Search Results - "STAPELFELD, Awilda" :: K.UTB vyhledávací portál

8-chlorodibenz[b,f][1,4]oxazepine-10(11H)-carboxylic acid,2-[3-[2-(furanylmethyl)thio]-1-oxopropyl]hydrazide (SC-51322): A potent PGE2 antagonist and analgesic

by Hallinan, E.Ann, Stapelfeld, Awilda, Savage, Michael A., Reichman, Melvin
Published in Bioorganic & medicinal chemistry letters (01.02.1994)

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Systemic analgesic activity and .delta.-opioid selectivity in [2,6-dimethyl-Tyr1, D-Pen2, D-Pen5]enkephalin

by Hansen, Donald W, Stapelfeld, Awilda, Savage, Michael A, Reichman, Melvin, Hammond, Donna L, Haaseth, Ronald C, Mosberg, Henry I
Published in Journal of medicinal chemistry (01.02.1992)

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Enkephalin Analogs as Systemically Active Antinociceptive Agents: O- and N-Alkylated Derivatives of the Dipeptide Amide L-2,6-Dimethyltyrosyl-N-(3-phenylpropyl)-D-alaninamide

by Pitzele, Barnett S, Hamilton, Robert W, Kudla, Kathleen D, Tsymbalov, Sofya, Stapelfeld, Awilda, Savage, Michael A, Clare, Michael, Hammond, Donna L, Hansen, Donald W
Published in Journal of medicinal chemistry (01.04.1994)

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Preparation and opioid activity of analogs of the analgesic dipeptide 2,6-dimethyl-L-tyrosyl-N-(3-phenylpropyl)-D-alaninamide

by Chandrakumar, Nizal S, Yonan, Peter K, Stapelfeld, Awilda, Savage, Michael, Rorbacher, Elaine, Contreras, Patricia C, Hammond, Donna
Published in Journal of medicinal chemistry (01.01.1992)

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2,4-disubstituted oxazoles and thiazoles as latent pharmacophores for diacylhydrazine of SC-51089, a potent PGE2 antagonist

by HALLINAN, E. Ann, HAGEN, Timothy J, TSYMBALOV, Sofya, STAPELFELD, Awilda, SAVAGE, Michael A
Published in Bioorganic & medicinal chemistry (2001)

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2,4-Disubstituted oxazoles and thiazoles as latent pharmacophores for diacylhydrazine of SC-51089, a potent PGE 2 antagonist

by Hallinan, E.Ann, Hagen, Timothy J., Tsymbalov, Sofya, Stapelfeld, Awilda, Savage, Michael A.
Published in Bioorganic & medicinal chemistry (2001)

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Aminoacetyl Moiety as a Potential Surrogate for Diacylhydrazine Group of SC-51089, a Potent PGE2 Antagonist, and Its Analogs

by Hallinan, E. Ann, Hagen, Timothy J, Tsymbalov, Sofya, Husa, Robert K, Lee, Albert C, Stapelfeld, Awilda, Savage, Michael A
Published in Journal of medicinal chemistry (19.01.1996)

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N-Substituted dibenzoxazepines as analgesic PGE2 antagonists

by Hallinan, E. Ann, Hagen, Timothy J, Husa, Robert K, Tsymbalov, Sofya, Rao, Shashidhar N, vanHoeck, Jean Pierre, Rafferty, Michael F, Stapelfeld, Awilda, Savage, Michael A, Reichman, Melvin
Published in Journal of medicinal chemistry (01.10.1993)

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8-chlorodibenz[b,f][1,4]oxazepine-10(11H)-carboxylic acid,2-[3-[2-(furanylmethyl)thio]-1-oxopropyl]hydrazide (SC-51322): A potent PGE 2 antagonist and analgesic

by Hallinan, E.Ann, Stapelfeld, Awilda, Savage, Michael A., Reichman, Melvin
Published in Bioorganic & medicinal chemistry letters (1994)

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Aminoacetyl Moiety as a Potential Surrogate for Diacylhydrazine Group of SC-51089, a Potent PGE 2 Antagonist, and Its Analogs

by Hallinan, E. Ann, Hagen, Timothy J., Tsymbalov, Sofya, Husa, Robert K., Lee, Albert C., Stapelfeld, Awilda, Savage, Michael A.
Published in Journal of medicinal chemistry (01.01.1996)

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Analogs of the .delta. opioid receptor selective cyclic peptide [cyclic][2-D-penicillamine,5-D-penicillamine]-enkephalin: 2',6'-dimethyltyrosine and Gly3-Phe4 amide bond isostere substitutions

by Chandrakumar, Nizal S, Stapelfeld, Awilda, Beardsley, Patrick M, Lopez, Oscar T, Drury, Bridget, Anthony, Elizabeth, Savage, Michael A, Williamson, L. Neil, Reichman, Melvin
Published in Journal of medicinal chemistry (07.08.1992)

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