Pharmacological characterization of potent and selective NaV1.7 inhibitors engineered from Chilobrachys jingzhao tarantula venom peptide JzTx-V
Moyer, Bryan D, Murray, Justin K, Ligutti, Joseph, Andrews, Kristin, Favreau, Philippe, Jordan, John B, Lee, Josie H, Liu, Dong, Long, Jason, Sham, Kelvin, Shi, Licheng, Stöcklin, Reto, Wu, Bin, Yin, Ruoyuan, Yu, Violeta, Zou, Anruo, Biswas, Kaustav, Miranda, Les P
Published in PloS one (01.05.2018)
Published in PloS one (01.05.2018)
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Journal Article
Quinolinone-based agonists of S1P1: Use of a N-scan SAR strategy to optimize in vitro and in vivo activity
Pennington, Lewis D., Croghan, Michael D., Sham, Kelvin K.C., Pickrell, Alexander J., Harrington, Paul E., Frohn, Michael J., Lanman, Brian A., Reed, Anthony B., Lee, Matthew R., Xu, Han, McElvain, Michele, Xu, Yang, Zhang, Xuxia, Fiorino, Michael, Horner, Michelle, Morrison, Henry G., Arnett, Heather A., Fotsch, Christopher, Tasker, Andrew S., Wong, Min, Cee, Victor J.
Published in Bioorganic & medicinal chemistry letters (01.01.2012)
Published in Bioorganic & medicinal chemistry letters (01.01.2012)
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Journal Article
Isoform-selective thiazolo[5,4-b]pyridine S1P1 agonists possessing acyclic amino carboxylate head-groups
Reed, Anthony B., Lanman, Brian A., Neira, Susana, Harrington, Paul E., Sham, Kelvin K.C., Frohn, Mike, Pickrell, Alexander J., Tasker, Andrew S., Gore, Anu, Fiorino, Mike, Itano, Andrea, McElvain, Michele, Middleton, Scot, Morrison, Henry, Xu, Han, Xu, Yang, Wong, Min, Cee, Victor J.
Published in Bioorganic & medicinal chemistry letters (15.02.2012)
Published in Bioorganic & medicinal chemistry letters (15.02.2012)
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Discovery of Highly Selective and Potent p38 Inhibitors Based on a Phthalazine Scaffold
Herberich, Brad, Cao, Guo-Qiang, Chakrabarti, Partha P, Falsey, James R, Pettus, Liping, Rzasa, Robert M, Reed, Anthony B, Reichelt, Andreas, Sham, Kelvin, Thaman, Maya, Wurz, Ryan P, Xu, Shimin, Zhang, Dawei, Hsieh, Faye, Lee, Matthew R, Syed, Rashid, Li, Vivian, Grosfeld, David, Plant, Matthew H, Henkle, Bradley, Sherman, Lisa, Middleton, Scot, Wong, Lu Min, Tasker, Andrew S
Published in Journal of medicinal chemistry (23.10.2008)
Published in Journal of medicinal chemistry (23.10.2008)
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Journal Article
Synthesis of Aromatic Heterocycles via Palladium-Catalyzed Annulation of Internal Alkynes
Larock, Richard C, Yum, Eul K, Doty, Mark J, Sham, Kelvin K. C
Published in Journal of organic chemistry (01.06.1995)
Published in Journal of organic chemistry (01.06.1995)
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Journal Article
The optimization of aminooxadiazoles as orally active inhibitors of Cdc7
Harrington, Paul E., Bourbeau, Matthew P., Fotsch, Christopher, Frohn, Michael, Pickrell, Alexander J., Reichelt, Andreas, Sham, Kelvin, Siegmund, Aaron C., Bailis, Julie M., Bush, Tammy, Escobar, Sonia, Hickman, Dean, Heller, Scott, Hsieh, Faye, Orf, Jessica N., Rong, Minqing, San Miguel, Tisha, Tan, Helming, Zalameda, Leeanne, Allen, John G.
Published in Bioorganic & medicinal chemistry letters (01.12.2013)
Published in Bioorganic & medicinal chemistry letters (01.12.2013)
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Journal Article
Optimization of a Potent, Orally Active S1P1 Agonist Containing a Quinolinone Core
Harrington, Paul E, Croghan, Michael D, Fotsch, Christopher, Frohn, Mike, Lanman, Brian A, Pennington, Lewis D, Pickrell, Alexander J, Reed, Anthony B, Sham, Kelvin K. C, Tasker, Andrew, Arnett, Heather A, Fiorino, Michael, Lee, Matthew R, McElvain, Michele, Morrison, Henry G, Xu, Han, Xu, Yang, Zhang, Xuxia, Wong, Min, Cee, Victor J
Published in ACS medicinal chemistry letters (12.01.2012)
Published in ACS medicinal chemistry letters (12.01.2012)
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Journal Article
4-Methoxy- N -[2-(trifluoromethyl)biphenyl-4-ylcarbamoyl]nicotinamide: A Potent and Selective Agonist of S1P 1
Pennington, Lewis D., Sham, Kelvin K. C., Pickrell, Alexander J., Harrington, Paul E., Frohn, Michael J., Lanman, Brian A., Reed, Anthony B., Croghan, Michael D., Lee, Matthew R., Xu, Han, McElvain, Michele, Xu, Yang, Zhang, Xuxia, Fiorino, Michael, Horner, Michelle, Morrison, Henry G., Arnett, Heather A., Fotsch, Christopher, Wong, Min, Cee, Victor J.
Published in ACS medicinal chemistry letters (13.10.2011)
Published in ACS medicinal chemistry letters (13.10.2011)
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Journal Article
First X-ray Cocrystal Structure of a Bacterial FabH Condensing Enzyme and a Small Molecule Inhibitor Achieved Using Rational Design and Homology Modeling
Daines, Robert A, Pendrak, Israil, Sham, Kelvin, Van Aller, Glenn S, Konstantinidis, Alex K, Lonsdale, John T, Janson, Cheryl A, Qiu, Xiayang, Brandt, Martin, Khandekar, Sanjay S, Silverman, Carol, Head, Martha S
Published in Journal of medicinal chemistry (02.01.2003)
Published in Journal of medicinal chemistry (02.01.2003)
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Journal Article
4-Methoxy-N-[2-(trifluoromethyl)biphenyl-4-ylcarbamoyl]nicotinamide: A Potent and Selective Agonist of S1P1
Pennington, Lewis D, Sham, Kelvin K. C, Pickrell, Alexander J, Harrington, Paul E, Frohn, Michael J, Lanman, Brian A, Reed, Anthony B, Croghan, Michael D, Lee, Matthew R, Xu, Han, McElvain, Michele, Xu, Yang, Zhang, Xuxia, Fiorino, Michael, Horner, Michelle, Morrison, Henry G, Arnett, Heather A, Fotsch, Christopher, Wong, Min, Cee, Victor J
Published in ACS medicinal chemistry letters (13.10.2011)
Published in ACS medicinal chemistry letters (13.10.2011)
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Journal Article
Purification of N-acetylgalactosamine-modified-oligonucleotides using orthogonal anion-exchange and mixed-mode chromatography approaches
Kazarian, Artaches A., Barnhart, Wesley, Long, Jason, Sham, Kelvin, Wu, Bin, Murray, Justin K.
Published in Journal of Chromatography A (04.01.2022)
Published in Journal of Chromatography A (04.01.2022)
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Journal Article
Purification of guanine-quadruplex using monolithic stationary phase under ion-exchange conditions
Kazarian, Artaches A., Barnhart, Wesley, Campuzano, Iain D.G., Cabrera, Jeremy, Fitch, Theodore, Long, Jason, Sham, Kelvin, Wu, Bin, Murray, Justin K.
Published in Journal of Chromatography A (20.12.2020)
Published in Journal of Chromatography A (20.12.2020)
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Journal Article
Plasma and Liver Protein Binding of N -Acetylgalactosamine-Conjugated Small Interfering RNA
Humphreys, Sara C, Thayer, Mai B, Lade, Julie M, Wu, Bin, Sham, Kelvin, Basiri, Babak, Hao, Yue, Huang, Xin, Smith, Richard, Rock, Brooke M
Published in Drug metabolism and disposition (01.10.2019)
Published in Drug metabolism and disposition (01.10.2019)
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Journal Article
Discovery of Tarantula Venom-Derived NaV1.7-Inhibitory JzTx‑V Peptide 5‑Br-Trp24 Analogue AM-6120 with Systemic Block of Histamine-Induced Pruritis
Wu, Bin, Murray, Justin K, Andrews, Kristin L, Sham, Kelvin, Long, Jason, Aral, Jennifer, Ligutti, Joseph, Amagasu, Shanti, Liu, Dong, Zou, Anruo, Min, Xiaoshan, Wang, Zhulun, Ilch, Christopher P, Kornecook, Thomas J, Lin, Min-Hwa Jasmine, Be, Xuhai, Miranda, Les P, Moyer, Bryan D, Biswas, Kaustav
Published in Journal of medicinal chemistry (08.11.2018)
Published in Journal of medicinal chemistry (08.11.2018)
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Journal Article
(E)-3-[6-[[(2,6-Dichlorophenyl)thio]methyl]-3-(2-phenylethoxy)-2-pyridinyl]-2- propenoic Acid: A High-Affinity Leukotriene B4 Receptor Antagonist with Oral Antiinflammatory Activity
Daines, Robert A, Chambers, Pamela A, Foley, James J, Griswold, Don E, Kingsbury, William D, Martin, Lenox D, Schmidt, Dulcie B, Sham, Kelvin K. C, Sarau, Henry M
Published in Journal of medicinal chemistry (13.09.1996)
Published in Journal of medicinal chemistry (13.09.1996)
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Journal Article
Pharmacological characterization of potent and selective Na.sub.V1.7 inhibitors engineered from Chilobrachys jingzhao tarantula venom peptide JzTx-V
Moyer, Bryan D, Murray, Justin K, Ligutti, Joseph, Andrews, Kristin, Favreau, Philippe, Jordan, John B, Lee, Josie H, Liu, Dong, Long, Jason, Sham, Kelvin, Shi, Licheng, Stöcklin, Reto, Wu, Bin, Yin, Ruoyuan, Yu, Violeta, Zou, Anruo, Biswas, Kaustav, Miranda, Les P
Published in PloS one (03.05.2018)
Published in PloS one (03.05.2018)
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Journal Article
Use of Cryopreserved Hepatocytes as Part of an Integrated Strategy to Characterize In Vivo Clearance for Peptide-Antibody Conjugate Inhibitors of Nav1.7 in Preclinical Species
Foti, Robert S, Biswas, Kaustav, Aral, Jennifer, Be, Xuhai, Berry, Loren, Cheng, Yuan, Conner, Kip, Falsey, James R, Glaus, Charles, Herberich, Brad, Hickman, Dean, Ikotun, Tayo, Li, Hongyan, Long, Jason, Huang, Liyue, Miranda, Les P, Murray, Justin, Moyer, Bryan, Netirojjanakul, Chawita, Nixey, Thomas E, Sham, Kelvin, Soto, Marcus, Tegley, Christopher M, Tran, Linh, Wu, Bin, Yin, Lin, Rock, Dan A
Published in Drug metabolism and disposition (01.10.2019)
Published in Drug metabolism and disposition (01.10.2019)
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Journal Article
Identification and Optimization of a Minor Allele-Specific siRNA to Prevent PNPLA3 I148M-Driven Nonalcoholic Fatty Liver Disease
Murray, Justin K, Long, Jason, Liu, Lei, Singh, Shivani, Pruitt, Danielle, Ollmann, Michael, Swearingen, Elissa, Hardy, Miki, Homann, Oliver, Wu, Bin, Holder, Jerry Ryan, Sham, Kelvin, Herberich, Brad, Lo, Mei-Chu, Dou, Hui, Shkumatov, Artem, Florio, Monica, Rulifson, Ingrid C
Published in Nucleic acid therapeutics (01.10.2021)
Published in Nucleic acid therapeutics (01.10.2021)
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Journal Article
Discovery of Tarantula Venom-Derived Na V 1.7-Inhibitory JzTx-V Peptide 5-Br-Trp24 Analogue AM-6120 with Systemic Block of Histamine-Induced Pruritis
Wu, Bin, Murray, Justin K, Andrews, Kristin L, Sham, Kelvin, Long, Jason, Aral, Jennifer, Ligutti, Joseph, Amagasu, Shanti, Liu, Dong, Zou, Anruo, Min, Xiaoshan, Wang, Zhulun, Ilch, Christopher P, Kornecook, Thomas J, Lin, Min-Hwa Jasmine, Be, Xuhai, Miranda, Les P, Moyer, Bryan D, Biswas, Kaustav
Published in Journal of medicinal chemistry (08.11.2018)
Published in Journal of medicinal chemistry (08.11.2018)
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Journal Article
Discovery of Tarantula Venom-Derived NaV 1.7-Inhibitory JzTx-V Peptide 5-Br-Trp24 Analogue AM-6120 with Systemic Block of Histamine-Induced Pruritis
Wu, Bin, Murray, Justin K., Andrews, Kristin L., Sham, Kelvin, Long, Jason, Aral, Jennifer, Ligutti, Joseph, Amagasu, Shanti, Liu, Dong, Zou, Anruo, Min, Xiaoshan, Wang, Zhulun, Ilch, Christopher P., Kornecook, Thomas J., Lin, Min-Hwa Jasmine, Be, Xuhai, Miranda, Les P., Moyer, Bryan D., Biswas, Kaustav
Published in Journal of medicinal chemistry (22.10.2018)
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Published in Journal of medicinal chemistry (22.10.2018)
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