Spongipyran synthetic studies. Evolution of a scalable total synthesis of (+)-spongistatin 1
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Scalable Synthesis of the Potent HIV Inhibitor BMS-986001 by Non-Enzymatic Dynamic Kinetic Asymmetric Transformation (DYKAT)
Ortiz, Adrian, Benkovics, Tamas, Beutner, Gregory L., Shi, Zhongping, Bultman, Michael, Nye, Jeffrey, Sfouggatakis, Chris, Kronenthal, David R.
Published in Angewandte Chemie (International ed.) (08.06.2015)
Published in Angewandte Chemie (International ed.) (08.06.2015)
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Challenges with the Synthesis of a Macrocyclic Thioether Peptide: From Milligram to Multigram Using Solid Phase Peptide Synthesis (SPPS)
Kempson, James, Zhao, Rulin, Pawluczyk, Joseph, Wang, Bei, Zhang, Huiping, Hou, Xiaoping, Allen, Martin P., Wu, Dauh-Rurng, Li, Peng, Yip, Shiuhang, Smith, Aaron, Traeger, Sarah C., Huang, Stella, Cutrone, Jingfang, Mukherjee, Subha, Sfouggatakis, Chris, Poss, Michael, Scola, Paul M., Meanwell, Nicholas A., Carter, Percy H., Mathur, Arvind
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Development of Two Synthetic Approaches to an APJ Receptor Agonist Containing a Tetra-ortho-Substituted Biaryl Pyridone
Goldfogel, Matthew J, Jamison, Christopher R, Savage, Scott A, Haley, Matthew W, Mukherjee, Subha, Sfouggatakis, Chris, Gujjar, Manjunath, Mohan, Jayaraj, Rakshit, Souvik, Vaidyanathan, Rajappa
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Published in Organic process research & development (18.03.2022)
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Development of a Commercial Process for Deucravacitinib, a Deuterated API for TYK2 Inhibition
Treitler, Daniel S, Soumeillant, Maxime C, Simmons, Eric M, Lin, Dong, Inankur, Bahar, Rogers, Amanda J, Dummeldinger, Michael, Kolotuchin, Sergei, Chan, Collin, Li, Jun, Freitag, Adam, Lora Gonzalez, Federico, Smith, Michael J, Sfouggatakis, Chris, Wang, Jianji, Benkovics, Tamas, Deerberg, Joerg, Simpson, James H, Chen, Ke, Tymonko, Steven
Published in Organic process research & development (15.04.2022)
Published in Organic process research & development (15.04.2022)
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Scalable Asymmetric Synthesis of the All Cis Triamino Cyclohexane Core of BMS-813160
La Cruz, Thomas E, González-Bobes, Francisco, Eastgate, Martin D, Sfouggatakis, Chris, Zheng, Bin, Kopp, Nathaniel, Xiao, Yi, Fan, Yu, Galindo, Kay A, Pathirana, Charles, Galella, Michael A, Deerberg, Joerg
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Published in Journal of organic chemistry (18.02.2022)
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Development of a Concise Multikilogram Synthesis of LPA‑1 Antagonist BMS-986020 via a Tandem Borylation–Suzuki Procedure
Smith, Michael J, Lawler, Michael J, Kopp, Nathaniel, Mcleod, Douglas D, Davulcu, Akin H, Lin, Dong, Katipally, Kishta, Sfouggatakis, Chris
Published in Organic process research & development (17.11.2017)
Published in Organic process research & development (17.11.2017)
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Development of a Scalable Synthesis of BMS-978587 Featuring a Stereospecific Suzuki Coupling of a Cyclopropane Carboxylic Acid
Maity, Prantik, Reddy, V. V. Ramana, Mohan, Jayaraj, Korapati, Satish, Narayana, Harishkumar, Cherupally, Nagesh, Chandrasekaran, Sathishkumar, Ramachandran, Ravikumar, Sfouggatakis, Chris, Eastgate, Martin D, Simmons, Eric M, Vaidyanathan, Rajappa
Published in Organic process research & development (20.07.2018)
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N-N migration of a carbamoyl group in a pyrazole derivative revealed by NMR
Pathirana, Charles, Sfouggatakis, Chris, Palaniswamy, Venkatapuram
Published in Magnetic resonance in chemistry (01.03.2013)
Published in Magnetic resonance in chemistry (01.03.2013)
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Stereoselective Bulk Synthesis of CCR2 Antagonist BMS-741672: Assembly of an All-cis (S,R,R)-1,2,4-Triaminocyclohexane (TACH) Core via Sequential Heterogeneous Asymmetric Hydrogenations
Deerberg, Joerg, Prasad, Siva J., Sfouggatakis, Chris, Eastgate, Martin D., Fan, Yu, Chidambaram, Ramakrishnan, Sharma, Praveen, Li, Li, Schild, Richard, Muslehiddinoglu, Jale, Chung, Hyei-Jha, Leung, Simon, Rosso, Victor
Published in Organic process research & development (18.11.2016)
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Gram-Scale Synthesis of (+)-Spongistatin 1: Development of An Improved, Scalable Synthesis of the F-Ring Subunit, Fragment Union, and Final Elaboration
Smith, Amos B, Tomioka, Takashi, Risatti, Christina A, Sperry, Jeffrey B, Sfouggatakis, Chris
Published in Organic letters (02.10.2008)
Published in Organic letters (02.10.2008)
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Engaging senior management to improve the safety culture of a chemical development organization thru the SPYDR (Safety as Part of Your Daily Routine) lab visit program
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Year of Publication 13.07.2023
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Multicomponent Linchpin Couplings. Reaction of Dithiane Anions with Terminal Epoxides, Epichlorohydrin, and Vinyl Epoxides: Efficient, Rapid, and Stereocontrolled Assembly of Advanced Fragments for Complex Molecule Synthesis
Smith, Amos B, Pitram, Suresh M, Boldi, Armen M, Gaunt, Matthew J, Sfouggatakis, Chris, Moser, William H
Published in Journal of the American Chemical Society (26.11.2003)
Published in Journal of the American Chemical Society (26.11.2003)
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The Development of a Robust Process for a CRF1 Receptor Antagonist
Broxer, Sévrine, Fitzgerald, Monica A, Sfouggatakis, Chris, Defreese, Jessica L, Barlow, Evan, Powers, Gerald L, Peddicord, Michael, Su, Bao-Ning, Tai-Yuen, Yue, Pathirana, Charles, Sherbine, James P
Published in Organic process research & development (18.03.2011)
Published in Organic process research & development (18.03.2011)
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