Evolution of a Manufacturing Route to Omarigliptin, A Long-Acting DPP‑4 Inhibitor for the Treatment of Type 2 Diabetes
Chung, John Y. L, Scott, Jeremy P, Anderson, Camille, Bishop, Brian, Bremeyer, Nadine, Cao, Yang, Chen, Qinghao, Dunn, Robert, Kassim, Amude, Lieberman, David, Moment, Aaron J, Sheen, Faye, Zacuto, Michael
Published in Organic process research & development (20.11.2015)
Published in Organic process research & development (20.11.2015)
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The First Large-Scale Synthesis of MK-4305: A Dual Orexin Receptor Antagonist for the Treatment of Sleep Disorder
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Published in Organic process research & development (18.03.2011)
Published in Organic process research & development (18.03.2011)
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A Mild and Efficient One-Pot Synthesis of 2-Aminated Benzoxazoles and Benzothiazoles
Stewart, Gavin W, Baxter, Carl A, Cleator, Ed, Sheen, Faye J
Published in Journal of organic chemistry (17.04.2009)
Published in Journal of organic chemistry (17.04.2009)
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Process Development and Multikilogram-Scale Synthesis of a TRPV1 Antagonist
Cleator, Ed, Scott, Jeremy P, Avalle, Paulo, Bio, Matthew M, Brewer, Sarah E, Davies, Antony J, Gibb, Andrew D, Sheen, Faye J, Stewart, Gavin W, Wallace, Debra J, Wilson, Robert D
Published in Organic process research & development (20.12.2013)
Published in Organic process research & development (20.12.2013)
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Process Development and Large-Scale Synthesis of MK-6186, a Non-Nucleoside Reverse Transcriptase Inhibitor for the Treatment of HIV
Goodyear, Adrian, Linghu, Xin, Bishop, Brian, Chen, Cheng, Cleator, Ed, McLaughlin, Mark, Sheen, Faye J, Stewart, Gavin W, Xu, Yingju, Yin, Jingjun
Published in Organic process research & development (20.04.2012)
Published in Organic process research & development (20.04.2012)
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Practical Asymmetric Synthesis of a γ-Secretase Inhibitor Exploiting Substrate-Controlled Intramolecular Nitrile Oxide−Olefin Cycloaddition
Scott, Jeremy P, Oliver, Steven F, Brands, Karel M. J, Brewer, Sarah E, Davies, Antony J, Gibb, Andrew D, Hands, David, Keen, Stephen P, Sheen, Faye J, Reamer, Robert A, Wilson, Robert D, Dolling, Ulf-H
Published in Journal of organic chemistry (14.04.2006)
Published in Journal of organic chemistry (14.04.2006)
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Development of a Scaleable Synthesis of a Partial Nicotinic Acid Receptor Agonist
Wilson, Robert D, Cleator, Ed, Ashwood, Michael S, Bio, Matthew M, Brands, Karel M. J, Davies, Antony J, Dolling, Ulf-H, Emerson, Khateeta M, Gibb, Andrew D, Hands, David, McKeown, Arlene E, Oliver, Steven F, Reamer, Robert A, Sheen, Faye J, Stewart, Gavin W, Zhou, George X
Published in Organic process research & development (15.05.2009)
Published in Organic process research & development (15.05.2009)
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Regioselective coupling reactions of 2,4-diaminopyridine derivatives with aryl halides: the synthesis of elaborated pyridines
Bio, Matthew M., Cleator, Ed, Davies, Antony J., Hamilton, Simon E., Lawrence, Andrew, Sheen, Faye J., Stewart, Gavin W., Wilson, Robert D.
Published in Tetrahedron (31.10.2009)
Published in Tetrahedron (31.10.2009)
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NOVEL CRYSTALLINE FORMS OF A DIPEPTIDYL PEPTIDASE-IV INHIBITOR
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Year of Publication 20.03.2014
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Year of Publication 20.03.2014
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Regioselective coupling reactions of 2,4-diaminopyridine derivatives with aryl halides: the synthesis of elaborated pyridines: Modern Applications of Transition Metal Catalysis in Heterocycle Synthesis
BIO, Matthew M, CLEATOR, Ed, DAVIES, Antony J, HAMILTON, Simon E, LAWRENCE, Andrew, SHEEN, Faye J, STEWART, Gavin W, WILSON, Robert D
Published in Tetrahedron (2009)
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Published in Tetrahedron (2009)
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Regioselective synthesis of N-substituted-4-substituted isothiazolidine-1,1-dioxides
Cleator, Ed, Sheen, Faye J., Bio, Matthew M., Jos Brands, K.M., Davies, Antony J., Dolling, Ulf-H.
Published in Tetrahedron letters (19.06.2006)
Published in Tetrahedron letters (19.06.2006)
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PROCESS FOR PREPARING CHIRAL DIPEPTIDYL PEPTIDASE-IV INHIBITORS
ZACUTO MICHAEL J, CHEN QINGHAO, DUNN ROBERT F, TAN LUSHI, JANEY JACOB M, KUETHE JEFFREY T, BREMEYER NADINE, LIEBERMAN DAVID, MOMENT AARON J, SHEEN FAYE, SCOTT JEREMY
Year of Publication 20.03.2014
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Year of Publication 20.03.2014
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Process for the Prepartion of an Orexin Receptor Antagonist
Krska, Shane W, Baxter, Carl A, Wright, Timothy, Sheen, Faye, Stewart, Gavin, Strotman, Neil, Cleator, Edward, Wallace, Debra J
Year of Publication 07.10.2021
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Year of Publication 07.10.2021
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PROCESS FOR THE PREPARATION OF AN OREXIN RECEPTOR ANTAGONIST
KRSKA, Shane, W, SHEEN, Faye, BAXTER, Carl, A, CLEARTOR, Edward, WALLACE, Debra, J, STROTMAN, Neil, WRIGHT, Timothy, STEWART, Gavin
Year of Publication 10.01.2018
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Year of Publication 10.01.2018
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Novel crystalline forms of a dipeptidyl peptidase-IV inhibitor
MOMENT, AARON, KRUEGER, DAVIDA, BIFTU, TESFAYE, CHEN, PING, SHEEN, FAYE, ARROYO, ITZIA, ZHANG, YANFENG
Year of Publication 12.05.2016
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Year of Publication 12.05.2016
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Crystalline forms of a dipeptidyl peptidase-IV inhibitors
CHEN PING, BIFTU TESFAYE, KRUEGER DAVIDA, ARROYO ITZIA Z, ZHANG YANFENG, MOMENT AARON J, SHEEN FAYE
Year of Publication 10.11.2015
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Year of Publication 10.11.2015
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NOVEL CRYSTALLINE FORMS OF A DIPEPTIDYL PEPTIDASE-IV INHIBITORS
CHEN PING, BIFTU TESFAYE, KRUEGER DAVIDA, ARROYO ITZIA Z, ZHANG YANFENG, MOMENT AARON J, SHEEN FAYE
Year of Publication 09.04.2015
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Year of Publication 09.04.2015
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Crystalline forms of a dipeptidyl peptidase-IV inhibitor
CHEN PING, BIFTU TESFAYE, KRUEGER DAVIDA, MOMENT AARON, ZHANG YANFENG, ARROYO ITZIA, SHEEN FAYE
Year of Publication 25.11.2014
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Year of Publication 25.11.2014
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