Drug Resistance via Feedback Activation of Stat3 in Oncogene-Addicted Cancer Cells
Lee, Ho-June, Zhuang, Guanglei, Cao, Yi, Du, Pan, Kim, Hyo-Jin, Settleman, Jeff
Published in Cancer cell (11.08.2014)
Published in Cancer cell (11.08.2014)
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Cell line-based platforms to evaluate the therapeutic efficacy of candidate anticancer agents
Sharma, Sreenath V, Haber, Daniel A, Settleman, Jeff
Published in Nature reviews. Cancer (01.04.2010)
Published in Nature reviews. Cancer (01.04.2010)
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The Cancer Stem Cell Marker Aldehyde Dehydrogenase Is Required to Maintain a Drug-Tolerant Tumor Cell Subpopulation
RAHA, Debasish, WILSON, Timothy R, JING PENG, PETERSON, David, PENG YUE, EVANGELISTA, Marie, WILSON, Catherine, MERCHANT, Mark, SETTLEMAN, Jeff
Published in Cancer research (Chicago, Ill.) (01.07.2014)
Published in Cancer research (Chicago, Ill.) (01.07.2014)
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Transcriptional control of autophagy-lysosome function drives pancreatic cancer metabolism
Perera, Rushika M, Stoykova, Svetlana, Nicolay, Brandon N, Ross, Kenneth N, Fitamant, Julien, Boukhali, Myriam, Lengrand, Justine, Deshpande, Vikram, Selig, Martin K, Ferrone, Cristina R, Settleman, Jeff, Stephanopoulos, Gregory, Dyson, Nicholas J, Zoncu, Roberto, Ramaswamy, Sridhar, Haas, Wilhelm, Bardeesy, Nabeel
Published in Nature (London) (20.08.2015)
Published in Nature (London) (20.08.2015)
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Widespread potential for growth-factor-driven resistance to anticancer kinase inhibitors
WILSON, Timothy R, FRIDLYAND, Jane, RIBAS, Antoni, JIANG LI, MOFFAT, John, SUTHERLIN, Daniel P, KOEPPEN, Hartmut, MERCHANT, Mark, NEVE, Richard, SETTLEMAN, Jeff, YIBING YAN, PENUEL, Elicia, BURTON, Luciana, CHAN, Emily, JING PENG, EVA LIN, YULEI WANG, SOSMAN, Jeff
Published in Nature (London) (26.07.2012)
Published in Nature (London) (26.07.2012)
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Unprovoked Stabilization and Nuclear Accumulation of the Naked Mole-Rat p53 Protein
Deuker, Marian M, Lewis, Kaitlyn N, Ingaramo, Maria, Kimmel, Jacob, Buffenstein, Rochelle, Settleman, Jeff
Published in Scientific reports (24.04.2020)
Published in Scientific reports (24.04.2020)
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A Chromatin-Mediated Reversible Drug-Tolerant State in Cancer Cell Subpopulations
Sharma, Sreenath V., Lee, Diana Y., Li, Bihua, Quinlan, Margaret P., Takahashi, Fumiyuki, Maheswaran, Shyamala, McDermott, Ultan, Azizian, Nancy, Zou, Lee, Fischbach, Michael A., Wong, Kwok-Kin, Brandstetter, Kathleyn, Wittner, Ben, Ramaswamy, Sridhar, Classon, Marie, Settleman, Jeff
Published in Cell (02.04.2010)
Published in Cell (02.04.2010)
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Identification of a mutation in the extracellular domain of the Epidermal Growth Factor Receptor conferring cetuximab resistance in colorectal cancer
Montagut, Clara, Dalmases, Alba, Bellosillo, Beatriz, Crespo, Marta, Pairet, Silvia, Iglesias, Mar, Salido, Marta, Gallen, Manuel, Marsters, Scot, Tsai, Siao Ping, Minoche, André, Seshagiri, Somasekar, Somasekar, Seshagiri, Serrano, Sergi, Himmelbauer, Heinz, Bellmunt, Joaquim, Rovira, Ana, Settleman, Jeff, Bosch, Francesc, Albanell, Joan
Published in Nature medicine (01.02.2012)
Published in Nature medicine (01.02.2012)
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Repression of Stress-Induced LINE-1 Expression Protects Cancer Cell Subpopulations from Lethal Drug Exposure
Guler, Gulfem Dilek, Tindell, Charles Albert, Pitti, Robert, Wilson, Catherine, Nichols, Katrina, KaiWai Cheung, Tommy, Kim, Hyo-Jin, Wongchenko, Matthew, Yan, Yibing, Haley, Benjamin, Cuellar, Trinna, Webster, Joshua, Alag, Navneet, Hegde, Ganapati, Jackson, Erica, Nance, Tracy Leah, Giresi, Paul Garrett, Chen, Kuan-Bei, Liu, Jinfeng, Jhunjhunwala, Suchit, Settleman, Jeff, Stephan, Jean-Philippe, Arnott, David, Classon, Marie
Published in Cancer cell (14.08.2017)
Published in Cancer cell (14.08.2017)
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TAK1 Inhibition Promotes Apoptosis in KRAS-Dependent Colon Cancers
Singh, Anurag, Sweeney, Michael F., Yu, Min, Burger, Alexa, Greninger, Patricia, Benes, Cyril, Haber, Daniel A., Settleman, Jeff
Published in Cell (17.02.2012)
Published in Cell (17.02.2012)
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AXL inhibition sensitizes mesenchymal cancer cells to antimitotic drugs
Wilson, Catherine, Ye, Xiaofen, Pham, Thinh, Lin, Eva, Chan, Sara, McNamara, Erin, Neve, Richard M, Belmont, Lisa, Koeppen, Hartmut, Yauch, Robert L, Ashkenazi, Avi, Settleman, Jeff
Published in Cancer research (Chicago, Ill.) (15.10.2014)
Published in Cancer research (Chicago, Ill.) (15.10.2014)
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Cotargeting of MEK and PDGFR/STAT3 Pathways to Treat Pancreatic Ductal Adenocarcinoma
Sahu, Nisebita, Chan, Emily, Chu, Felix, Pham, Thinh, Koeppen, Hartmut, Forrest, William, Merchant, Mark, Settleman, Jeff
Published in Molecular cancer therapeutics (01.09.2017)
Published in Molecular cancer therapeutics (01.09.2017)
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Mechanisms of acquired resistance to targeted cancer therapies
Lackner, Mark R, Wilson, Timothy R, Settleman, Jeff
Published in Future oncology (London, England) (01.08.2012)
Published in Future oncology (London, England) (01.08.2012)
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Acquired Resistance of Non―Small Cell Lung Cancer Cells to MET Kinase Inhibition Is Mediated by a Switch to Epidermal Growth Factor Receptor Dependency
MCDERMOTT, Ultan, PUSAPATI, Raju V, CHRISTENSEN, James G, GRAY, Nathanael S, SETTLEMAN, Jeff
Published in Cancer research (Chicago, Ill.) (15.02.2010)
Published in Cancer research (Chicago, Ill.) (15.02.2010)
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Genome and transcriptome sequencing of lung cancers reveal diverse mutational and splicing events
Liu, Jinfeng, Lee, William, Jiang, Zhaoshi, Chen, Zhongqiang, Jhunjhunwala, Suchit, Haverty, Peter M, Gnad, Florian, Guan, Yinghui, Gilbert, Houston N, Stinson, Jeremy, Klijn, Christiaan, Guillory, Joseph, Bhatt, Deepali, Vartanian, Steffan, Walter, Kimberly, Chan, Jocelyn, Holcomb, Thomas, Dijkgraaf, Peter, Johnson, Stephanie, Koeman, Julie, Minna, John D, Gazdar, Adi F, Stern, Howard M, Hoeflich, Klaus P, Wu, Thomas D, Settleman, Jeff, de Sauvage, Frederic J, Gentleman, Robert C, Neve, Richard M, Stokoe, David, Modrusan, Zora, Seshagiri, Somasekar, Shames, David S, Zhang, Zemin
Published in Genome research (01.12.2012)
Published in Genome research (01.12.2012)
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Recent advances in pathway-targeted cancer drug therapies emerging from cancer genome analysis
Yauch, Robert L, Settleman, Jeff
Published in Current opinion in genetics & development (01.02.2012)
Published in Current opinion in genetics & development (01.02.2012)
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