A novel benzothiazole derivative YLT322 induces apoptosis via the mitochondrial apoptosis pathway in vitro with anti-tumor activity in solid malignancies
Xuejiao, Song, Yong, Xia, Ningyu, Wang, Lidan, Zhang, Xuanhong, Shi, Youzhi, Xu, Tinghong, Ye, Yaojie, Shi, Yongxia, Zhu, Luoting, Yu
Published in PloS one (30.05.2013)
Published in PloS one (30.05.2013)
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Application and Study of ROCK Inhibitors in Pulmonary Fibrosis: Recent Developments and Future Perspectives
Xie, Yuting, Yue, Lin, Shi, Yaojie, Su, Xingping, Gan, Cailing, Liu, Hongyao, Xue, Taixiong, Ye, Tinghong
Published in Journal of medicinal chemistry (13.04.2023)
Published in Journal of medicinal chemistry (13.04.2023)
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Structure-guided discovery of novel potent and efficacious proteolysis targeting chimera (PROTAC) degrader of BRD4
Xiang, Wang, Wang, Qiwei, Ran, Kai, Ren, Jing, Shi, Yaojie, Yu, Luoting
Published in Bioorganic chemistry (01.10.2021)
Published in Bioorganic chemistry (01.10.2021)
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Design, synthesis and biological evaluation of 7-((7H-pyrrolo[2,3-d]pyrimidin-4-yl)oxy)-2,3-dihydro-1H-inden-1-one derivatives as potent FAK inhibitors for the treatment of ovarian cancer
Wei, Wei, Feng, Zhanzhan, Liu, Zhihao, Li, Xinyue, He, Hualong, Ran, Kai, Shi, Yaojie, Zhu, Yongxia, Ye, Tinghong, Gao, Chao, Wang, Ningyu, Yu, Luoting
Published in European journal of medicinal chemistry (15.01.2022)
Published in European journal of medicinal chemistry (15.01.2022)
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Design and synthesis of the first PARP-1 and proteasome dual inhibitors to treat breast cancer
He, Hualong, Yang, Wan, Shi, Yaojie, Chen, Xin, Chen, Xinyi, Hu, Xiang, Li, Xinyue, Yang, Yingyue, Liu, Zhihao, Ye, Tinghong, Wang, Ningyu, Yu, Luoting
Published in European journal of medicinal chemistry (15.01.2024)
Published in European journal of medicinal chemistry (15.01.2024)
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Synthesis and biological evaluation of (1,2,4)triazole[4,3-a]pyridine derivatives as potential therapeutic agents for concanavalin A-induced hepatitis
Shi, Yaojie, Wang, Qianqian, Rong, Juan, Ren, Jing, Song, Xuejiao, Fan, Xiaoli, Shen, Mengyi, Xia, Yong, Wang, Ningyu, Liu, Zhihao, Hu, Quanfang, Ye, Tinghong, Yu, Luoting
Published in European journal of medicinal chemistry (01.10.2019)
Published in European journal of medicinal chemistry (01.10.2019)
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Selective inhibition of EZH2 by ZLD1039 blocks H3K27methylation and leads to potent anti-tumor activity in breast cancer
Song, Xuejiao, Gao, Tiantao, Wang, Ningyu, Feng, Qiang, You, Xinyu, Ye, Tinghong, Lei, Qian, Zhu, Yongxia, Xiong, Menghua, Xia, Yong, Yang, Fangfang, Shi, Yaojie, Wei, Yuquan, Zhang, Lidan, Yu, Luoting
Published in Scientific reports (12.02.2016)
Published in Scientific reports (12.02.2016)
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Journal Article
Synthesis and biological evaluation of (E)-4-(3-arylvinyl-1H-indazol-6-yl)pyrimidin-2-amine derivatives as PLK4 inhibitors for the treatment of breast cancer
Liu, Zhihao, Lei, Qian, Wei, Wei, Xiong, Lu, Shi, Yaojie, Yan, Guoyi, Gao, Chao, Ye, Tinghong, Wang, Ningyu, Yu, Luoting
Published in RSC advances (01.01.2017)
Published in RSC advances (01.01.2017)
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Journal Article
Benzothiazinethione is a potent preclinical candidate for the treatment of drug-resistant tuberculosis
Gao, Chao, Peng, Cuiting, Shi, Yaojie, You, Xinyu, Ran, Kai, Xiong, Lu, Ye, Ting-hong, Zhang, Lidan, Wang, Ningyu, Zhu, Yongxia, Liu, Kun, Zuo, Weiqiong, Yu, Luoting, Wei, Yuquan
Published in Scientific reports (13.07.2016)
Published in Scientific reports (13.07.2016)
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Journal Article
Selective and efficient synthesis of trans-arylvinylboronates and trans-hetarylvinylboronates using palladium catalyzed cross-couplingElectronic supplementary information (ESI) available: See DOI: 10.1039/c6nj03984g
Liu, Zhihao, Wei, Wei, Xiong, Lu, Feng, Qiang, Shi, Yaojie, Wang, Ningyu, Yu, Luoting
Year of Publication 10.04.2017
Year of Publication 10.04.2017
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Journal Article
Identification of novel 2-aminothiazole conjugated nitrofuran as antitubercular and antibacterial agents
Ran, Kai, Gao, Chao, Deng, Hongxia, Lei, Qian, You, Xinyu, Wang, Ningyu, Shi, Yaojie, Liu, Zhihao, Wei, Wei, Peng, Cuiting, Xiong, Lu, Xiao, Kunjie, Yu, Luoting
Published in Bioorganic & medicinal chemistry letters (01.08.2016)
Published in Bioorganic & medicinal chemistry letters (01.08.2016)
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Journal Article
Corrigendum: Selective inhibition of EZH2 by ZLD1039 blocks H3K27methylation and leads to potent anti-tumor activity in breast cancer
Song, Xuejiao, Gao, Tiantao, Wang, Ningyu, Feng, Qiang, You, Xinyu, Ye, Tinghong, Lei, Qian, Zhu, Yongxia, Xiong, Menghua, Xia, Yong, Yang, Fangfang, Shi, Yaojie, Wei, Yuquan, Zhang, Lidan, Yu, Luoting
Published in Scientific reports (29.04.2016)
Published in Scientific reports (29.04.2016)
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A novel small-molecule YLT256 inhibits proliferation and induces apoptosis both in vitro and in vivo in solid tumors
Deng, Hongxia, Zeng, Jun, Zhu, Yongxia, Ye, Tinghong, Xia, Yong, Shi, Yaojie, Wang, Ningyu, Zhang, Lidan, Song, Xuejiao, Zuo, Weiqiong, Gao, Tiantao, Yu, Luoting
Published in Biomedicine & pharmacotherapy (01.07.2016)
Published in Biomedicine & pharmacotherapy (01.07.2016)
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Journal Article
Correction: Corrigendum: Selective inhibition of EZH2 by ZLD1039 blocks H3K27methylation and leads to potent anti-tumor activity in breast cancer
Song, Xuejiao, Gao, Tiantao, Wang, Ningyu, Feng, Qiang, You, Xinyu, Ye, Tinghong, Lei, Qian, Zhu, Yongxia, Xiong, Menghua, Xia, Yong, Yang, Fangfang, Shi, Yaojie, Wei, Yuquan, Zhang, Lidan, Yu, Luoting
Published in Scientific reports (29.04.2016)
Published in Scientific reports (29.04.2016)
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Journal Article
Synthesis and biological evaluation of (E)-4-(3-arylvinyl-1H-indazol-6-yl)pyrimidin-2-amine derivatives as PLK4 inhibitors for the treatment of breast cancerElectronic supplementary information (ESI) available. See DOI: 10.1039/c7ra02518a
Liu, Zhihao, Lei, Qian, Wei, Wei, Xiong, Lu, Shi, Yaojie, Yan, Guoyi, Gao, Chao, Ye, Tinghong, Wang, Ningyu, Yu, Luoting
Year of Publication 24.05.2017
Year of Publication 24.05.2017
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