Bax Channel Inhibitors Prevent Mitochondrion-mediated Apoptosis and Protect Neurons in a Model of Global Brain Ischemia
Hetz, Claudio, Vitte, Pierre-Alain, Bombrun, Agnes, Rostovtseva, Tatiana K., Montessuit, Sylvie, Hiver, Agnes, Schwarz, Matthias K., Church, Dennis J., Korsmeyer, Stanley J., Martinou, Jean-Claude, Antonsson, Bruno
Published in The Journal of biological chemistry (30.12.2005)
Published in The Journal of biological chemistry (30.12.2005)
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Journal Article
Identification and Characterization of Novel Small Molecules as Potent Inhibitors of the Plasmodial Calcium-Dependent Protein Kinase 1
Lemercier, Guillaume, Fernandez-Montalvan, Amaury, Shaw, Jeffrey P, Kugelstadt, Dominik, Bomke, Joerg, Domostoj, Mathias, Schwarz, Matthias K, Scheer, Alexander, Kappes, Barbara, Leroy, Didier
Published in Biochemistry (Easton) (14.07.2009)
Published in Biochemistry (Easton) (14.07.2009)
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Journal Article
Discovery of a New Class of Potent, Selective, and Orally Bioavailable CRTH2 (DP2) Receptor Antagonists for the Treatment of Allergic Inflammatory Diseases
Crosignani, Stefano, Page, Patrick, Missotten, Marc, Colovray, Véronique, Cleva, Christophe, Arrighi, Jean-François, Atherall, John, Macritchie, Jackie, Martin, Thierry, Humbert, Yves, Gaudet, Marilène, Pupowicz, Doris, Maio, Maurizio, Pittet, Pierre-André, Golzio, Lucia, Giachetti, Claudio, Rocha, Cynthia, Bernardinelli, Gérald, Filinchuk, Yaroslav, Scheer, Alexander, Schwarz, Matthias K, Chollet, André
Published in Journal of medicinal chemistry (10.04.2008)
Published in Journal of medicinal chemistry (10.04.2008)
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Journal Article
PI3Kγ inhibition: towards an 'aspirin of the 21st century'?
Schwarz, Matthias K, Rommel, Christian, Rückle, Thomas
Published in Nature reviews. Drug discovery (01.11.2006)
Published in Nature reviews. Drug discovery (01.11.2006)
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Journal Article
The p110δ structure: mechanisms for selectivity and potency of new PI(3)K inhibitors
Williams, Roger L, Berndt, Alex, Miller, Simon, Williams, Olusegun, Le, Daniel D, Houseman, Benjamin T, Pacold, Joseph I, Gorrec, Fabrice, Hon, Wai-Ching, Ren, Pingda, Liu, Yi, Rommel, Christian, Gaillard, Pascale, Rückle, Thomas, Schwarz, Matthias K, Shokat, Kevan M, Shaw, Jeffrey P
Published in Nature chemical biology (01.02.2010)
Published in Nature chemical biology (01.02.2010)
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Journal Article
Anti-chemokine small molecule drugs: a promising future?
Proudfoot, Amanda E I, Power, Christine A, Schwarz, Matthias K
Published in Expert opinion on investigational drugs (01.03.2010)
Published in Expert opinion on investigational drugs (01.03.2010)
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Journal Article
Blockade of PI3Kγ suppresses joint inflammation and damage in mouse models of rheumatoid arthritis
Rommel, Christian, Camps, Montserrat, Rückle, Thomas, Ji, Hong, Ardissone, Vittoria, Rintelen, Felix, Shaw, Jeffrey, Ferrandi, Chiara, Chabert, Christian, Gillieron, Corine, Françon, Bernard, Martin, Thierry, Gretener, Denise, Perrin, Dominique, Leroy, Didier, Vitte, Pierre-Alain, Hirsch, Emilio, Wymann, Matthias P, Cirillo, Rocco, Schwarz, Matthias K
Published in Nature medicine (01.09.2005)
Published in Nature medicine (01.09.2005)
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Journal Article
Solid-Phase Synthesis of 3,5-Disubstituted 2,3-Dihydro-1,5-benzothiazepin-4(5H)-ones
Schwarz, Matthias K, Tumelty, David, Gallop, Mark A
Published in Journal of organic chemistry (02.04.1999)
Published in Journal of organic chemistry (02.04.1999)
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Journal Article
Furan-2-ylmethylene Thiazolidinediones as Novel, Potent, and Selective Inhibitors of Phosphoinositide 3-Kinase γ
Pomel, Vincent, Klicic, Jasna, Covini, David, Church, Dennis D, Shaw, Jeffrey P, Roulin, Karen, Burgat-Charvillon, Fabienne, Valognes, Delphine, Camps, Montserrat, Chabert, Christian, Gillieron, Corinne, Françon, Bernard, Perrin, Dominique, Leroy, Didier, Gretener, Denise, Nichols, Anthony, Vitte, Pierre Alain, Carboni, Susanna, Rommel, Christian, Schwarz, Matthias K, Rückle, Thomas
Published in Journal of medicinal chemistry (29.06.2006)
Published in Journal of medicinal chemistry (29.06.2006)
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Journal Article
PI3Kγ inhibition blocks glomerulonephritis and extends lifespan in a mouse model of systemic lupus
Carrera, Ana C, Barber, Domingo F, Bartolomé, Almira, Hernandez, Carmen, Flores, Juana M, Redondo, Clara, Fernandez-Arias, Cristina, Camps, Montserrat, Rückle, Thomas, Schwarz, Matthias K, Rodríguez, Santiago, Martinez-A, Carlos, Balomenos, Dimitrios, Rommel, Christian
Published in Nature medicine (01.09.2005)
Published in Nature medicine (01.09.2005)
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Journal Article
Genetic and Pharmacological Targeting of Phosphoinositide 3-Kinase-γ Reduces Atherosclerosis and Favors Plaque Stability by Modulating Inflammatory Processes
FOUGERAT, Anne, GAYRAL, Stéphanie, PERRET, Bertrand, BRETON-DOUILLON, Monique, WYMANN, Matthias P, LAFFARGUE, Muriel, GOURDY, Pierre, SCHAMBOURG, Alexia, RÜCKLE, Thomas, SCHWARZ, Matthias K, ROMMEL, Christian, HIRSCH, Emilio, ARNAL, Jean-Francois, SALLES, Jean-Pierre
Published in Circulation (New York, N.Y.) (11.03.2008)
Published in Circulation (New York, N.Y.) (11.03.2008)
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Journal Article
Pharmacology of (2S,4Z)-N-[(2S)-2-Hydroxy-2-phenylethyl]-4-(methoxyimino) -1-[(2â²-methyl[1,1â²-biphenyl]-4-yl)carbonyl]-2-pyrrolidinecarboxamide, a New Potent and Selective Nonpeptide Antagonist of the Oxytocin Receptor
Cirillo, Rocco, Gillio Tos, Enrico, Schwarz, Matthias K, Quattropani, Anna, Scheer, Alexander, Missotten, Marc, Dorbais, Jerome, Nichols, Anthony, Borrelli, Francesco, Giachetti, Claudio, Golzio, Lucia, Marinelli, Paolo, Thomas, Russell J, Chevillard, Claude, Laurent, Florence, Portet, Karine, Barberis, Claude, Chollet, Andre
Published in The Journal of pharmacology and experimental therapeutics (01.07.2003)
Published in The Journal of pharmacology and experimental therapeutics (01.07.2003)
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Journal Article
Glycosaminoglycan analogs as a novel anti-inflammatory strategy
Severin, India C, Soares, Adriano, Hantson, Jennifer, Teixeira, Mauro, Sachs, Daniela, Valognes, Delphine, Scheer, Alexander, Schwarz, Matthias K, Wells, Timothy N C, Proudfoot, Amanda E I, Shaw, Jeffrey
Published in Frontiers in immunology (01.01.2012)
Published in Frontiers in immunology (01.01.2012)
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Journal Article
The p110δ structure: mechanisms for selectivity and potency of new PI(3)K inhibitors
Berndt, Alex, Miller, Simon, Williams, Olusegun, Le, Daniel D, Houseman, Benjamin T, Pacold, Joseph I, Gorrec, Fabrice, Hon, Wai-Ching, Ren, Pingda, Liu, Yi, Rommel, Christian, Gaillard, Pascale, Rückle, Thomas, Schwarz, Matthias K, Shokat, Kevan M, Shaw, Jeffrey P, Williams, Roger L
Published in Nature chemical biology (01.03.2010)
Published in Nature chemical biology (01.03.2010)
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Journal Article
Importance of phosphoinositide 3-kinase γ in the host defense against pneumococcal infection
MAUS, Ulrich A, BACKI, Myriam, MAUS, Regina, BOHLE, Rainer M, SEEGER, Werner, ROMMEL, Christian, HIRSCH, Emilio, LOHMEYER, Jürgen, PREISSNER, Klaus T, WINTER, Christine, SRIVASTAVA, Mrigank, SCHWARZ, Matthias K, RÜCKLE, Thomas, PATON, James C, BRILES, David, MACK, Matthias, WELTE, Tobias
Published in American journal of respiratory and critical care medicine (01.05.2007)
Published in American journal of respiratory and critical care medicine (01.05.2007)
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Journal Article
Arrest of preterm labor in rat and mouse by an oral and selective nonprostanoid antagonist of the prostaglandin F2α receptor (FP)
Cirillo, Rocco, PhD, Tos, Enrico Gillio, Page, Patrick, PhD, Missotten, Marc, Dipl Biol, Quattropani, Anna, PhD, Scheer, Alexander, PhD, Schwarz, Matthias K., PhD, Chollet, André, PhD
Published in American journal of obstetrics and gynecology (2007)
Published in American journal of obstetrics and gynecology (2007)
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Journal Article
The p110δ structure: mechanisms for selectivity and potency of new PI(3)K inhibitors
Berndt, Alex, Miller, Simon, Williams, Olusegun, Le, Daniel D, Houseman, Benjamin T, Pacold, Joseph I, Gorrec, Fabrice, Hon, Wai-Ching, Ren, Pingda, Liu, Yi, Rommel, Christian, Gaillard, Pascale, Rückle, Thomas, Schwarz, Matthias K, Shokat, Kevan M, Shaw, Jeffrey P, Williams, Roger L
Published in Nature chemical biology (01.04.2010)
Published in Nature chemical biology (01.04.2010)
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