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Huang, Xin, Shaffer, Paul L, Ayube, Shawn, Bregman, Howard, Chen, Hao, Lehto, Sonya G, Luther, Jason A, Matson, David J, McDonough, Stefan I, Michelsen, Klaus, Plant, Matthew H, Schneider, Stephen, Simard, Jeffrey R, Teffera, Yohannes, Yi, Shuyan, Zhang, Maosheng, DiMauro, Erin F, Gingras, Jacinthe
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Published in Nature structural & molecular biology (01.02.2017)
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Published in Bioorganic & medicinal chemistry letters (01.08.2012)
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The Discovery and Hit-to-Lead Optimization of Tricyclic Sulfonamides as Potent and Efficacious Potentiators of Glycine Receptors
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Published in Journal of medicinal chemistry (09.02.2017)
Published in Journal of medicinal chemistry (09.02.2017)
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Purinylpyridinylamino-based DFG-in/αC-helix-out B-Raf inhibitors: Applying mutant versus wild-type B-Raf selectivity indices for compound profiling
Liu, Longbin, Lee, Matthew R., Kim, Joseph L., Whittington, Douglas A., Bregman, Howard, Hua, Zihao, Lewis, Richard T., Martin, Matthew W., Nishimura, Nobuko, Potashman, Michele, Yang, Kevin, Yi, Shuyan, Vaida, Karina R., Epstein, Linda F., Babij, Carol, Fernando, Manory, Carnahan, Josette, Norman, Mark H.
Published in Bioorganic & medicinal chemistry (15.05.2016)
Published in Bioorganic & medicinal chemistry (15.05.2016)
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Crystal structures of human glycine receptor [alpha]3 bound to a novel class of analgesic potentiators
Huang, Xin, Shaffer, Paul L, Ayube, Shawn, Bregman, Howard, Chen, Hao, Lehto, Sonya G, Luther, Jason A, Matson, David J, McDonough, Stefan I, Michelsen, Klaus, Plant, Matthew H, Schneider, Stephen, Simard, Jeffrey R, Teffera, Yohannes, Yi, Shuyan, Zhang, Maosheng, DiMauro, Erin F, Gingras, Jacinthe
Published in Nature structural & molecular biology (01.02.2017)
Published in Nature structural & molecular biology (01.02.2017)
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Design, synthesis, and testing of an 6-O-linked series of benzimidazole based inhibitors of CDK5/p25
Jain, Prashi, Flaherty, Patrick T., Yi, Shuyan, Chopra, Ishveen, Bleasdell, Gwenyth, Lipay, Josh, Ferandin, Yoan, Meijer, Laurent, Madura, Jeffry D.
Published in Bioorganic & medicinal chemistry (01.01.2011)
Published in Bioorganic & medicinal chemistry (01.01.2011)
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Corrigendum to “Purinylpyridinylamino-based DFG-in/αC-helix-out B-Raf inhibitors: Applying mutant versus wild-type B-Raf selectivity indices for compound profiling” [Bioorg. Med. Chem. 24 (2016) 2215–2234]
Liu, Longbin, Lee, Matthew R., Kim, Joseph L., Whittington, Douglas A., Bregman, Howard, Hua, Zihao, Lewis, Richard T., Martin, Matthew W., Nishimura, Nobuko, Potashman, Michele, Yang, Kevin, Yi, Shuyan, Vaida, Karina R., Epstein, Linda F., Babij, Carol, Fernando, Manory, Carnahan, Josette, Norman, Mark H.
Published in Bioorganic & medicinal chemistry (01.07.2016)
Published in Bioorganic & medicinal chemistry (01.07.2016)
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Design, synthesis, and testing of an 6-0-linked series of benzimidazole based inhibitors of CDK5/p25
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Published in Bioorganic & medicinal chemistry (2011)
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Published in Bioorganic & medicinal chemistry (2011)
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Year of Publication 25.03.2022
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Year of Publication 02.01.2018
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PYRAZOLE AMIDE DERIVATIVE
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Year of Publication 30.11.2016
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