Substituted 4‑(Thiazol-5-yl)-2-(phenylamino)pyrimidines Are Highly Active CDK9 Inhibitors: Synthesis, X‑ray Crystal Structures, Structure–Activity Relationship, and Anticancer Activities
Shao, Hao, Shi, Shenhua, Huang, Shiliang, Hole, Alison J, Abbas, Abdullahi Y, Baumli, Sonja, Liu, Xiangrui, Lam, Frankie, Foley, David W, Fischer, Peter M, Noble, Martin, Endicott, Jane A, Pepper, Chris, Wang, Shudong
Published in Journal of medicinal chemistry (14.02.2013)
Published in Journal of medicinal chemistry (14.02.2013)
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Comparative Structural and Functional Studies of 4‑(Thiazol-5-yl)-2-(phenylamino)pyrimidine-5-carbonitrile CDK9 Inhibitors Suggest the Basis for Isotype Selectivity
Hole, Alison J, Baumli, Sonja, Shao, Hao, Shi, Shenhua, Huang, Shiliang, Pepper, Chris, Fischer, Peter M, Wang, Shudong, Endicott, Jane A, Noble, Martin E
Published in Journal of medicinal chemistry (14.02.2013)
Published in Journal of medicinal chemistry (14.02.2013)
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Synthesis, structure–activity relationship and biological evaluation of 2,4,5-trisubstituted pyrimidine CDK inhibitors as potential anti-tumour agents
Shao, Hao, Shi, Shenhua, Foley, David W., Lam, Frankie, Abbas, Abdullah Y., Liu, Xiangrui, Huang, Shiliang, Jiang, Xiangrui, Baharin, Nadiah, Fischer, Peter M., Wang, Shudong
Published in European journal of medicinal chemistry (01.12.2013)
Published in European journal of medicinal chemistry (01.12.2013)
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In vitro antitumor mechanism of a novel cyclin-dependent kinase inhibitor CDKI-83
Liu, Xiangrui, Lam, Frankie, Shi, Shenhua, Fischer, Peter M., Wang, Shudong
Published in Investigational new drugs (01.06.2012)
Published in Investigational new drugs (01.06.2012)
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Abstract 697: Synthesis and biological evaluation of 2,4,5-substituted pyrimidines as highly selective CDK9 inhibitors for cancer treatment
Shao, Hao, Foley, David, Abbas, Abdullahi Y., Hole, Alison J., Huang, Shiliang, Shi, Shenhua, Baumli, Sonja, Bradshaw, Tracey D., Noble, Martin, Endicott, Jane A., Pepper, Chris, Wang, Shudong, Fischer, Peter M.
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Published in Cancer research (Chicago, Ill.) (15.04.2013)
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Fragmentation study of hexanitrostilbene by ion trap multiple mass spectrometry and analysis by liquid chromatography/mass spectrometry
Fu, Xiaofang, Zhang, Yong, Shi, Shenhua, Gao, Fei, Wen, Dawei, Li, Wei, Liao, Yiping, Liu, Huwei
Published in Rapid communications in mass spectrometry (01.01.2006)
Published in Rapid communications in mass spectrometry (01.01.2006)
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