Topical delivery of siRNA into skin using SPACE-peptide carriers
Chen, Ming, Zakrewsky, Michael, Gupta, Vivek, Anselmo, Aaron C., Slee, Deborah H., Muraski, John A., Mitragotri, Samir
Published in Journal of controlled release (10.04.2014)
Published in Journal of controlled release (10.04.2014)
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Journal Article
Topical delivery of Cyclosporine A into the skin using SPACE-peptide
Chen, Ming, Kumar, Sunny, Anselmo, Aaron C., Gupta, Vivek, Slee, Deborah H., Muraski, John A., Mitragotri, Samir
Published in Journal of controlled release (10.02.2015)
Published in Journal of controlled release (10.02.2015)
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Journal Article
Evaluation of KP‐1199: a novel acetaminophen analog for hemostatic function and antinociceptive effects
Reddoch‐Cardenas, Kristin M., Cheppudira, Bopaiah P., Garza, Thomas, Hopkins, Chad D., Bunker, Kevin D., Slee, Deborah H., Cap, Andrew P., Bynum, James A., Christy, Robert J.
Published in Transfusion (Philadelphia, Pa.) (01.07.2021)
Published in Transfusion (Philadelphia, Pa.) (01.07.2021)
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Journal Article
Drugability of Extracellular Targets: Discovery of Small Molecule Drugs Targeting Allosteric, Functional, and Subunit-Selective Sites on GPCRs and Ion Channels
Grigoriadis, Dimitri E, Hoare, Samuel R J, Lechner, Sandra M, Slee, Deborah H, Williams, John A
Published in Neuropsychopharmacology (New York, N.Y.) (01.01.2009)
Published in Neuropsychopharmacology (New York, N.Y.) (01.01.2009)
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Journal Article
Discovery of NBI-77860/GSK561679, a potent corticotropin-releasing factor (CRF 1) receptor antagonist with improved pharmacokinetic properties
Tellew, John E., Lanier, Marion, Moorjani, Manisha, Lin, Emily, Luo, Zhiyong, Slee, Deborah H., Zhang, Xiaohu, Hoare, Sam R.J., Grigoriadis, Dimitri E., Denis, Yves St, Fabio, Romano Di, Modugno, Enza Di, Saunders, John, Williams, John P.
Published in Bioorganic & medicinal chemistry letters (15.12.2010)
Published in Bioorganic & medicinal chemistry letters (15.12.2010)
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Journal Article
Lead Optimization of 4-Acetylamino-2-(3,5-dimethylpyrazol-1-yl)-6-pyridylpyrimidines as A2A Adenosine Receptor Antagonists for the Treatment of Parkinson’s Disease
Zhang, Xiaohu, Tellew, John E, Luo, Zhiyong, Moorjani, Manisha, Lin, Emily, Lanier, Marion C, Chen, Yongsheng, Williams, John P, Saunders, John, Lechner, Sandra M, Markison, Stacy, Joswig, Tanya, Petroski, Robert, Piercey, Jaime, Kargo, William, Malany, Siobhan, Santos, Mark, Gross, Raymond S, Wen, Jenny, Jalali, Kayvon, O’Brien, Zhihong, Stotz, Carol E, Crespo, María I, Díaz, José-Luis, Slee, Deborah H
Published in Journal of medicinal chemistry (27.11.2008)
Published in Journal of medicinal chemistry (27.11.2008)
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Journal Article
Identification of Novel, Water-Soluble, 2-Amino-N-pyrimidin-4-yl Acetamides as A2A Receptor Antagonists with In Vivo Efficacy
Slee, Deborah H, Zhang, Xiaohu, Moorjani, Manisha, Lin, Emily, Lanier, Marion C, Chen, Yongsheng, Rueter, Jaimie K, Lechner, Sandra M, Markison, Stacy, Malany, Siobhan, Joswig, Tanya, Santos, Mark, Gross, Raymond S, Williams, John P, Castro-Palomino, Julio C, Crespo, María I, Prat, Maria, Gual, Silvia, Díaz, José-Luis, Wen, Jenny, O’Brien, Zhihong, Saunders, John
Published in Journal of medicinal chemistry (14.02.2008)
Published in Journal of medicinal chemistry (14.02.2008)
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Journal Article
2-Amino-N-pyrimidin-4-ylacetamides as A2A Receptor Antagonists: 1. Structure−Activity Relationships and Optimization of Heterocyclic Substituents
Slee, Deborah H, Chen, Yongsheng, Zhang, Xiaohu, Moorjani, Manisha, Lanier, Marion C, Lin, Emily, Rueter, Jaimie K, Williams, John P, Lechner, Sandra M, Markison, Stacy, Malany, Siobhan, Santos, Mark, Gross, Raymond S, Jalali, Kayvon, Sai, Yang, Zuo, Zhiyang, Yang, Chun, Castro-Palomino, Julio C, Crespo, María I, Prat, Maria, Gual, Silvia, Díaz, José-Luis, Saunders, John
Published in Journal of medicinal chemistry (27.03.2008)
Published in Journal of medicinal chemistry (27.03.2008)
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Journal Article
Selection, synthesis, and structure–activity relationship of tetrahydropyrido[4,3- d]pyrimidine-2,4-diones as human GnRH receptor antagonists
Lanier, Marion C., Feher, Miklos, Ashweek, Neil J., Loweth, Colin J., Rueter, Jaimie K., Slee, Deborah H., Williams, John P., Zhu, Yun-Fei, Sullivan, Susan K., Brown, Michael S.
Published in Bioorganic & medicinal chemistry (15.08.2007)
Published in Bioorganic & medicinal chemistry (15.08.2007)
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Journal Article
2-Amino-N-pyrimidin-4-ylacetamides as A2A Receptor Antagonists: 2. Reduction of hERG Activity, Observed Species Selectivity, and Structure−Activity Relationships
Slee, Deborah H, Moorjani, Manisha, Zhang, Xiaohu, Lin, Emily, Lanier, Marion C, Chen, Yongsheng, Rueter, Jaimie K, Lechner, Sandra M, Markison, Stacy, Malany, Siobhan, Joswig, Tanya, Santos, Mark, Gross, Raymond S, Williams, John P, Castro-Palomino, Julio C, Crespo, María I, Prat, Maria, Gual, Silvia, Díaz, José-Luis, Jalali, Kayvon, Sai, Yang, Zuo, Zhiyang, Yang, Chun, Wen, Jenny, O’Brien, Zhihong, Petroski, Robert, Saunders, John
Published in Journal of medicinal chemistry (27.03.2008)
Published in Journal of medicinal chemistry (27.03.2008)
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Journal Article
Synthesis of N-pyrimidinyl-2-phenoxyacetamides as adenosine A2A receptor antagonists
XIAOHU ZHANG, RUETER, Jaimie K, MARKISON, Stacy, JOSWIG, Tanya, MALANY, Siobhan, SANTOS, Mark, CASTRO-PALOMINO, Julio C, CRESPO, Maria I, PRAT, Maria, GUAL, Silvia, DIAZ, José-Luis, SAUNDERS, John, YONGSHENG CHEN, SLEE, Deborah H, MOORJANI, Manisha, LANIER, Marion C, LIN, Emily, GROSS, Raymond S, TELLEW, John E, WILLIAMS, John P, LECHNER, Sandra M
Published in Bioorganic & medicinal chemistry letters (15.03.2008)
Published in Bioorganic & medicinal chemistry letters (15.03.2008)
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Journal Article
2,6-Diaryl-4-acylaminopyrimidines as potent and selective adenosine A(2A) antagonists with improved solubility and metabolic stability
Moorjani, Manisha, Luo, Zhiyong, Lin, Emily, Vong, Binh G, Chen, Yongsheng, Zhang, Xiaohu, Rueter, Jaimie K, Gross, Raymond S, Lanier, Marion C, Tellew, John E, Williams, John P, Lechner, Sandra M, Malany, Siobhan, Santos, Mark, Crespo, María I, Díaz, José-Luis, Saunders, John, Slee, Deborah H
Published in Bioorganic & medicinal chemistry letters (15.10.2008)
Published in Bioorganic & medicinal chemistry letters (15.10.2008)
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Journal Article
2,6-Diaryl-4-acylaminopyrimidines as potent and selective adenosine A2A antagonists with improved solubility and metabolic stability
MOORJANI, Manisha, ZHIYONG LUO, WILLIAMS, John P, LECHNER, Sandra M, MALANY, Siobhan, SANTOS, Mark, CRESPO, Maria I, DIAZ, José-Luis, SAUNDERS, John, SLEE, Deborah H, LIN, Emily, VONG, Binh G, YONGSHENG CHEN, XIAOHU ZHANG, RUETER, Jaimie K, GROSS, Raymond S, LANIER, Marion C, TELLEW, John E
Published in Bioorganic & medicinal chemistry letters (15.10.2008)
Published in Bioorganic & medicinal chemistry letters (15.10.2008)
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Journal Article
Inhibition of Fructose-1,6-bisphosphatase by a New Class of Allosteric Effectors
Choe, Jun-Young, Nelson, Scott W., Arienti, Kristen L., Axe, Frank U., Collins, Tassie L., Jones, Todd K., Kimmich, Rachel D.A., Newman, Michael J., Norvell, Karl, Ripka, William C., Romano, Suzanne J., Short, Kevin M., Slee, Deborah H., Fromm, Herbert J., Honzatko, Richard B.
Published in The Journal of biological chemistry (19.12.2003)
Published in The Journal of biological chemistry (19.12.2003)
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Journal Article
Pyrrolopyrazinedione-Based Inhibitors of Human Hormone-Sensitive Lipase
Slee, Deborah H, Bhat, Abhijit S, Nguyen, Truc N, Kish, Mary, Lundeen, Katy, Newman, Michael J, McConnell, Stephen J
Published in Journal of medicinal chemistry (27.03.2003)
Published in Journal of medicinal chemistry (27.03.2003)
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Journal Article
2,6-Diaryl-4-phenacylaminopyrimidines as potent and selective adenosine A(2A) antagonists with reduced hERG liability
Moorjani, Manisha, Zhang, Xiaohu, Chen, Yongsheng, Lin, Emily, Rueter, Jaimie K, Gross, Raymond S, Lanier, Marion C, Tellew, John E, Williams, John P, Lechner, Sandra M, Malany, Siobhan, Santos, Mark, Ekhlassi, Paddi, Castro-Palomino, Julio C, Crespo, María I, Prat, Maria, Gual, Silvia, Díaz, José-Luis, Saunders, John, Slee, Deborah H
Published in Bioorganic & medicinal chemistry letters (15.02.2008)
Published in Bioorganic & medicinal chemistry letters (15.02.2008)
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Journal Article
Development of Potent Non-Carbohydrate Imidazole-Based Small Molecule Selectin Inhibitors with Antiinflammatory Activity
Slee, Deborah H, Romano, Suzanne J, Yu, Jinghua, Nguyen, Truc N, John, Judy K, Raheja, Neil K, Axe, Frank U, Jones, Todd K, Ripka, William C
Published in Journal of medicinal chemistry (21.06.2001)
Published in Journal of medicinal chemistry (21.06.2001)
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Journal Article
2,6-Diaryl-4-phenacylaminopyrimidines as potent and selective adenosine A2A antagonists with reduced hERG liability
MOORJANI, Manisha, XIAOHU ZHANG, MALANY, Siobhan, SANTOS, Mark, EKHLASSI, Paddi, CASTRO-PALOMINO, Julio C, CRESPO, Maria I, PRAT, Maria, GUAL, Silvia, DIAZ, José-Luis, SAUNDERS, John, SLEE, Deborah H, YONGSHENG CHEN, LIN, Emily, RUETER, Jaimie K, GROSS, Raymond S, LANIER, Marion C, TELLEW, John E, WILLIAMS, John P, LECHNER, Sandra M
Published in Bioorganic & medicinal chemistry letters (15.02.2008)
Published in Bioorganic & medicinal chemistry letters (15.02.2008)
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Journal Article
Selectivity in the Inhibition of HIV and FIV Protease: Inhibitory and Mechanistic Studies of Pyrrolidine-Containing .alpha.-Keto Amide and Hydroxyethylamine Core Structures
Slee, Deborah H, Laslo, Karen L, Elder, John H, Ollmann, Ian R, Gustchina, Alla, Kervinen, Jukka, Zdanov, Alexander, Wlodawer, Alexander, Wong, Chi-Huey
Published in Journal of the American Chemical Society (01.12.1995)
Published in Journal of the American Chemical Society (01.12.1995)
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Journal Article
Inhaled seralutinib exhibits potent efficacy in models of pulmonary arterial hypertension
Galkin, Anna, Sitapara, Ravikumar, Clemons, Bryan, Garcia, Eduardo, Kennedy, Michael, Guimond, David, Carter, Laura L, Douthitt, Ashley, Osterhout, Robin, Gandjeva, Aneta, Slee, Deborah, Salter-Cid, Luisa, Tuder, Rubin M, Zisman, Lawrence S
Published in The European respiratory journal (01.12.2022)
Published in The European respiratory journal (01.12.2022)
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