Design of Selective PARP‑1 Inhibitors and Antitumor Studies
Zhang, Yiting, Li, Xiangqian, Liu, Fang, Bai, Xiaoyi, Liu, Xiaochun, Sun, Hao, Gao, Chenxia, Lin, Yuxi, Xing, Pan, Zhu, Jiqiang, Liu, Ruihua, Wang, Zemin, Dai, Jiajia, Shi, Dayong
Published in Journal of medicinal chemistry (22.05.2024)
Published in Journal of medicinal chemistry (22.05.2024)
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Journal Article
Design, synthesis and biological evaluation of bromophenol-thiazolylhydrazone hybrids inhibiting the interaction of translation initiation factors eIF4E/eIF4G as multifunctional agents for cancer treatment
Wang, Lijun, Guo, Chuanlong, Li, Xiuxue, Yu, Xuemin, Li, Xiangqian, Xu, Kuo, Jiang, Bo, Jia, Xiaoling, Li, Chao, Shi, Dayong
Published in European journal of medicinal chemistry (01.09.2019)
Published in European journal of medicinal chemistry (01.09.2019)
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Journal Article
BTH-8, a novel poly (ADP-ribose) polymerase-1 (PARP-1) inhibitor, causes DNA double-strand breaks and exhibits anticancer activities in vitro and in vivo
Guo, Chuanlong, Zhang, Fan, Wu, Xiaochen, Yu, Xuemin, Wu, Xianggen, Shi, Dayong, Wang, Lijun
Published in International journal of biological macromolecules (01.05.2020)
Published in International journal of biological macromolecules (01.05.2020)
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Journal Article
Selectivity, cell permeability and oral availability studies of novel bromophenol derivative HPN as protein tyrosine phosphatase 1B inhibitor
Luo, Jiao, Xu, Qi, Jiang, Bo, Zhang, Renshuai, Jia, Xiaoling, Li, Xiangqian, Wang, Lijun, Guo, Chuanlong, Wu, Ning, Shi, Dayong
Published in British journal of pharmacology (01.01.2018)
Published in British journal of pharmacology (01.01.2018)
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Journal Article
AcOH-mediated aerobic oxidative synthesis of 2-thioalkylbenzothiazoles via a three-component reaction
Li, Xiaowei, Li, Yuxiu, Liu, Ruihua, Wang, Zemin, Li, Xiangqian, Shi, Dayong
Published in Tetrahedron letters (25.06.2020)
Published in Tetrahedron letters (25.06.2020)
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Journal Article
Antidiabetic activity in vitro and in vivo of BDB, a selective inhibitor of protein tyrosine phosphatase 1B, from Rhodomela confervoides
Luo, Jiao, Zheng, Meiling, Jiang, Bo, Li, Chao, Guo, Shuju, Wang, Lijun, Li, Xiangqian, Yu, Rilei, Shi, Dayong
Published in British journal of pharmacology (01.10.2020)
Published in British journal of pharmacology (01.10.2020)
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Journal Article
The chemical constituents from red alga Gymnogongrus flabelliformis Harv
Yuan, Zhaohui, Han, Lijun, Su, Hua, Shi, Dayong, Sun, Jie, Li, Shuai, Shi, Jiangong
Published in Chinese journal of oceanology and limnology (01.05.2008)
Published in Chinese journal of oceanology and limnology (01.05.2008)
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Journal Article
Zinc-doped copper oxide nanocomposites reverse temozolomide resistance in glioblastoma by inhibiting AKT and ERK1/2
Wu, Ning, Zhang, Chunyun, Wang, Changhui, Song, Lairong, Yao, Weicheng, Gedanken, Aharon, Lin, Xiukun, Shi, Dayong
Published in Nanomedicine (London, England) (01.06.2018)
Published in Nanomedicine (London, England) (01.06.2018)
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Journal Article
Discovery and evaluation of the hybrid of bromophenol and saccharide as potent and selective protein tyrosine phosphatase 1B inhibitors
Zhang, Renshuai, Yu, Rilei, Xu, Qi, Li, Xiangqian, Luo, Jiao, Jiang, Bo, Wang, Lijun, Guo, Shuju, Wu, Ning, Shi, Dayong
Published in European journal of medicinal chemistry (07.07.2017)
Published in European journal of medicinal chemistry (07.07.2017)
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Journal Article
Highly Selective Protein Tyrosine Phosphatase Inhibitor, 2,2′,3,3′-Tetrabromo-4,4′,5,5′-tetrahydroxydiphenylmethane, Ameliorates Type 2 Diabetes Mellitus in BKS db Mice
Li, Chao, Luo, Jiao, Guo, Shuju, Jia, Xiaoling, Guo, Chuanlong, Li, Xiangqian, Xu, Qi, Shi, Dayong
Published in Molecular pharmaceutics (06.05.2019)
Published in Molecular pharmaceutics (06.05.2019)
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Journal Article
Phytochemical and chemotaxonomic study on Leathesia nana (Chordariaceae)
Xu, Kuo, Guo, Shuju, Jia, Xiaoling, Li, Xiang, Shi, Dayong
Published in Biochemical systematics and ecology (01.12.2018)
Published in Biochemical systematics and ecology (01.12.2018)
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Journal Article
Discovery of novel bromophenol 3,4-dibromo-5-(2-bromo-3,4-dihydroxy-6-(isobutoxymethyl)benzyl)benzene-1,2-diol as protein tyrosine phosphatase 1B inhibitor and its anti-diabetic properties in C57BL/KsJ-db/db mice
Jiang, Bo, Guo, Shuju, Shi, Dayong, Guo, Chao, Wang, Tao
Published in European journal of medicinal chemistry (01.06.2013)
Published in European journal of medicinal chemistry (01.06.2013)
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Journal Article
Cardamonin induces apoptosis by suppressing STAT3 signaling pathway in glioblastoma stem cells
Wu, Ning, Liu, Jia, Zhao, Xiangzhong, Yan, Zhiyong, Jiang, Bo, Wang, Lijun, Cao, Shousong, Shi, Dayong, Lin, Xiukun
Published in Tumor biology (01.12.2015)
Published in Tumor biology (01.12.2015)
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Journal Article
Iron-catalyzed alkynylation of tertiary aliphatic amines with 1-iodoalkynes to synthesize propargylamines
Ma, Lina, Shi, Xiaolin, Li, Xiaowei, Shi, Dayong
Published in ORGANIC CHEMISTRY FRONTIERS (21.12.2018)
Published in ORGANIC CHEMISTRY FRONTIERS (21.12.2018)
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Journal Article
A novel fluorinated thiosemicarbazone derivative- 2-(3,4-difluorobenzylidene) hydrazinecarbothioamide induces apoptosis in human A549 lung cancer cells via ROS-mediated mitochondria-dependent pathway
Zhao, Yue, Guo, Chuanlong, Wang, Lijun, Wang, Shuaiyu, Li, Xiangqian, Jiang, Bo, Wu, Ning, Guo, Shuju, Zhang, Renshuai, Liu, Kun, Shi, Dayong
Published in Biochemical and biophysical research communications (09.09.2017)
Published in Biochemical and biophysical research communications (09.09.2017)
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Journal Article
BOS-93, a novel bromophenol derivative, induces apoptosis and autophagy in human A549 lung cancer cells via PI3K/Akt/mTOR and MAPK signaling pathway
Guo, Chuanlong, Wang, Lijun, Zhao, Yue, Jiang, Bo, Luo, Jiao, Shi, Dayong
Published in Experimental and therapeutic medicine (01.05.2019)
Published in Experimental and therapeutic medicine (01.05.2019)
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Journal Article
Analysis of the seasonal water quality variation at the hydraulic junction of a dual-source water distribution system
Dong, Bowen, Huang, Hui, Wang, Chengyan, Zhang, Xiaolong, Gao, Chenyu, Su, Nan, Shi, Dayong, Ren, Jie
Published in RSC advances (28.05.2024)
Published in RSC advances (28.05.2024)
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Journal Article
Visible light-initiated radical 1,3-difunctionalization of β,γ-unsaturated ketones
Liu, Ruihua, Tian, Yang, Wang, Jie, Wang, Zemin, Li, Xiangqian, Zhao, Chenyang, Yao, Ruoyu, Li, Shuo, Yuan, Leifeng, Yang, Jinbo, Shi, Dayong
Published in Science advances (09.12.2022)
Published in Science advances (09.12.2022)
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Journal Article