Search Results - "SHUANGHUA HU" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Initial SAR studies on apamin-displacing 2-aminothiazole blockers of calcium-activated small conductance potassium channels

Initial SAR studies on apamin-displacing 2-aminothiazole blockers of calcium-activated small conductance potassium channels

by Gentles, Robert G., Grant-Young, Katherine, Hu, Shuanghua, Huang, Yazhong, Poss, Michael A., Andres, Charles, Fiedler, Tracey, Knox, Ronald, Lodge, Nicholas, Weaver, C. David, Harden, David G.
Published in Bioorganic & medicinal chemistry (01.10.2008)

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Journal Article

Preliminary SAR studies on non-apamin-displacing 4-(aminomethylaryl)pyrrazolopyrimidine KCa channel blockers

Preliminary SAR studies on non-apamin-displacing 4-(aminomethylaryl)pyrrazolopyrimidine KCa channel blockers

by GENTLES, Robert G, SHUANGHUA HU, HARDEN, David G, YAZHONG HUANG, GRANT-YOUNG, Katherine, POSS, Michael A, ANDRES, Charles, FIEDLER, Tracey, KNOX, Ronald, LODGE, Nicholas, WEAVER, C. David
Published in Bioorganic & medicinal chemistry letters (15.10.2008)

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Journal Article

Identification of a Potent and Selective 5-HT6 Antagonist: One-Step Synthesis of (E)-3-(Benzenesulfonyl)-2- (methylsulfanyl)pyrido[1,2-a]pyrimidin- 4-ylidenamine from 2-(Benzenesulfonyl)-3,3- bis(methylsulfanyl)acrylonitrile

Identification of a Potent and Selective 5-HT6 Antagonist: One-Step Synthesis of (E)-3-(Benzenesulfonyl)-2- (methylsulfanyl)pyrido[1,2-a]pyrimidin- 4-ylidenamine from 2-(Benzenesulfonyl)-3,3- bis(methylsulfanyl)acrylonitrile

by Wu, Yong-Jin, He, Huan, Hu, Shuanghua, Huang, Yazhong, Scola, Paul M, Grant-Young, Katharine, Bertekap, Robert L, Wu, Dedong, Gao, Qi, Li, Yi, Klakouski, Cheryl, Westphal, Ryan S
Published in Journal of medicinal chemistry (06.11.2003)

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Journal Article

Total Synthesis of a Human Breast Tumor Associated Antigen

Total Synthesis of a Human Breast Tumor Associated Antigen

by Bilodeau, Mark T, Park, Tae Kyo, Hu, Shuanghua, Randolph, John T, Danishefsky, Samuel J, Livingston, Philip O, Zhang, Shengli
Published in Journal of the American Chemical Society (01.07.1995)

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Journal Article

Discovery of D1 Dopamine Receptor Positive Allosteric Modulators: Characterization of Pharmacology and Identification of Residues that Regulate Species Selectivity

Discovery of D1 Dopamine Receptor Positive Allosteric Modulators: Characterization of Pharmacology and Identification of Residues that Regulate Species Selectivity

by Lewis, Martin A, Hunihan, Lisa, Watson, John, Gentles, Robert G, Hu, Shuanghua, Huang, Yazhong, Bronson, Joanne, Macor, John E, Beno, Brett R, Ferrante, Meredith, Hendricson, Adam, Knox, Ronald J, Molski, Thaddeus F, Kong, Yan, Cvijic, Mary Ellen, Rockwell, Kristin L, Weed, Michael R, Cacace, Angela M, Westphal, Ryan S, Alt, Andrew, Brown, Jeffrey M
Published in The Journal of pharmacology and experimental therapeutics (01.09.2015)

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Journal Article

Structure activity relationship studies on chemically non-reactive glycine sulfonamide inhibitors of diacylglycerol lipase

Structure activity relationship studies on chemically non-reactive glycine sulfonamide inhibitors of diacylglycerol lipase

by Chupak, Louis S., Zheng, Xiaofan, Hu, Shuanghua, Huang, Yazhong, Ding, Min, Lewis, Martin A., Westphal, Ryan S., Blat, Yuval, McClure, Andrea, Gentles, Robert G.
Published in Bioorganic & medicinal chemistry (01.04.2016)

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Journal Article

Structure activity relationship studies of 3-arylsulfonyl-pyrido[1,2-a]pyrimidin-4-imines as potent 5-HT6 antagonists

Structure activity relationship studies of 3-arylsulfonyl-pyrido[1,2-a]pyrimidin-4-imines as potent 5-HT6 antagonists

by Hu, Shuanghua, Huang, Yazhong, Wu, Yong-Jin, He, Huan, Grant-Young, Katherine A., Bertekap, Robert L., Whiterock, Valerie, Brassil, Patrick, Lentz, Kimberley, Sivaprakasam, Prasanna, Langley, David R., Westphal, Ryan S., Scola, Paul M.
Published in Bioorganic & medicinal chemistry (01.03.2014)

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Journal Article

Peramivir Dry Powder Inhaler and Method of Preparing the Same

Peramivir Dry Powder Inhaler and Method of Preparing the Same

by Hu, Shuanghua, Miao, Dong
Year of Publication 16.02.2023

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Patent

Heterocyclic modification of a novel bicyclo[3.1.0]hexane NPY1 receptor antagonist

Heterocyclic modification of a novel bicyclo[3.1.0]hexane NPY1 receptor antagonist

by Luo, Guanglin, Chen, Ling, Hu, Shuanghua, Huang, Yazhong, Mattson, Gail, Iben, Lawrence G., Russell, John W., Clarke, Wendy J., Hogan, John B., Antal-Zimanyi, Ildiko, Poindexter, Graham S.
Published in Bioorganic & medicinal chemistry letters (01.07.2013)

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Journal Article

Preliminary SAR studies on non-apamin-displacing 4-(aminomethylaryl)pyrrazolopyrimidine K Ca channel blockers

Preliminary SAR studies on non-apamin-displacing 4-(aminomethylaryl)pyrrazolopyrimidine K Ca channel blockers

by Gentles, Robert G., Hu, Shuanghua, Huang, Yazhong, Grant-Young, Katherine, Poss, Michael A., Andres, Charles, Fiedler, Tracey, Knox, Ronald, Lodge, Nicholas, Weaver, C. David, Harden, David G.
Published in Bioorganic & medicinal chemistry letters (15.10.2008)

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Journal Article

Preliminary SAR studies on non-apamin-displacing 4- (aminomethylaryl)pyrrazolopyrimidine K sub(Ca) channel blockers

Preliminary SAR studies on non-apamin-displacing 4- (aminomethylaryl)pyrrazolopyrimidine K sub(Ca) channel blockers

by Gentles, Robert G, Hu, Shuanghua, Huang, Yazhong, Grant-Young, Katherine, Poss, Michael A, Andres, Charles, Fiedler, Tracey, Knox, Ronald, Lodge, Nicholas, Weaver, CDavid, Harden, David G
Published in Bioorganic & medicinal chemistry (01.10.2008)

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Journal Article

Discovery of a Novel Class of Bicyclo[3.1.0]hexanylpiperazines as Noncompetitive Neuropeptide Y Y1 Antagonists

Discovery of a Novel Class of Bicyclo[3.1.0]hexanylpiperazines as Noncompetitive Neuropeptide Y Y1 Antagonists

by Hu, Shuanghua, Huang, Yazhong, Deshpande, Milind, Luo, Guanglin, Bruce, Marc A, Chen, Ling, Mattson, Gail, Iben, Lawrence G, Zhang, Jie, Russell, John W, Clarke, Wendy J, Hogan, John B, Ortiz, Astrid, Flint, Oliver, Henwood, Andrew, Gao, Qi, Antal-Zimanyi, Ildiko, Poindexter, Graham S
Published in ACS medicinal chemistry letters (08.03.2012)

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Journal Article

Unbleachable rhodopsin with an 11-cis-locked eight-membered ring retinal: The visual transduction process

Unbleachable rhodopsin with an 11-cis-locked eight-membered ring retinal: The visual transduction process

by Hu, Shuanghua, Franklin, Paul J, Wang, Jun, Silva, Beatriz E. Ruiz, Derguini, Fadila, Nakanishi, Koji
Published in Biochemistry (Easton) (18.01.1994)

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Journal Article

A highly convergent total synthetic route to glycopeptides carrying a high-mannose core pentasaccharide domain N-linked to a natural peptide motif

A highly convergent total synthetic route to glycopeptides carrying a high-mannose core pentasaccharide domain N-linked to a natural peptide motif

by Danishefsky, SJ, Hu, S, Cirillo, PF, Eckhardt, M, Seeberger, PH
Published in Chemistry : a European journal (01.10.1997)

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Journal Article

A novel route to the 5,6-dihydro-4-h-thieno[3,2-b]pyrrol-5-one ring system involving an intermediate substituted-thiophene synthesis

A novel route to the 5,6-dihydro-4-h-thieno[3,2-b]pyrrol-5-one ring system involving an intermediate substituted-thiophene synthesis

by Hu, SH, Huang, YZ, Poss, MA, Gentles, RG
Published in Journal of heterocyclic chemistry (01.05.2005)

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Journal Article

Synthesis of retinals with eight- and nine-membered rings in the side chain. Models for rhodopsin photobleaching intermediates

Synthesis of retinals with eight- and nine-membered rings in the side chain. Models for rhodopsin photobleaching intermediates

by Caldwell, Charles G, Derguini, Fadila, Bigge, Christopher F, Chen, Arh Hwang, Hu, Shuanghua, Wang, Jun, Sastry, Lakshmi, Nakanishi, Koji
Published in Journal of organic chemistry (01.06.1993)

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Journal Article

Identification of a potent and selective 5-HT(6) antagonist: one-step synthesis of (E)-3-(benzenesulfonyl)-2- (methylsulfanyl)pyrido[1,2-a]pyrimidin-4-ylidenamine from 2-(benzenesulfonyl)-3,3-bis(methylsulfanyl)acrylonitrile

Identification of a potent and selective 5-HT(6) antagonist: one-step synthesis of (E)-3-(benzenesulfonyl)-2- (methylsulfanyl)pyrido[1,2-a]pyrimidin-4-ylidenamine from 2-(benzenesulfonyl)-3,3-bis(methylsulfanyl)acrylonitrile

by Wu, Yong-Jin, He, Huan, Hu, Shuanghua, Huang, Yazhong, Scola, Paul M, Grant-Young, Katharine, Bertekap, Robert L, Wu, Dedong, Gao, Qi, Li, Yi, Klakouski, Cheryl, Westphal, Ryan S
Published in Journal of medicinal chemistry (06.11.2003)

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Journal Article

Identification of a Potent and Selective 5-HT 6 Antagonist: One-Step Synthesis of ( E )-3-(Benzenesulfonyl)-2- (methylsulfanyl)pyrido[1,2- a ]pyrimidin- 4-ylidenamine from 2-(Benzenesulfonyl)-3,3- bis(methylsulfanyl)acrylonitrile

Identification of a Potent and Selective 5-HT 6 Antagonist: One-Step Synthesis of ( E )-3-(Benzenesulfonyl)-2- (methylsulfanyl)pyrido[1,2- a ]pyrimidin- 4-ylidenamine from 2-(Benzenesulfonyl)-3,3- bis(methylsulfanyl)acrylonitrile

by Wu, Yong-Jin, He, Huan, Hu, Shuanghua, Huang, Yazhong, Scola, Paul M., Grant-Young, Katharine, Bertekap, Robert L., Wu, Dedong, Gao, Qi, Li, Yi, Klakouski, Cheryl, Westphal, Ryan S.
Published in Journal of medicinal chemistry (01.11.2003)

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Journal Article

Preliminary SAR studies on non-apamin-displacing 4-(aminomethylaryl)pyrrazolopyrimidine K(Ca) channel blockers

Preliminary SAR studies on non-apamin-displacing 4-(aminomethylaryl)pyrrazolopyrimidine K(Ca) channel blockers

by Gentles, Robert G, Hu, Shuanghua, Huang, Yazhong, Grant-Young, Katherine, Poss, Michael A, Andres, Charles, Fiedler, Tracey, Knox, Ronald, Lodge, Nicholas, Weaver, C David, Harden, David G
Published in Bioorganic & medicinal chemistry letters (15.10.2008)

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Journal Article

DEFINING THE MOLECULAR RECOGNITION OF GLOBO-H (HUMAN BREAST-CANCER) ANTIGEN THROUGH PROBE STRUCTURES PREPARED BY TOTAL SYNTHESIS

DEFINING THE MOLECULAR RECOGNITION OF GLOBO-H (HUMAN BREAST-CANCER) ANTIGEN THROUGH PROBE STRUCTURES PREPARED BY TOTAL SYNTHESIS

by KIM, IJ, PARK, TK, HU, SH, ABRAMPAH, K, ZHANG, SL, LIVINGSTON, PO, DANISHEFSKY, SJ
Published in Journal of organic chemistry (01.12.1995)

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Journal Article