Cys-Scanning Disulfide Crosslinking and Bayesian Modeling Probe the Transmembrane Signaling Mechanism of the Histidine Kinase, PhoQ
Molnar, Kathleen S., Bonomi, Massimiliano, Pellarin, Riccardo, Clinthorne, Graham D., Gonzalez, Gabriel, Goldberg, Shalom D., Goulian, Mark, Sali, Andrej, DeGrado, William F.
Published in Structure (London) (02.09.2014)
Published in Structure (London) (02.09.2014)
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Journal Article
Trastuzumab-MMAU Antibody-Auristatin Conjugates: Valine-Glucoserine Linker with Stabilized Maleimide Conjugation Improves In Vivo Efficacy and Tolerability
Goldberg, Shalom D, Satomaa, Tero, Aina, Olulanu, Aitio, Olli, Burke, Krista, Dudkin, Vadim, Geist, Brian, Irrechukwu, Onyi, Hänninen, Anna-Liisa, Heiskanen, Annamari, Helin, Jari, Hiltunen, Jukka O, Kinyamu-Akunda, Jacqueline, Klein, Donna M, Kohli, Neeraj, Kotiranta, Titta, Lähteenmäki, Tuula, Niemelä, Ritva, Pitkänen, Virve, Pynnönen, Henna, Rittase, William, Wiley, Kristen, Zhou, Junguo, Saarinen, Juhani
Published in Molecular cancer therapeutics (07.02.2024)
Published in Molecular cancer therapeutics (07.02.2024)
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Journal Article
Engineering a targeted delivery platform using Centyrins
Goldberg, Shalom D, Cardoso, Rosa M F, Lin, Tricia, Spinka-Doms, Tracy, Klein, Donna, Jacobs, Steven A, Dudkin, Vadim, Gilliland, Gary, O'Neil, Karyn T
Published in Protein engineering, design and selection (01.12.2016)
Published in Protein engineering, design and selection (01.12.2016)
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Journal Article
Site-specific protein modification using immobilized sortase in batch and continuous-flow systems
Witte, Martin D, Wu, Tongfei, Guimaraes, Carla P, Theile, Christopher S, Blom, Annet E M, Ingram, Jessica R, Li, Zeyang, Kundrat, Lenka, Goldberg, Shalom D, Ploegh, Hidde L
Published in Nature protocols (01.03.2015)
Published in Nature protocols (01.03.2015)
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Journal Article
A Strategy for Selective Deletion of Autoimmunity-Related T Cells by pMHC-Targeted Delivery
Goldberg, Shalom D., Felix, Nathan, McCauley, Michael, Eberwine, Ryan, Casta, Lou, Haskell, Kathleen, Lin, Tricia, Palovick, Elizabeth, Klein, Donna, Getts, Lori, Getts, Robert, Zhou, Mimi, Bansal-Pakala, Pratima, Dudkin, Vadim
Published in Pharmaceutics (13.10.2021)
Published in Pharmaceutics (13.10.2021)
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Journal Article
Engineered single- and multi-cell chemotaxis pathways in E. coli
Goulian, Mark, Goldberg, Shalom D, Derr, Paige, DeGrado, William F
Published in Molecular systems biology (16.06.2009)
Published in Molecular systems biology (16.06.2009)
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Journal Article
Mixed Quantum Mechanical/Molecular Mechanical (QM/MM) Study of the Deacylation Reaction in a Penicillin Binding Protein (PBP) versus in a Class C β-Lactamase
Gherman, Benjamin F, Goldberg, Shalom D, Cornish, Virginia W, Friesner, Richard A
Published in Journal of the American Chemical Society (23.06.2004)
Published in Journal of the American Chemical Society (23.06.2004)
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Journal Article
Determination of the Physiological Dimer Interface of the PhoQ Sensor Domain
Goldberg, Shalom D., Soto, Cinque S., Waldburger, Carey D., DeGrado, William F.
Published in Journal of molecular biology (13.06.2008)
Published in Journal of molecular biology (13.06.2008)
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Journal Article
Correlation between Catalytic Efficiency and the Transcription Read-Out in Chemical Complementation: A General Assay for Enzyme Catalysis
Sengupta, Debleena, Lin, Hening, Goldberg, Shalom D, Mahal, Jacqueline J, Cornish, Virginia W
Published in Biochemistry (Easton) (30.03.2004)
Published in Biochemistry (Easton) (30.03.2004)
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Journal Article
Investigation of the Mechanism of Resistance to Third-Generation Cephalosporins by Class C β-Lactamases by Using Chemical Complementation
Carter, Brian T., Lin, Hening, Goldberg, Shalom D., Althoff, Eric A., Raushel, Jessica, Cornish, Virginia W.
Published in Chembiochem : a European journal of chemical biology (01.11.2005)
Published in Chembiochem : a European journal of chemical biology (01.11.2005)
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Journal Article
Centyrin ligands for extrahepatic delivery of siRNA
Klein, Donna, Goldberg, Shalom, Theile, Christopher S., Dambra, Richard, Haskell, Kathleen, Kuhar, Elise, Lin, Tricia, Parmar, Rubina, Manoharan, Muthiah, Richter, Mark, Wu, Meizhen, Mendrola Zarazowski, Jeannine, Jadhav, Vasant, Maier, Martin A., Sepp-Lorenzino, Laura, O’Neil, Karyn, Dudkin, Vadim
Published in Molecular therapy (02.06.2021)
Published in Molecular therapy (02.06.2021)
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Journal Article
Evaluation of a Centyrin-Based Near-Infrared Probe for Fluorescence-Guided Surgery of Epidermal Growth Factor Receptor Positive Tumors
Mahalingam, Sakkarapalayam M, Dudkin, Vadim Y, Goldberg, Shalom, Klein, Donna, Yi, Fang, Singhal, Sunil, O’Neil, Karyn T, Low, Philip S
Published in Bioconjugate chemistry (15.11.2017)
Published in Bioconjugate chemistry (15.11.2017)
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Journal Article
LC/MS/MS Bioanalysis of Protein–Drug ConjugatesThe Importance of Incorporating Succinimide Hydrolysis Products
Shi, Chuan, Goldberg, Shalom, Lin, Tricia, Dudkin, Vadim, Widdison, Wayne, Harris, Luke, Wilhelm, Sharon, Jmeian, Yazen, Davis, Darryl, O’Neil, Karyn, Weng, Naidong, Jian, Wenying
Published in Analytical chemistry (Washington) (17.04.2018)
Published in Analytical chemistry (Washington) (17.04.2018)
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Journal Article
Abstract 4972: Detection of PSMA on circulating tumor cells from blood of prostate cancer patients using anti-PSMA Centyrin
Vaidya, Bhavesh, Vulfson, Peter, Sanders, Renouard, Klein, Donna, Goldberg, Shalom, Jacobs, Steve, Rao, Chandra
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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Journal Article
RADIOLABELING OF POLYPEPTIDE
THERESA M MCDEVITT, RHYS SALTER, VADIM DUDKIN, SHALOM GOLDBERG, JOSEPH ERHARDT
Year of Publication 06.06.2023
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Year of Publication 06.06.2023
Patent
Abstract LB-062: Evaluation of drug conjugation sites in an anti-EGFR Centyrin
Cardoso, Rosa, Goldberg, Shalom, Lin, Tricia, Spinka-Doms, Tracy, Klein, Donna, Jacobs, Steven, Gilliland, Gary, O’Neil, Karyn
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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Journal Article
Bioanalytical workflow for novel scaffold protein-drug conjugates: quantitation of total Centyrin protein, conjugated Centyrin and free payload for Centyrin-drug conjugate in plasma and tissue samples using liquid chromatography-tandem mass spectrometry
Shi, Chuan, Goldberg, Shalom, Lin, Tricia, Dudkin, Vadim, Widdison, Wayne, Harris, Luke, Wilhelm, Sharon, Jmeian, Yazen, Davis, Darryl, O'Neil, Karyn, Weng, Naidong, Jian, Wenying
Published in Bioanalysis (01.10.2018)
Published in Bioanalysis (01.10.2018)
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Journal Article
Abstract 3222: Structural evaluation of several antitumor Tencon variants
Cardoso, Rosa, Goldberg, Shalom, Luo, Jinquan, Barnakov, Alexander, Swift, Edward, Jacobs, Steven, Gilliland, Gary
Published in Cancer research (Chicago, Ill.) (01.10.2014)
Published in Cancer research (Chicago, Ill.) (01.10.2014)
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Journal Article