Valsartan, a potent, orally active angiotensin II antagonist developed from the structurally new amino acid series
Bühlmayer, Peter, Furet, Pascual, Criscione, Leoluca, de Gasparo, Marc, Whitebread, Steven, Schmidlin, Tibur, Lattmann, René, Wood, Jeanette
Published in Bioorganic & medicinal chemistry letters (01.01.1994)
Published in Bioorganic & medicinal chemistry letters (01.01.1994)
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Discovery and SAR of potent, orally available and brain-penetrable 5,6-dihydro-4H-3-thia-1-aza-benzo[e]azulen- and 4,5-dihydro-6-oxa-3-thia-1-aza-benzo[e]azulen derivatives as neuropeptide Y Y5 receptor antagonists
Rueeger, Heinrich, Gerspacher, Marc, Buehlmayer, Peter, Rigollier, Pascal, Yamaguchi, Yasuchika, Schmidlin, Tibur, Whitebread, Steven, Nuesslein-Hildesheim, Barbara, Nick, Hanspeter, Cricione, Leoluca
Published in Bioorganic & medicinal chemistry letters (17.05.2004)
Published in Bioorganic & medicinal chemistry letters (17.05.2004)
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Design, synthesis and SAR of a series of 2-substituted 4-amino-quinazoline neuropeptide Y Y5 receptor antagonists
RUEEGER, H, RIGOLLIER, P, ISLAM, I, ZHANG, J, GLUCHOWSKI, C, YAMAGUCHI, Y, SCHMIDLIN, T, SCHILLING, W, CRISCIONE, L, WHITEBREAD, S, CHIESI, M, WALKER, M. W, DHANOA, D
Published in Bioorganic & medicinal chemistry letters (05.06.2000)
Published in Bioorganic & medicinal chemistry letters (05.06.2000)
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Discovery and SAR of potent, orally available and brain-penetrable 5,6-dihydro-4H-3-this-1-aza-benzo[e]azulen- and 4,5-dihydro-6-oxa-3-this-1-aza-benzo[e]azulen derivatives as neuropeptide Y Y5 receptor antagonists
RUEEGER, Heinrich, GERSPACHER, Marc, BUEHLMAYER, Peter, RIGOLLIER, Pascal, YAMAGUCHI, Yasuchika, SCHMIDLIN, Tibur, WHITEBREAD, Steven, NUESSLEIN-HILDESHEIM, Barbara, NICK, Hanspeter, CRICIONE, Leoluca
Published in Bioorganic & medicinal chemistry letters (2004)
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Published in Bioorganic & medicinal chemistry letters (2004)
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Discovery and SAR of potent, orally available and brain-penetrable 5,6-dihydro-4 H-3-thia-1-aza-benzo[ e]azulen- and 4,5-dihydro-6-oxa-3-thia-1-aza-benzo[ e]azulen derivatives as neuropeptide Y Y5 receptor antagonists
Rueeger, Heinrich, Gerspacher, Marc, Buehlmayer, Peter, Rigollier, Pascal, Yamaguchi, Yasuchika, Schmidlin, Tibur, Whitebread, Steven, Nuesslein-Hildesheim, Barbara, Nick, Hanspeter, Cricione, Leoluca
Published in Bioorganic & medicinal chemistry letters (2004)
Published in Bioorganic & medicinal chemistry letters (2004)
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Journal Article
Design, synthesis and SAR of a series of 2-substituted 4-amino-quinazoline neuropeptide Y Y 5 receptor antagonists
Rueeger, Heinrich, Rigollier, Pascal, Yamaguchi, Yasuchika, Schmidlin, Tibur, Schilling, Walter, Criscione, Leoluca, Whitebread, Steven, Chiesi, Michele, Walker, Mary W, Dhanoa, Dale, Islam, Imadul, Zhang, Jack, Gluchowski, Charles
Published in Bioorganic & medicinal chemistry letters (01.06.2000)
Published in Bioorganic & medicinal chemistry letters (01.06.2000)
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Modeling the G-protein-coupled neuropeptide Y Y1 receptor agonist and antagonist binding sites
Du, P, Salon, J A, Tamm, J A, Hou, C, Cui, W, Walker, M W, Adham, N, Dhanoa, D S, Islam, I, Vaysse, P J, Dowling, B, Shifman, Y, Boyle, N, Rueger, H, Schmidlin, T, Yamaguchi, Y, Branchek, T A, Weinshank, R L, Gluchowski, C
Published in Protein engineering (01.02.1997)
Published in Protein engineering (01.02.1997)
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