BMS-201620: a selective beta 3 agonist
Washburn, W.N., Sun, C.-Q., Bisacchi, G., Wu, G., Cheng, P.T., Sher, P.M., Ryono, D., Gavai, A.V., Poss, K., Girotra, R.N., McCann, P.J., Mikkilineni, A.B., Dejneka, T.C., Wang, T.C., Merchant, Z., Morella, M., Arbeeny, C.M., Harper, T.W., Slusarchyk, D.A., Skwish, S., Russell, A.D., Allen, G.T., Tesfamariam, B., Frohlich, B.H., Abboa-Offei, B.E., Cap, M., Waldron, T.L., George, R.J., Young, D., Dickinson, K.E., Seymour, A.A.
Published in Bioorganic & medicinal chemistry letters (05.07.2004)
Published in Bioorganic & medicinal chemistry letters (05.07.2004)
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Beta 3 agonists. Part 1: evolution from inception to BMS-194449
Washburn, W.N., Sher, P.M., Poss, K.M., Girotra, R.N., McCann, P.J., Gavai, A.V., Mikkilineni, A.B., Mathur, A., Cheng, P., Dejneka, T.C., Sun, C.Q., Wang, T.C., Harper, T.W., Russell, A.D., Slusarchyk, D.A., Skwish, S., Allen, G.T., Hillyer, D.E., Frohlich, B.H., Abboa-Offei, B.E., Cap, M., Waldron, T.L., George, R.J., Tesfamariam, B., Ciosek, C.P., Ryono, D., Young, D.A., Dickinson, K.E., Seymour, A.A., Arbeeny, C.M., Gregg, R.E.
Published in Bioorganic & medicinal chemistry letters (03.12.2001)
Published in Bioorganic & medicinal chemistry letters (03.12.2001)
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Gavai, A V, Sher, P M, Mikkilineni, A B, Poss, K M, McCann, P J, Girotra, R N, Fisher, L G, Wu, G, Bednarz, M S, Mathur, A, Wang, T C, Sun, C Q, Slusarchyk, D A, Skwish, S, Allen, G T, Hillyer, D E, Frohlich, B H, Abboa-Offei, B E, Cap, M, Waldron, T L, George, R J, Tesfamariam, B, Harper, T W, Ciosek, Jr, C P, Young, D A, Dickinson, K E, Seymour, A A, Arbeeny, C M, Washburn, W N
Published in Bioorganic & medicinal chemistry letters (03.12.2001)
Published in Bioorganic & medicinal chemistry letters (03.12.2001)
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INTERPHENYLENE 7-OXABICYCLO[2.2.1]HEPTANE OXAZOLES - HIGHLY POTENT, SELECTIVE, AND LONG-ACTING THROMBOXANE A(2)-RECEPTOR ANTAGONISTS
MISRA, RN, BROWN, BR, SHER, PM, PATEL, MM, HALL, SE, HAN, WC, BARRISH, JC, KOCY, O, HARRIS, DN, GOLDENBERG, HJ, MICHEL, IM, SCHUMACHER, WA, WEBB, ML, MONSHIZADEGAN, H, OGLETREE, ML
Published in Journal of medicinal chemistry (14.05.1993)
Published in Journal of medicinal chemistry (14.05.1993)
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Addition of Benzylic and Allylic Organozinc and Grignard Reagents to Resin-Bound Imines To Provide α-Branched Secondary Amines Bearing a Wide Variety of Functional Groups. Utility in the Synthesis of β-3 Adrenergic Receptor Agonists
Wu, Gang, Cai, Zhen-Wei, Bednarz, Mark S, Kocy, Octavian R, Gavai, Ashvinikumar V, Godfrey, Jollie D, Washburn, William N, Poss, Michael A, Sher, Philip M
Published in Journal of combinatorial chemistry (01.01.2005)
Published in Journal of combinatorial chemistry (01.01.2005)
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C-ARYL GLUCOSIDE SGLT2 INHIBITORS AND METHOD C- SGLT2
SHER, PHILIP, M. PM, MENG, WEI W, WU, GANG G, ELLSWORTH, BRUCE B, WASHBURN, WILLIAM, N. WN
Year of Publication 11.12.2015
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Year of Publication 11.12.2015
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