Practical Asymmetric Synthesis of (S)-4-Ethyl-7,8-dihydro-4-hydroxy-1H-pyrano[3,4-f]indolizine- 3,6,10(4H)-trione, a Key Intermediate for the Synthesis of Irinotecan and Other Camptothecin Analogs
Henegar, Kevin E, Ashford, Scott W, Baughman, Ted A, Sih, John C, Gu, Rui-Lin
Published in Journal of organic chemistry (19.09.1997)
Published in Journal of organic chemistry (19.09.1997)
Get full text
Journal Article
(S)-(−)-4-[4-[2-(Isochroman-1-yl)ethyl]piperazin-1-yl]benzenesulfonamide, a Selective Dopamine D4 Antagonist
TenBrink, Ruth E, Bergh, Carol L, Duncan, J. Neil, Harris, Douglas W, Huff, R. M, Lahti, Robert A, Lawson, Charles F, Lutzke, Barry S, Martin, Iain J, Rees, Susan A, Schlachter, Siusaidh K, Sih, John C, Smith, Martin W
Published in Journal of medicinal chemistry (21.06.1996)
Published in Journal of medicinal chemistry (21.06.1996)
Get full text
Journal Article
Synthesis and Biological Activity of Analogues of the Antidiabetic/Antiobesity Agent 3-Guanidinopropionic Acid: Discovery of a Novel Aminoguanidinoacetic Acid Antidiabetic Agent
Larsen, Scott D, Connell, Mark A, Cudahy, Michele M, Evans, Bruce R, May, Paul D, Meglasson, Martin D, O'Sullivan, Theresa J, Schostarez, Heinrich J, Sih, John C, Stevens, F. Craig, Tanis, Steven P, Tegley, Christopher M, Tucker, John A, Vaillancourt, Valerie A, Vidmar, Thomas J, Watt, William, Yu, Jen H
Published in Journal of medicinal chemistry (12.04.2001)
Published in Journal of medicinal chemistry (12.04.2001)
Get full text
Journal Article
Studies on (H+-K+)-ATPase inhibitors of gastric acid secretion. Prodrugs of 2-[(2-pyridinylmethyl)sulfinyl]benzimidazole proton-pump inhibitors
Sih, John C, Wha bin Im, Robert, Andre, Graber, David R, Blakeman, David P
Published in Journal of medicinal chemistry (01.03.1991)
Published in Journal of medicinal chemistry (01.03.1991)
Get full text
Journal Article
An unusual dimer resulting from the addition of ethyl chloroformate to a 2-lithio-1,3-dithiane
Sih, John C, Graber, David R, Mizsak, Stephen A, Scahill, Terrence A
Published in Journal of organic chemistry (01.10.1982)
Published in Journal of organic chemistry (01.10.1982)
Get full text
Journal Article
(S)-(-)-4-[4-[2-(isochroman-1-yl)ethyl]-piperazin-1-yl]benzenesulfonamide, a selective dopamine D-4 antagonist
TenBrink, RE, Bergh, CL, Duncan, JN, Harris, DW, Huff, RM, Lahti, RA, Lawson, CF, Lutzke, BS, Martin, IJ, Rees, SA, Schlachter, SK, Sih, JC, Smith, MW
Published in Journal of medicinal chemistry (21.06.1996)
Published in Journal of medicinal chemistry (21.06.1996)
Get full text
Journal Article