Current Concepts and Treatments of Schizophrenia
Stępnicki, Piotr, Kondej, Magda, Kaczor, Agnieszka A
Published in Molecules (Basel, Switzerland) (20.08.2018)
Published in Molecules (Basel, Switzerland) (20.08.2018)
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Journal Article
Multi-Target Approach for Drug Discovery against Schizophrenia
Kondej, Magda, Stępnicki, Piotr, Kaczor, Agnieszka A
Published in International journal of molecular sciences (10.10.2018)
Published in International journal of molecular sciences (10.10.2018)
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Overcoming Depression with 5-HT2A Receptor Ligands
Zięba, Agata, Stępnicki, Piotr, Matosiuk, Dariusz, Kaczor, Agnieszka A.
Published in International journal of molecular sciences (01.01.2022)
Published in International journal of molecular sciences (01.01.2022)
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Screening and Structure-Activity Relationship of D2AAK1 Derivatives for Potential Application in the Treatment of Neurodegenerative Diseases
Koszła, Oliwia, Sołek, Przemysław, Stępnicki, Piotr, Kaczor, Agnieszka A
Published in Molecules (Basel, Switzerland) (30.03.2022)
Published in Molecules (Basel, Switzerland) (30.03.2022)
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What are the challenges with multi-targeted drug design for complex diseases?
Zięba, Agata, Stępnicki, Piotr, Matosiuk, Dariusz, Kaczor, Agnieszka A
Published in Expert opinion on drug discovery (03.07.2022)
Published in Expert opinion on drug discovery (03.07.2022)
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Journal Article
Experimental and computational structural studies of 5-substituted-3-(1-arylmethyl-1,2,3,6-tetrahydropyridin-4-yl)-1H-indoles
Bartyzel, Agata, Kondej, Magda, Stępnicki, Piotr, Wróbel, Tomasz M., Kaczor, Agnieszka A.
Published in Journal of molecular structure (05.12.2021)
Published in Journal of molecular structure (05.12.2021)
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Journal Article
Effects of small molecules on neurogenesis: Neuronal proliferation and differentiation
Jastrzębski, Michał K., Wójcik, Piotr, Stępnicki, Piotr, Kaczor, Agnieszka A.
Published in Acta pharmaceutica Sinica. B (01.01.2024)
Published in Acta pharmaceutica Sinica. B (01.01.2024)
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Journal Article
Multi-targeted drug design strategies for the treatment of schizophrenia
Stępnicki, Piotr, Kondej, Magda, Koszła, Oliwia, Żuk, Justyna, Kaczor, Agnieszka A
Published in Expert opinion on drug discovery (02.01.2021)
Published in Expert opinion on drug discovery (02.01.2021)
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Journal Article
Development and Characterization of Novel Selective, Non-Basic Dopamine D2 Receptor Antagonists for the Treatment of Schizophrenia
Stępnicki, Piotr, Wośko, Sylwia, Bartyzel, Agata, Zięba, Agata, Bartuzi, Damian, Szałaj, Klaudia, Wróbel, Tomasz M., Fornal, Emilia, Carlsson, Jens, Kędzierska, Ewa, Poleszak, Ewa, Castro, Marián, Kaczor, Agnieszka A.
Published in Molecules (Basel, Switzerland) (20.05.2023)
Published in Molecules (Basel, Switzerland) (20.05.2023)
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Journal Article
Thermal behavior and determination of physicochemical properties of novel candidates for antipsychotic drugs
Stępnicki, Piotr, Gwarda, Radosław Ł., Bartyzel, Agata, Karcz, Tadeusz, Szczepańska, Katarzyna, Wróbel, Tomasz M., Kaczor, Agnieszka A.
Published in Journal of thermal analysis and calorimetry (2024)
Published in Journal of thermal analysis and calorimetry (2024)
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Funnel metadynamics and behavioral studies reveal complex effect of D2AAK1 ligand on anxiety-like processes
Bartuzi, Damian, Kędzierska, Ewa, Targowska-Duda, Katarzyna M, Koszła, Oliwia, Wróbel, Tomasz M, Jademyr, Simon, Karcz, Tadeusz, Szczepańska, Katarzyna, Stępnicki, Piotr, Wronikowska-Denysiuk, Olga, Biała, Grażyna, Handzlik, Jadwiga, Kristensen, Jesper L, Poso, Antti, Kaczor, Agnieszka A
Published in Scientific reports (07.12.2022)
Published in Scientific reports (07.12.2022)
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Journal Article
Novel multi-target ligands of dopamine and serotonin receptors for the treatment of schizophrenia based on indazole and piperazine scaffolds-synthesis, biological activity, and structural evaluation
Stępnicki, Piotr, Wronikowska-Denysiuk, Olga, Zięba, Agata, Targowska-Duda, Katarzyna M., Bartyzel, Agata, Wróbel, Martyna Z., Wróbel, Tomasz M., Szałaj, Klaudia, Chodkowski, Andrzej, Mirecka, Karolina, Budzyńska, Barbara, Fornal, Emilia, Turło, Jadwiga, Castro, Marián, Kaczor, Agnieszka A.
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2023)
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2023)
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Journal Article
Discovery and in vitro Evaluation of Novel Serotonin 5‐HT2A Receptor Ligands Identified Through Virtual Screening
Zięba, Agata, Bartuzi, Damian, Stępnicki, Piotr, Matosiuk, Dariusz, Wróbel, Tomasz M., Laitinen, Tuomo, Castro, Marián, Kaczor, Agnieszka A.
Published in ChemMedChem (15.07.2024)
Published in ChemMedChem (15.07.2024)
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Journal Article
The Antipsychotic D2AAK1 as a Memory Enhancer for Treatment of Mental and Neurodegenerative Diseases
Koszła, Oliwia, Sołek, Przemysław, Woźniak, Sylwia, Kędzierska, Ewa, Wróbel, Tomasz M, Kondej, Magda, Archała, Aneta, Stępnicki, Piotr, Biała, Grażyna, Matosiuk, Dariusz, Kaczor, Agnieszka A
Published in International journal of molecular sciences (23.11.2020)
Published in International journal of molecular sciences (23.11.2020)
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Journal Article
Synthesis, pharmacological and structural studies of 5-substituted-3-(1-arylmethyl-1,2,3,6-tetrahydropyridin-4-yl)-1H-indoles as multi-target ligands of aminergic GPCRs
Kondej, Magda, Wróbel, Tomasz M., Silva, Andrea G., Stępnicki, Piotr, Koszła, Oliwia, Kędzierska, Ewa, Bartyzel, Agata, Biała, Grażyna, Matosiuk, Dariusz, Loza, Maria I., Castro, Marián, Kaczor, Agnieszka A.
Published in European journal of medicinal chemistry (15.10.2019)
Published in European journal of medicinal chemistry (15.10.2019)
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Journal Article
N-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}propyl)-1H-indazole-3-carboxamide (D2AAK3) as a potential antipsychotic: In vitro, in silico and in vivo evaluation of a multi-target ligand
Kaczor, Agnieszka A., Targowska-Duda, Katarzyna M., Stępnicki, Piotr, Silva, Andrea G., Koszła, Oliwia, Kędzierska, Ewa, Grudzińska, Angelika, Kruk-Słomka, Marta, Biała, Grażyna, Castro, Marián
Published in Neurochemistry international (01.06.2021)
Published in Neurochemistry international (01.06.2021)
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Journal Article
Development and Characterization of Novel Selective, Non-Basic Dopamine D 2 Receptor Antagonists for the Treatment of Schizophrenia
Stępnicki, Piotr, Wośko, Sylwia, Bartyzel, Agata, Zięba, Agata, Bartuzi, Damian, Szałaj, Klaudia, Wróbel, Tomasz M, Fornal, Emilia, Carlsson, Jens, Kędzierska, Ewa, Poleszak, Ewa, Castro, Marián, Kaczor, Agnieszka A
Published in Molecules (Basel, Switzerland) (20.05.2023)
Published in Molecules (Basel, Switzerland) (20.05.2023)
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Journal Article
Discovery of novel arylpiperazine-based DA/5-HT modulators as potential antipsychotic agents – Design, synthesis, structural studies and pharmacological profiling
Stępnicki, Piotr, Targowska-Duda, Katarzyna M., Martínez, Antón L., Zięba, Agata, Wronikowska-Denysiuk, Olga, Wróbel, Martyna Z., Bartyzel, Agata, Trzpil, Alicja, Wróbel, Tomasz M., Chodkowski, Andrzej, Mirecka, Karolina, Karcz, Tadeusz, Szczepańska, Katarzyna, Loza, Maria I., Budzyńska, Barbara, Turło, Jadwiga, Handzlik, Jadwiga, Fornal, Emilia, Poleszak, Ewa, Castro, Marián, Kaczor, Agnieszka A.
Published in European journal of medicinal chemistry (05.04.2023)
Published in European journal of medicinal chemistry (05.04.2023)
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Journal Article
Multitarget Derivatives of D2AAK1 as Potential Antipsychotics: The Effect of Substitution in the Indole Moiety
Kondej, Magda, Wróbel, Tomasz M., Targowska‐Duda, Katarzyna M., Leandro Martínez, Antón, Koszła, Oliwia, Stępnicki, Piotr, Zięba, Agata, Paz, Alba, Wronikowska‐Denysiuk, Olga, Loza, Maria I., Castro, Marián, Kaczor, Agnieszka A.
Published in ChemMedChem (03.08.2022)
Published in ChemMedChem (03.08.2022)
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