Eribulin penetrates brain tumor tissue and prolongs survival of mice harboring intracerebral glioblastoma xenografts
Takahashi, Masamichi, Miki, Shunichiro, Fujimoto, Kenji, Fukuoka, Kohei, Matsushita, Yuko, Maida, Yoshiko, Yasukawa, Mami, Hayashi, Mitsuhiro, Shinkyo, Raku, Kikuchi, Kiyomi, Mukasa, Akitake, Nishikawa, Ryo, Tamura, Kenji, Narita, Yoshitaka, Hamada, Akinobu, Masutomi, Kenkichi, Ichimura, Koichi
Published in Cancer science (01.07.2019)
Published in Cancer science (01.07.2019)
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Factors Influencing ADME properties of therapeutic antisense oligonucleotides: physicochemical characteristics and beyond
Jiang, Rongrong, Hooshfar, Shirin, Rebecca Eno, Marsha, Yun, Cassandra, Sonego Zimmermann, Estevan, Shinkyo, Raku
Published in Current drug metabolism (01.01.2023)
Published in Current drug metabolism (01.01.2023)
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Conversion of 7-Dehydrocholesterol to 7-Ketocholesterol Is Catalyzed by Human Cytochrome P450 7A1 and Occurs by Direct Oxidation without an Epoxide Intermediate
Shinkyo, Raku, Xu, Libin, Tallman, Keri A., Cheng, Qian, Porter, Ned A., Guengerich, F. Peter
Published in The Journal of biological chemistry (23.09.2011)
Published in The Journal of biological chemistry (23.09.2011)
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Metabolism of mono- and dichloro-dibenzo-p-dioxins by Phanerochaete chrysosporium cytochromes P450
Kasai, Noriyuki, Ikushiro, Shin-ichi, Shinkyo, Raku, Yasuda, Kaori, Hirosue, Shinji, Arisawa, Akira, Ichinose, Hirofumi, Wariishi, Hiroyuki, Sakaki, Toshiyuki
Published in Applied microbiology and biotechnology (01.03.2010)
Published in Applied microbiology and biotechnology (01.03.2010)
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Molecular Cloning and Characterization of CYP719, a Methylenedioxy Bridge-forming Enzyme That Belongs to a Novel P450 Family, from cultured Coptis japonica Cells
Ikezawa, Nobuhiro, Tanaka, Masaru, Nagayoshi, Masanori, Shinkyo, Raku, Sakaki, Toshiyuki, Inouye, Kuniyo, Sato, Fumihiko
Published in The Journal of biological chemistry (03.10.2003)
Published in The Journal of biological chemistry (03.10.2003)
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Metabolism of vitamin D by human microsomal CYP2R1
Shinkyo, Raku, Sakaki, Toshiyuki, Kamakura, Masaki, Ohta, Miho, Inouye, Kuniyo
Published in Biochemical and biophysical research communications (05.11.2004)
Published in Biochemical and biophysical research communications (05.11.2004)
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Structure-Based Design of a Highly Active Vitamin D Hydroxylase from Streptomyces griseolus CYP105A1
Hayashi, Keiko, Sugimoto, Hiroshi, Shinkyo, Raku, Yamada, Masato, Ikeda, Shinnosuke, Ikushiro, Shinichi, Kamakura, Masaki, Shiro, Yoshitsugu, Sakaki, Toshiyuki
Published in Biochemistry (Easton) (18.11.2008)
Published in Biochemistry (Easton) (18.11.2008)
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Requirements for human iPS cell-derived hepatocytes as an alternative to primary human hepatocytes for assessing absorption, distribution, metabolism, excretion and toxicity of pharmaceuticals
Araki, Tetsuro, Iwazaki, Norihiko, Ishiguro, Naoki, Sakamoto, Atsushi, Nagata, Keisuke, Ohbuchi, Masato, Moriguchi, Hiroyuki, Motoi, Makiko, Shinkyo, Raku, Homma, Toshiki, Sakamoto, Sakae, Iwase, Yumiko, Ise, Ryota, Nakanishi, Yasuharu, Uto, Masahiro, Inoue, Tomoaki
Published in Fundamental Toxicological Sciences (2016)
Published in Fundamental Toxicological Sciences (2016)
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cDNA cloning and characterization of feline CYP1A1 and CYP1A2
Tanaka, Nagako, Miyasho, Taku, Shinkyo, Raku, Sakaki, Toshiyuki, Yokota, Hiroshi
Published in Life sciences (1973) (25.11.2006)
Published in Life sciences (1973) (25.11.2006)
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Metabolism of polychlorinated dibenzo-p-dioxins by cytochrome P450 BM-3 and its mutant
Sulistyaningdyah, W.T, Ogawa, J, Li, Q.S, Shinkyo, R, Sakaki, T, Inouye, K, Schmid, R.D, Shimizu, S
Published in Biotechnology letters (01.12.2004)
Published in Biotechnology letters (01.12.2004)
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Rat cytochrome P450-mediated transformation of dichlorodibenzo-p-dioxins by recombinant white-rot basidiomycete Coriolus hirsutus
ORIHARA, Kanami, YAMAZAKI, Takashi, SHINKYO, Raku, SAKAKI, Toshiyuki, INOUYE, Kuniyo, TSUKAMOTO, Akira, SUGIURA, Jun, SHISHIDO, Kazuo
Published in Applied microbiology and biotechnology (01.11.2005)
Published in Applied microbiology and biotechnology (01.11.2005)
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SEQUENTIAL METABOLISM OF 2,3,7-TRICHLORODIBENZO-P-DIOXIN (2,3,7-triCDD) BY CYTOCHROME P450 AND UDP-GLUCURONOSYLTRANSFERASE IN HUMAN LIVER MICROSOMES
KASAI, Noriyuki, SAKAKI, Toshiyuki, SHINKYO, Raku, IKUSHIRO, Shin-Ichi, LYANAGI, Takashi, KAMAO, Maya, OKANO, Toshio, OHTA, Miho, INOUYE, Kuniyo
Published in Drug metabolism and disposition (01.08.2004)
Published in Drug metabolism and disposition (01.08.2004)
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A new paradigm for drug-induced torsadogenic risk assessment using human iPS cell-derived cardiomyocytes
Ando, Hiroyuki, Yoshinaga, Takashi, Yamamoto, Wataru, Asakura, Keiichi, Uda, Takaaki, Taniguchi, Tomohiko, Ojima, Atsuko, Shinkyo, Raku, Kikuchi, Kiyomi, Osada, Tomoharu, Hayashi, Seiji, Kasai, Chieko, Miyamoto, Norimasa, Tashibu, Hiroyuki, Yamazaki, Daiju, Sugiyama, Atsushi, Kanda, Yasunari, Sawada, Kohei, Sekino, Yuko
Published in Journal of pharmacological and toxicological methods (01.03.2017)
Published in Journal of pharmacological and toxicological methods (01.03.2017)
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Insight into functional diversity of cytochrome P450 in the white-rot basidiomycete Phanerochaete chrysosporium: Involvement of versatile monooxygenase
Hirosue, Shinji, Tazaki, Masahiro, Hiratsuka, Nobuhiro, Yanai, Satoshi, Kabumoto, Hiroki, Shinkyo, Raku, Arisawa, Akira, Sakaki, Toshiyuki, Tsunekawa, Hiroshi, Johdo, Osamu, Ichinose, Hirofumi, Wariishi, Hiroyuki
Published in Biochemical and biophysical research communications (01.04.2011)
Published in Biochemical and biophysical research communications (01.04.2011)
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Crystal Structure of CYP105A1 (P450SU-1) in Complex with 1α,25-Dihydroxyvitamin D 3
Sugimoto, Hiroshi, Shinkyo, Raku, Hayashi, Keiko, Yoneda, Sachiyo, Yamada, Masato, Kamakura, Masaki, Ikushiro, Shin-ichi, Shiro, Yoshitsugu, Sakaki, Toshiyuki
Published in Biochemistry (Easton) (01.04.2008)
Published in Biochemistry (Easton) (01.04.2008)
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