Design and synthesis of potent, orally bioavailable dihydroquinazolinone inhibitors of p38 MAP kinase
Stelmach, John E., Liu, Luping, Patel, Sangita B., Pivnichny, James V., Scapin, Giovanna, Singh, Suresh, Hop, Cornelis E.C.A., Wang, Zhen, Strauss, John R., Cameron, Patricia M., Nichols, Elizabeth A., O'Keefe, Stephen J., O'Neill, Edward A., Schmatz, Dennis M., Schwartz, Cheryl D., Thompson, Chris M., Zaller, Dennis M., Doherty, James B.
Published in Bioorganic & medicinal chemistry letters (01.01.2003)
Published in Bioorganic & medicinal chemistry letters (01.01.2003)
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Synthesis and biological activity of quinolinone and dihydroquinolinone p38 MAP kinase inhibitors
Chen, Meng-Hsin, Fitzgerald, Patricia, Singh, Suresh B., O’Neill, Edward A., Schwartz, Cheryl D., Thompson, Chris M., O’Keefe, Stephen J., Zaller, Dennis M., Doherty, James B.
Published in Bioorganic & medicinal chemistry letters (15.03.2008)
Published in Bioorganic & medicinal chemistry letters (15.03.2008)
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Journal Article
SAR of 3,4-Dihydropyrido[3,2- d]pyrimidone p38 inhibitors
Liu, Luping, Stelmach, John E., Natarajan, Swaminathan R., Chen, Meng-Hsin, Singh, Suresh B., Schwartz, Cheryl D., Fitzgerald, Catherine E., O'Keefe, Stephen J., Zaller, Dennis M., Schmatz, Dennis M., Doherty, James B.
Published in Bioorganic & medicinal chemistry letters (17.11.2003)
Published in Bioorganic & medicinal chemistry letters (17.11.2003)
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Hybrid-Designed Inhibitors of p38 MAP Kinase Utilizing N-Arylpyridazinones
Colletti, Steven L, Frie, Jessica L, Dixon, Elizabeth C, Singh, Suresh B, Choi, Bernard K, Scapin, Giovanna, Fitzgerald, Catherine E, Kumar, Sanjeev, Nichols, Elizabeth A, O'Keefe, Stephen J, O'Neill, Edward A, Porter, Gene, Samuel, Koppara, Schmatz, Dennis M, Schwartz, Cheryl D, Shoop, Wesley L, Thompson, Chris M, Thompson, James E, Wang, Ruixiu, Woods, Andrea, Zaller, Dennis M, Doherty, James B
Published in Journal of medicinal chemistry (30.01.2003)
Published in Journal of medicinal chemistry (30.01.2003)
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Pyridazine based inhibitors of p38 MAPK
McIntyre, Charles J, Ponticello, Gerald S, Liverton, Nigel J, O’Keefe, Stephen J, O’Neill, Edward A, Pang, Margaret, Schwartz, Cheryl D, Claremon, David A
Published in Bioorganic & medicinal chemistry letters (25.02.2002)
Published in Bioorganic & medicinal chemistry letters (25.02.2002)
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p38MAP kinase inhibitors. Part 1: design and development of a new class of potent and highly selective inhibitors based on 3,4-dihydropyrido[3,2-d]pyrimidone scaffold
Natarajan, Swaminathan R, Wisnoski, David D, Singh, Suresh B, Stelmach, John E, O'Neill, Edward A, Schwartz, Cheryl D, Thompson, Chris M, Fitzgerald, Catherine E, O'Keefe, Stephen J, Kumar, Sanjeev, Hop, Cornelis E C A, Zaller, Dennis M, Schmatz, Dennis M, Doherty, James B
Published in Bioorganic & medicinal chemistry letters (20.01.2003)
Published in Bioorganic & medicinal chemistry letters (20.01.2003)
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SAR for MHC class II binding tetrapeptides: Correlation with potential binding site
Cunningham, Barry R, Rivetna, Meheryar, Tolman, Richard L, Flattery, Stacey J, Nichols, Elizabeth A, Schwartz, Cheryl D, Wicker, Linda S, Hermes, Jeffrey D, Jones, A.Brian
Published in Bioorganic & medicinal chemistry letters (07.01.1997)
Published in Bioorganic & medicinal chemistry letters (07.01.1997)
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L-156, 602, A C5a ANTAGONIST WITH A NOVEL CYCLIC HEXADEPSIPEPTIDE STRUCTURE FROM Streptomyces sp. MA6348: FERMENTATION, ISOLATION AND STRUCTURE DETERMINATION
HENSENS, OTTO D., BORRIS, ROBERT P., KOUPAL, LAWRENCE R., CALDWELL, CHARLES G., CURRIE, SARA A., HAIDRI, AKBER A., HOMNICK, CARL F., HONEYCUTT, SUSAN S., LINDENMAYER, SUSAN M., SCHWARTZ, CHERYL D., WEISSBERGER, BARBARA A., WOODRUFF, H. B., ZINK, DEBORAH L., ZITANO, LAURETTA, FIELDHOUSE, JILL M., ROLLINS, THOMAS, SPRINGER, MARTIN S., SPRINGER, JAMES P.
Published in Journal of antibiotics (1991)
Published in Journal of antibiotics (1991)
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NOVEL AND POTENT GASTRIN AND BRAIN CHOLECYSTOKININ ANTAGONISTS FROM Streptomyces olivaceus: TAXONOMY, FERMENTATION, ISOLATION, CHEMICAL CONVERSIONS, AND PHYSICO-CHEMICAL AND BIOCHEMICAL PROPERTIES
LAM, Y. K. TONY, BOGEN, DEBRA, CHANG, RAYMOND S., FAUST, KRISTINE A., HENSENS, OTTO D., ZINK, DEBORAH L., SCHWARTZ, CHERYL D., ZITANO, LORETTA, GARRITY, GEORGE M., GAGLIARDI, MAGDA M., CURRIE, SARA A., WOODRUFF, H. BOYD
Published in Journal of antibiotics (1991)
Published in Journal of antibiotics (1991)
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Journal Article
p38 MAP kinase inhibitors. part 1: design and development of a new class of potent and highly selective inhibitors based on 3,4-dihydropyrido[3,2- d]pyrimidone scaffold
Natarajan, Swaminathan R., Wisnoski, David D., Singh, Suresh B., Stelmach, John E., O'Neill, Edward A., Schwartz, Cheryl D., Thompson, Chris M., Fitzgerald, Catherine E., O'Keefe, Stephen J., Kumar, Sanjeev, Hop, Cornelis E.C.A., Zaller, Dennis M., Schmatz, Dennis M., Doherty, James B.
Published in Bioorganic & medicinal chemistry letters (01.01.2003)
Published in Bioorganic & medicinal chemistry letters (01.01.2003)
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Difficidin and oxydifficidin: Novel broad spectrum antibacterial antibiotics produced by Bacillus subtilis. I.Production, taxonomy and antibacterial activity
ZIMMERMAN, SHELDON B., SCHWARTZ, CHERYL D., MONAGHAN, RICHARD L., PELAK, BARBARA ANN, WEISSBERGER, BARBARA, GILFILLAN, EVEMARIE C., MOCHALES, SAGRARIO, HERNANDEZ, SEBASTIAN, CURRIE, SARA A., TEJERA, ENRIQUE, STAPLEY, EDWARD O.
Published in Journal of antibiotics (1987)
Published in Journal of antibiotics (1987)
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Journal Article
p38 MAP kinase inhibitors. Part1: Design and development of a new class of potent and highly selective inhibitors based on 3,4-dihydropyrido[3,2-d]pyrimidone scaffold
NATARAJAN, Swaminathan R, WISNOSKI, David D, HOP, Cornelis E. C. A, ZALLER, Dennis M, SCHMATZ, Dennis M, DOHERTY, James B, SINGH, Suresh B, STELMACH, John E, O'NEILL, Edward A, SCHWARTZ, Cheryl D, THOMPSON, Chris M, FITZGERALD, Catherine E, O'KEEFE, Stephen J, KUMAR, Sanjeev
Published in Bioorganic & medicinal chemistry letters (2003)
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Published in Bioorganic & medicinal chemistry letters (2003)
Journal Article
Tetrapeptide derived inhibitors of complexation of a class II MHC: fully unnatural ligands
Brian Jones, A., Acton, John J., Adams, Alan D., Yuen, Winston, Nichols, Elizabeth A., Schwartz, Cheryl D., Wicker, Linda S., Hermes, Jeffrey D.
Published in Bioorganic & medicinal chemistry letters (19.07.1999)
Published in Bioorganic & medicinal chemistry letters (19.07.1999)
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Journal Article
Tetrapeptide derived inhibitors of complexation of a class II MHC: the peptide backbone is not inviolate
Jones, A.Brian, Acton, John J., Rivetna, Meheryar N., Cummings, Richard T., Cubbon, Rose M., Nichols, Elizabeth A., Schwartz, Cheryl D., Wicker, Linda S., Hermes, Jeffrey D.
Published in Bioorganic & medicinal chemistry letters (19.07.1999)
Published in Bioorganic & medicinal chemistry letters (19.07.1999)
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DIFFICIDIN AND OXYDIFFICIDIN: NOVEL BROAD SPECTRUM ANTIBACTERIAL ANTIBIOTICS PRODUCED BY BACILLUS SUBTILIS: I. PRODUCTION, TAXONOMY AND ANTIBACTERIAL ACTIVITY
ZIMMERMAN, SHELDON B., SCHWARTZ, CHERYL D., MONAGHAN, RICHARD L., PELAK, BARBARA ANN, WEISSBERGER, BARBARA, GILFILLAN, EVEMARIE C., MOCHALES, SAGRARIO, HERNANDEZ, SEBASTIAN, CURRIE, SARA A., TEJERA, ENRIQUE, STAPLEY, EDWARD O.
Published in Journal of antibiotics (1987)
Published in Journal of antibiotics (1987)
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Journal Article
Therapeutic virginiamycin M1 analogs
LAM; YIU-KUEN T, CHANG; RAYMOND S, HENSENS; OTTO D, ZINK; DEBORAH L, SCHWARTZ; CHERYL D
Year of Publication 11.08.1992
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Year of Publication 11.08.1992
Patent
Fermentation analogs of virginiamycin M1
LAM; YIU-KUEN T, CHANG; RAYMOND S, HENSENS; OTTO D, ZINK; DEBORAH L, SCHWARTZ; CHERYL D
Year of Publication 09.04.1991
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Year of Publication 09.04.1991
Patent
Compositions having fermentation analogs of virginiamycin M1 as active ingredient
LAM; YIU-KUEN T, CHANG; RAYMOND S, HENSENS; OTTO D, ZINK; DEBORAH L, SCHWARTZ; CHERYL D
Year of Publication 16.01.1990
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Year of Publication 16.01.1990
Patent
Therapeutic virginiamycin M1 analogs
LAM; YIU-KUEN T, CHANG; RAYMOND S, HENSENS; OTTO D, ZINK; DEBORAH L, SCHWARTZ; CHERYL D
Year of Publication 22.08.1989
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Year of Publication 22.08.1989
Patent
Fermentation analogs of virginiamycin M1
LAM; YIU-KUEN T, CHANG; RAYMOND S, HENSENS; OTTO D, ZINK; DEBORAH L, SCHWARTZ; CHERYL D
Year of Publication 09.08.1988
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Year of Publication 09.08.1988
Patent