, Shumei, Girard, Anne-Marie, Schneider, Emilie, Gravé, Fabienne, Studeny, Aurélie, Guasconi, Ghislaine, Rocchetti, Francesca, Maïga, Sophie, Henlin, Jean-Michel, Colland, Frédéric, Kraus-Berthier, Laurence, Le Gouill, Steven, Dyer, Martin J S, Hubbard, Roderick, Wood, Mike, Amiot, Martine, Cohen, Gerald M, Hickman, John A, Morris, Erick, Murray, James, Geneste, Olivier
Published in Oncotarget (13.04.2018)
Published in Oncotarget (13.04.2018)
Get full text
Journal Article
NOVEL INDOLIZINE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME
DE NANTEUIL, Guillaume, MURRAY, James Brooke, STARCK, Jerôme-Benoît, GENESTE, Olivier, LE DIGUARHER, Thierry, LE TIRAN, Arnaud, CHEN, I-Jen, DAVIDSON, James Edward Paul, HENLIN, Jean-Michel
Year of Publication 28.11.2018
Get full text
Year of Publication 28.11.2018
Patent
NOVEL INDOLIZINE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME
DE NANTEUIL, Guillaume, MURRAY, James Brooke, STARCK, Jerôme-Benoît, GENESTE, Olivier, LE DIGUARHER, Thierry, LE TIRAN, Arnaud, CHEN, I-Jen, DAVIDSON, James Edward Paul, HENLIN, Jean-Michel
Year of Publication 28.08.2018
Get full text
Year of Publication 28.08.2018
Patent
NEW ISOINDOLINE OR ISOQUINOLINE COMPOUNDS, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
Le Diguarher, Thierry, BROUGH, Paul, MURRAY, James, STARCK, Jerôme-Benoît, GENESTE, Olivier, KOTSCHY, Andras, CHEN, I-Jen, MEISSNER, Johannes, WALMSLEY, Claire, NYERGES, Miklos, Le Tiran, Arnaud, de Nanteuil, Guillaume, SZLAVIK, Zoltan, DAVIDSON, James, TATAI, Janos, DODSWORTH, Mark, FEJES, Imre, HENLIN, Jean-Michel, Guillouzic, Anne-Françoise
Year of Publication 28.05.2019
Get full text
Year of Publication 28.05.2019
Patent
NOVEL DERIVATIVES OF INDOLE AND PYRROLE, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME
MURRAY, James Brooke, STARCK, Jerôme-Benoît, GENESTE, Olivier, CHEN, I-Jen, DAVIDSON, James Edward Paul, WALMSLEY, Claire, RAY, Stuart, DE NANTEUIL, Guillaume, BEDFORD, Simon, LE DIGUARHER, Thierry, MADDOX, Daniel, LE TIRAN, Arnaud, GRAHAM, Christopher John, CASARA, Patrick, HENLIN, Jean-Michel
Year of Publication 28.01.2019
Get full text
Year of Publication 28.01.2019
Patent
PARA-AMINO-BENZYL LINKERS, PROCESS FOR THEIR PREPARATION AND THEIR USE IN CONJUGATES
KOSTOVA, VESELA, FRANZETTI, GEORGES-ALAIN, DESOS, PATRICE, STARCK, JÉRÔME-BENOÎT
Year of Publication 23.09.2024
Get full text
Year of Publication 23.09.2024
Patent
New pyrrole derivatives, method of preparing same and pharmaceutical compositions containing them
Le Diguarher, Thierry, Geneste, Olivier, Fejes, Imre, Davidson, James Edward Paul, Chen, I-Jen, Le Tiran, Arnaud, Starck, Jerôme-Benoît, De Nanteuil, Guillaume, Murray, James Brooke, Nyerges, Miklos, Henlin, Jean-Michel, Durand, Didier, Tatai, Janos, Guillouzic, Anne-Françoise
Year of Publication 28.11.2017
Get full text
Year of Publication 28.11.2017
Patent
PARA-AMINO-BENZYL LINKERS, PROCESS FOR THEIR PREPARATION AND THEIR USE IN CONJUGATES
KOSTOVA, VESELA, FRANZETTI, GEORGES-ALAIN, DESOS, PATRICE, STARCK, JÉRÔME-BENOÎT
Year of Publication 30.08.2024
Get full text
Year of Publication 30.08.2024
Patent
PARA-AMINO-BENZYL LINKERS, PROCESS FOR THEIR PREPARATION AND THEIR USE IN CONJUGATES
FRANZETTI, Georges-Alain, DESOS, Patrice, STARCK, Jérôme-Benoît, KOSTOVA, Vesela
Year of Publication 18.07.2024
Get full text
Year of Publication 18.07.2024
Patent
PARA-AMINO-BENZYL LINKERS, PROCESS FOR THEIR PREPARATION AND THEIR USE IN CONJUGATES
FRANZETTI, Georges-Alain, DESOS, Patrice, STARCK, Jérôme-Benoît, KOSTOVA, Vesela
Year of Publication 25.06.2024
Get full text
Year of Publication 25.06.2024
Patent
PARA-AMINO-BENZYL LINKERS, PROCESS FOR THEIR PREPARATION AND THEIR USE IN CONJUGATES
FRANZETTI, Georges-Alain, DESOS, Patrice, STARCK, Jérôme-Benoît, KOSTOVA, Vesela
Year of Publication 15.05.2024
Get full text
Year of Publication 15.05.2024
Patent
New phosphate derivatives, method of preparing same and pharmaceutical compositions containing them
Le Diguarher, Thierry, Geneste, Olivier, Starck, Jerôme-Benoît, Davidson, James Edward Paul, De Nanteuil, Guillaume, Murray, James Brooke, Chen, I-Jen, Henlin, Jean-Michel, Le Tiran, Arnaud, Guillouzic, Anne-Françoise
Year of Publication 28.03.2017
Get full text
Year of Publication 28.03.2017
Patent
NUEVOS DERIVADOS MACROCICLICOS, SU PROCEDIMIENTO DE PREPARACION Y LAS COMPOSICIONES FARMACEUTICAS QUE LOS CONTIENEN
STARCK, Jerôme-Benoît, DURAND, Didier, CHEN, I-Jen, LE TIRAN, Arnaud, LIGETI, Melinda, NYERGES, Miklos, ORTUNO, Jean-Claude, FEJES, Imre
Year of Publication 29.12.2020
Get full text
Year of Publication 29.12.2020
Patent
PARA-AMINO-BENZYL LINKERS, PROCESS FOR THEIR PREPARATION AND THEIR USE IN CONJUGATES
FRANZETTI, Georges-Alain, DESOS, Patrice, STARCK, Jérôme-Benoît, KOSTOVA, Vesela
Year of Publication 13.07.2023
Get full text
Year of Publication 13.07.2023
Patent
NEW INDOLIZINE DERIVATIVES, METHOD FOR PREPARING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM FOR THE TREATMENT OF CANCER
MURRAY, James Brooke, STARCK, Jerôme-Benoît, GENESTE, Olivier, NYERGES Miklos, CHEN, I-Jen, DAVIDSON, James Edward Paul, DEPIL, Stephane, DE NANTEUIL, Guillaume, LE DIGUARHER, Thierry, GRAHAM, Christopher John, LE TIRAN, Arnaud, CASARA, Patrick, HICKMAN, John, HENLIN, Jean-Michel
Year of Publication 28.08.2017
Get full text
Year of Publication 28.08.2017
Patent
DERIVADOS DE 3,6-DIAMINO-PIRIDAZIN-3-ILO, COMPOSICIONES FARMACEUTICAS QUE LOS CONTIENEN Y SUS USOS COMO AGENTES PROAPOPTOTICOS
CHANRION, Maia, MARAGNO, Ana Leticia, MURRAY, James Brooke, STARCK, Jerôme-Benoît, COLLAND, Frederic, NOVAK, Tibor, KOTSCHY, Andras, MOLNAR, Mark, DAVIDSON, James Edward Paul, NYERGES, Miklos, DUNKEL, Petra, DODSWORTH, Mark Philip, BEDFORD, Simon, HERNER, Andras, MADARASZ, Zoltan, DESOS, Patrice, TIMARI, Matyas Pal, RUDASOVA, Monika, PACZAL, Attila, SZIGETI, Marianna, PARSONS, Rachel Jane, STROFEK, Agnes, WEBB, Paul
Year of Publication 04.05.2022
Get full text
Year of Publication 04.05.2022
Patent
PARA-AMINO-BENZYL LINKERS, PROCESS FOR THEIR PREPARATION AND THEIR USE IN CONJUGATES
FRANZETTI, Georges-Alain, DESOS, Patrice, STARCK, Jérôme-Benoît, KOSTOVA, Vesela
Year of Publication 29.03.2023
Get full text
Year of Publication 29.03.2023
Patent
Para-amino-benzyl linkers, process for their preparation and their use in conjugates
FRANZETTI, Georges-Alain, DESOS, Patrice, STARCK, Jérôme-Benoît, KOSTOVA, Vesela
Year of Publication 05.01.2023
Get full text
Year of Publication 05.01.2023
Patent