Discovery of A‑971432, An Orally Bioavailable Selective Sphingosine-1-Phosphate Receptor 5 (S1P5) Agonist for the Potential Treatment of Neurodegenerative Disorders
Hobson, Adrian D, Harris, Christopher M, van der Kam, Elizabeth L, Turner, Sean C, Abibi, Ayome, Aguirre, Ana L, Bousquet, Peter, Kebede, Tegest, Konopacki, Donald B, Gintant, Gary, Kim, Youngjae, Larson, Kelly, Maull, John W, Moore, Nigel S, Shi, Dan, Shrestha, Anurupa, Tang, Xiubo, Zhang, Peng, Sarris, Kathy K
Published in Journal of medicinal chemistry (10.12.2015)
Published in Journal of medicinal chemistry (10.12.2015)
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Journal Article
Bound To Shock: Protection from Lethal Endotoxemic Shock by a Novel, Nontoxic, Alkylpolyamine Lipopolysaccharide Sequestrant
SIL, Diptesh, SHRESTHA, Anurupa, CROMER, Jens R, ARORA, Shravan, DATTA, Apurba, DAVID, Sunil A, KIMBRELL, Matthew R, NGUYEN, Thuan B, ADISECHAN, Ashok K, BALAKRISHNA, Rajalakshmi, ABBO, Benjamin G, MALLADI, Subbalakshmi, MILLER, Kelly A, SHORT, Shannon
Published in Antimicrobial Agents and Chemotherapy (01.08.2007)
Published in Antimicrobial Agents and Chemotherapy (01.08.2007)
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Journal Article
The Chosen Few: Parallel Library Reaction Methodologies for Drug Discovery
Dombrowski, Amanda W, Aguirre, Ana L, Shrestha, Anurupa, Sarris, Kathy A, Wang, Ying
Published in Journal of organic chemistry (18.02.2022)
Published in Journal of organic chemistry (18.02.2022)
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Journal Article
Discovery of ABBV-3373, an Anti-TNF Glucocorticoid Receptor Modulator
Hobson, Adrian D., McPherson, Michael J., Hayes, Martin E., Goess, Christian, Li, Xiang, Zhou, Jian, Wang, Zhongyuan, Yu, Yajie, Yang, Jindong, Sun, Liang, Zhang, Qiang, Qu, Pei, Yang, Shi, Hernandez, Axel, Bryant, Shaughn H., Mathieu, Suzanne L., Bischoff, Agnieszka K., Fitzgibbons, Julia, Santora, Ling C., Wang, Lu, Fettis, Margaret M., Li, Xiaofeng, Marvin, Christopher C., Wang, Zhi, V. Patel, Meena, Schmidt, Diana L., Li, Tongmei, Randolph, John T., Henry, Rodger F., Graff, Candace, Tian, Yu, Aguirre, Ana L., Shrestha, Anurupa
Published in Journal of medicinal chemistry (08.12.2022)
Published in Journal of medicinal chemistry (08.12.2022)
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Journal Article
Design and Development of Glucocorticoid Receptor Modulators as Immunology Antibody–Drug Conjugate Payloads
Hobson, Adrian D, McPherson, Michael J, Waegell, Wendy, Goess, Christian A, Stoffel, Robert H, Li, Xiang, Zhou, Jian, Wang, Zhongyuan, Yu, Yajie, Hernandez, Axel, Bryant, Shaughn H, Mathieu, Suzanne L, Bischoff, Agnieszka K, Fitzgibbons, Julia, Pawlikowska, Martyna, Puthenveetil, Sujiet, Santora, Ling C, Wang, Lu, Wang, Lu, Marvin, Christopher C, Hayes, Martin E, Shrestha, Anurupa, Sarris, Kathy A, Li, Biqin
Published in Journal of medicinal chemistry (24.03.2022)
Published in Journal of medicinal chemistry (24.03.2022)
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Journal Article
Discovery of GLPG2737, a Potent Type 2 Corrector of CFTR for the Treatment of Cystic Fibrosis in Combination with a Potentiator and a Type 1 Co-corrector
Pizzonero, Mathieu, Akkari, Rhalid, Bock, Xavier, Gosmini, Romain, De Lemos, Elsa, Duthion, Béranger, Newsome, Gregory, Mai, Thi-Thu-Trang, Roques, Virginie, Jary, Hélène, Lefrancois, Jean-Michel, Cherel, Laetitia, Quenehen, Vanessa, Babel, Marielle, Merayo, Nuria, Bienvenu, Natacha, Mammoliti, Oscar, Coti, Ghjuvanni, Palisse, Adeline, Cowart, Marlon, Shrestha, Anurupa, Greszler, Stephen, Van Der Plas, Steven, Jansen, Koen, Claes, Pieter, Jans, Mia, Gees, Maarten, Borgonovi, Monica, De Wilde, Gert, Conrath, Katja
Published in Journal of medicinal chemistry (11.04.2024)
Published in Journal of medicinal chemistry (11.04.2024)
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Journal Article
Discovery of ABBV-3373, an Anti-TNF Glucocorticoid Receptor Modulator Immunology Antibody Drug Conjugate
Hobson, Adrian D., McPherson, Michael J., Hayes, Martin E., Goess, Christian, Li, Xiang, Zhou, Jian, Wang, Zhongyuan, Yu, Yajie, Yang, Jindong, Sun, Liang, Zhang, Qiang, Qu, Pei, Yang, Shi, Hernandez, Axel, Bryant, Shaughn H., Mathieu, Suzanne L., Bischoff, Agnieszka K., Fitzgibbons, Julia, Santora, Ling C., Wang, Lu, Wang, Lu, Fettis, Margaret M., Li, Xiaofeng, Marvin, Christopher C., Wang, Zhi, Patel, Meena V., Schmidt, Diana L., Li, Tongmei, Randolph, John T., Henry, Rodger F., Graff, Candace, Tian, Yu, Aguirre, Ana L., Shrestha, Anurupa
Published in Journal of medicinal chemistry (08.12.2022)
Published in Journal of medicinal chemistry (08.12.2022)
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Journal Article
Correction to “Design and Development of Glucocorticoid Receptor Modulators as Immunology Antibody–Drug Conjugate Payloads”
Hobson, Adrian D., McPherson, Michael J., Waegell, Wendy, Goess, Christian A., Stoffel, Robert H., Li, Xiang, Zhou, Jian, Wang, Zhongyuan, Yu, Yajie, Hernandez, Axel, Bryant, Shaughn H., Mathieu, Suzanne L., Bischoff, Agnieszka K., Fitzgibbons, Julia, Pawlikowska, Martyna, Puthenveetil, Sujiet, Santora, Ling C., Wang, Lu, Wang, Lu, Marvin, Christopher C., Hayes, Martin E., Shrestha, Anurupa, Sarris, Kathy A., Li, Biqin
Published in Journal of medicinal chemistry (27.04.2023)
Published in Journal of medicinal chemistry (27.04.2023)
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Journal Article
Discovery of Small Molecule Interleukin 17A Inhibitors with Novel Binding Mode and Stoichiometry: Optimization of DNA-Encoded Chemical Library Hits to In Vivo Active Compounds
Ramos, Ashley L., Goedken, Eric R., Frank, Kristine E., Argiriadi, Maria A., Bazzaz, Sana, Bian, Zhiguo, Brown, Jesse T. C., Centrella, Paolo A., Chen, Hui-Ju, Disch, Jeremy S., Donner, Pamela L., Duignan, David B., Gikunju, Diana, Greszler, Stephen N., Guié, Marie-Aude, Habeshian, Sevan, Hartl, Hajnalka E., Hein, Christopher D., Hutchins, Charles W., Jetson, Rachael, Keefe, Anthony D., Khan, Hasan, Li, Huan-Qiu, Olszewski, Allison, Ortiz Cardona, Benjamin J., Osuma, Augustine, Panchal, Sanjay C., Phelan, Ryan, Qiu, Wei, Shotwell, J. Brad, Shrestha, Anurupa, Srikumaran, Myron, Su, Zhi, Sun, Chaohong, Upadhyay, Anup K., Wood, Michael D., Wu, Haihong, Zhang, Ruijie, Zhang, Ying, Zhao, Gang, Zhu, Haizhong, Webster, Matthew P.
Published in Journal of medicinal chemistry (25.04.2024)
Published in Journal of medicinal chemistry (25.04.2024)
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Journal Article
Correction to “Discovery of ABBV-3373, an Anti-TNF Glucocorticoid Receptor Modulator Immunology Antibody Drug Conjugate”
Hobson, Adrian D., McPherson, Michael J., Hayes, Martin E., Goess, Christian, Li, Xiang, Zhou, Jian, Wang, Zhongyuan, Yu, Yajie, Yang, Jindong, Sun, Liang, Zhang, Qiang, Qu, Pei, Yang, Shi, Hernandez, Axel, Bryant, Shaughn H., Mathieu, Suzanne L., Bischoff, Agnieszka K., Fitzgibbons, Julia, Santora, Ling C., Wang, Lu, Wang, Lu, Fettis, Margaret M., Li, Xiaofeng, Marvin, Christopher C., Wang, Zhi, Patel, Meena V., Schmidt, Diana L., Li, Tongmei, Randolph, John T., Henry, Rodger F., Graff, Candace, Tian, Yu, Aguirre, Ana L., Shrestha, Anurupa
Published in Journal of medicinal chemistry (27.04.2023)
Published in Journal of medicinal chemistry (27.04.2023)
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Journal Article
SAR and characterization of non-substrate isoindoline urea inhibitors of nicotinamide phosphoribosyltransferase (NAMPT)
Curtin, Michael L., Heyman, H. Robin, Clark, Richard F., Sorensen, Bryan K., Doherty, George A., Hansen, T. Matthew, Frey, Robin R., Sarris, Kathy A., Aguirre, Ana L., Shrestha, Anurupa, Tu, Noah, Woller, Kevin, Pliushchev, Marina A., Sweis, Ramzi F., Cheng, Min, Wilsbacher, Julie L., Kovar, Peter J., Guo, Jun, Cheng, Dong, Longenecker, Kenton L., Raich, Diana, Korepanova, Alla V., Soni, Nirupama B., Algire, Mikkel A., Richardson, Paul L., Marin, Violeta L., Badagnani, Ilaria, Vasudevan, Anil, Buchanan, F. Greg, Maag, David, Chiang, Gary G., Tse, Chris, Michaelides, Michael R.
Published in Bioorganic & medicinal chemistry letters (01.08.2017)
Published in Bioorganic & medicinal chemistry letters (01.08.2017)
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Journal Article
Synthesis and Pharmacology of (Pyridin-2-yl)methanol Derivatives as Novel and Selective Transient Receptor Potential Vanilloid 3 Antagonists
Gomtsyan, Arthur, Schmidt, Robert G, Bayburt, Erol K, Gfesser, Gregory A, Voight, Eric A, Daanen, Jerome F, Schmidt, Diana L, Cowart, Marlon D, Liu, Huaqing, Altenbach, Robert J, Kort, Michael E, Clapham, Bruce, Cox, Phil B, Shrestha, Anurupa, Henry, Rodger, Whittern, David N, Reilly, Regina M, Puttfarcken, Pamela S, Brederson, Jill-Desiree, Song, Ping, Li, Bin, Huang, Susan M, McDonald, Heath A, Neelands, Torben R, McGaraughty, Steve P, Gauvin, Donna M, Joshi, Shailen K, Banfor, Patricia N, Segreti, Jason A, Shebley, Mohamad, Faltynek, Connie R, Dart, Michael J, Kym, Philip R
Published in Journal of medicinal chemistry (26.05.2016)
Published in Journal of medicinal chemistry (26.05.2016)
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Journal Article
Pharmacokinetics of DS‐96, an Alkylpolyamine Lipopolysaccharide Sequestrant, in Rodents
Shrestha, Anurupa, Li, Rongti, Sil, Diptesh, Pardeshi, Neha N., Schwarting, Nancy, Schorno, Karl S., Rajewski, Roger A., Datta, Apurba, David, Sunil A.
Published in Journal of pharmaceutical sciences (01.12.2008)
Published in Journal of pharmaceutical sciences (01.12.2008)
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N-설포닐화 피라졸로[3,4-b]피리딘-6-카복스아미드 및 사용 방법
AKKARI RHALID, BROWN BRIAN S, BOCK XAVIER MARIE, HOUSSEMAN CHRISTOPHER GAETAN, PATEL SACHIN V, JI JIANGUO, DE BLIECK ANN, KYM PHILIP R, SHRESTHA ANURUPA, WANG XUEQING, GFESSER GREGORY A, SWIFT ELIZABETH C, ALVEY LUKE JONATHAN, PALISSE ADELINE MARIE ELISE, NEWSOME GREGORY JOHN ROBERT, PIZZONERO MATHIEU RAFAEL, DESROY NICOLAS, MERAYO NURIA MERAYO, CLAES PIETER ISABELLE ROGER, GOSMINI ROMAIN LUC MARIE, DUTHION BERANGER, MENET CHRISTEL JEANNE MARIE, DE LEMOS ELSA, LEFRANCOIS JEAN MICHEL, MAMMOLITI OSCAR, VAN DER PLAS STEVEN EMIEL, JANSEN KOEN KAREL, COWART MARLON D
Year of Publication 20.07.2018
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Year of Publication 20.07.2018
Patent
N-sulfonylated pyrazolo[3,4-b]pyridin-6-carboxamides and method of use
Alvey, Luke Jonathan, Mammoliti, Oscar, Desroy, Nicolas, Wang, Xueqing, Cowart, Marlon D, Patel, Sachin V, Duthion, Béranger, Merayo, Nuria Merayo, De Lemos, Elsa, Swift, Elizabeth C, Palisse, Adeline Marie Elise, Pizzonero, Mathieu Rafaël, Jansen, Koen Karel, Shrestha, Anurupa, Newsome, Gregory John Robert, De Blieck, Ann, Gfesser, Gregory A, Gosmini, Romain, Claes, Pieter, Bock, Xavier Marie, Menet, Christel Jeanne Marie, Akkari, Rhalid, Brown, Brian S, Housseman, Christopher Gaëtan, Lefrancois, Jean-Michel, Van Der Plas, Steven Emiel, Ji, Jianguo, Kym, Philip R
Year of Publication 31.03.2023
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Year of Publication 31.03.2023
Patent
N-sulfonylated pyrazolo[3,4-b]pyridin-6-carboxamides and method of use
Alvey, Luke Jonathan, Mammoliti, Oscar, Desroy, Nicolas, Wang, Xueqing, Cowart, Marlon D, Patel, Sachin V, Duthion, Béranger, Merayo, Nuria Merayo, De Lemos, Elsa, Swift, Elizabeth C, Palisse, Adeline Marie Elise, Claes, Pieter Isabelle Roger, Gosmini, Romain Luc Marie, Pizzonero, Mathieu Rafaël, Jansen, Koen Karel, Shrestha, Anurupa, Newsome, Gregory John Robert, De Blieck, Ann, Gfesser, Gregory A, Bock, Xavier Marie, Menet, Christel Jeanne Marie, Akkari, Rhalid, Brown, Brian S, Housseman, Christopher Gaëtan, Lefrancois, Jean-Michel, Van Der Plas, Steven Emiel, Ji, Jianguo, Kym, Philip R
Year of Publication 09.12.2021
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Year of Publication 09.12.2021
Patent
N-sulfonylated pyrazolo[3,4-b]pyridin-6-carboxamides and method of use
Alvey, Luke Jonathan, Mammoliti, Oscar, Desroy, Nicolas, Wang, Xueqing, Cowart, Marlon D, Patel, Sachin V, Duthion, Béranger, Merayo, Nuria Merayo, De Lemos, Elsa, Swift, Elizabeth C, Palisse, Adeline Marie Elise, Claes, Pieter Isabelle Roger, Gosmini, Romain Luc Marie, Pizzonero, Mathieu Rafaël, Jansen, Koen Karel, Shrestha, Anurupa, Newsome, Gregory John Robert, De Blieck, Ann, Gfesser, Gregory A, Bock, Xavier Marie, Menet, Christel Jeanne Marie, Akkari, Rhalid, Brown, Brian S, Housseman, Christopher Gaëtan, Lefrancois, Jean-Michel, Van Der Plas, Steven Emiel, Ji, Jianguo, Kym, Philip R
Year of Publication 20.05.2021
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Year of Publication 20.05.2021
Patent
N-SULFONYLATED PYRAZOLO(3,4-B)PYRIDIN-6-CARBOXAMIDES AND METHOD OF USE
MAMMOLITI Oscar, ALVEY Luke Jonathan, MERAYO Nuria Merayo, NEWSOME Gregory John Robert, AKKARI Rhalid, GOSMINI Romain Luc Marie, BROWN Brian S, DE BLIECK Ann, COWART Marlon D, LEFRANCOIS Jean-Michel, MENET Christel Jeanne Marie, SWIFT Elizabeth C, JI Jianguo, PATEL Sachin V, PIZZONERO Mathieu Rafael, KYM Philip R, VAN DER PLAS Steven Emiel, CLAES Pieter Isabelle Roger, HOUSSEMAN Christopher Gaetan, GFESSER Gregory A, BOCK Xavier Marie, DESROY Nicolas, DE LEMOS Elsa, JANSEN Koen Karel, PALISSE Adeline Marie Elise, SHRESTHA Anurupa, WANG Xueqing, DUTHION Beranger
Year of Publication 29.01.2021
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Year of Publication 29.01.2021
Patent