Humanized UGT2 and CYP3A transchromosomic rats for improved prediction of human drug metabolism
Kazuki, Yasuhiro, Kobayashi, Kaoru, Hirabayashi, Masumi, Abe, Satoshi, Kajitani, Naoyo, Kazuki, Kanako, Takehara, Shoko, Takiguchi, Masato, Satoh, Daisuke, Kuze, Jiro, Sakuma, Tetsushi, Kaneko, Takehito, Mashimo, Tomoji, Osamura, Minori, Hashimoto, Mari, Wakatsuki, Riko, Hirashima, Rika, Fujiwara, Ryoichi, Deguchi, Tsuneo, Kurihara, Atsushi, Tsukazaki, Yasuko, Senda, Naoto, Yamamoto, Takashi, Scheer, Nico, Oshimura, Mitsuo
Published in Proceedings of the National Academy of Sciences - PNAS (19.02.2019)
Published in Proceedings of the National Academy of Sciences - PNAS (19.02.2019)
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Journal Article
Generation and utility of genetically humanized mouse models
Scheer, Nico, Snaith, Mike, Wolf, C. Roland, Seibler, Jost
Published in Drug discovery today (01.12.2013)
Published in Drug discovery today (01.12.2013)
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Journal Article
A novel panel of mouse models to evaluate the role of human pregnane X receptor and constitutive androstane receptor in drug response
Scheer, Nico, Ross, Jillian, Rode, Anja, Zevnik, Branko, Niehaves, Sandra, Faust, Nicole, Wolf, C Roland
Published in The Journal of clinical investigation (01.09.2008)
Published in The Journal of clinical investigation (01.09.2008)
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Journal Article
Quantitative prediction of human pregnane X receptor and cytochrome P450 3A4 mediated drug-drug interaction in a novel multiple humanized mouse line
Hasegawa, Maki, Kapelyukh, Yury, Tahara, Harunobu, Seibler, Jost, Rode, Anja, Krueger, Sylvia, Lee, Dongtao N, Wolf, C Roland, Scheer, Nico
Published in Molecular pharmacology (01.09.2011)
Published in Molecular pharmacology (01.09.2011)
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Journal Article
Modeling human cytochrome P450 2D6 metabolism and drug-drug interaction by a novel panel of knockout and humanized mouse lines
Scheer, Nico, Kapelyukh, Yury, McEwan, Jillian, Beuger, Vincent, Stanley, Lesley A, Rode, Anja, Wolf, C Roland
Published in Molecular pharmacology (01.01.2012)
Published in Molecular pharmacology (01.01.2012)
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Journal Article
Defining Human Pathways of Drug Metabolism In Vivo through the Development of a Multiple Humanized Mouse Model
Scheer, Nico, Kapelyukh, Yury, Rode, Anja, Oswald, Stefan, Busch, Diana, McLaughlin, Lesley A, Lin, De, Henderson, Colin J, Wolf, C Roland
Published in Drug metabolism and disposition (01.11.2015)
Published in Drug metabolism and disposition (01.11.2015)
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Journal Article
Notch signaling is required for arterial-venous differentiation during embryonic vascular development
Lawson, N D, Scheer, N, Pham, V N, Kim, C H, Chitnis, A B, Campos-Ortega, J A, Weinstein, B M
Published in Development (Cambridge) (01.10.2001)
Published in Development (Cambridge) (01.10.2001)
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Journal Article
Generation and Characterization of a Breast Cancer Resistance Protein Humanized Mouse Model
Dallas, Shannon, Salphati, Laurent, Gomez-Zepeda, David, Wanek, Thomas, Chen, Liangfu, Chu, Xiaoyan, Kunta, Jeevan, Mezler, Mario, Menet, Marie-Claude, Chasseigneaux, Stephanie, Declèves, Xavier, Langer, Oliver, Pierre, Esaie, DiLoreto, Karen, Hoft, Carolin, Laplanche, Loic, Pang, Jodie, Pereira, Tony, Andonian, Clara, Simic, Damir, Rode, Anja, Yabut, Jocelyn, Zhang, Xiaolin, Scheer, Nico
Published in Molecular pharmacology (01.05.2016)
Published in Molecular pharmacology (01.05.2016)
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Journal Article
Evaluation of organic anion transporting polypeptide 1B1 and 1B3 humanized mice as a translational model to study the pharmacokinetics of statins
Salphati, Laurent, Chu, Xiaoyan, Chen, Liangfu, Prasad, Bhagwat, Dallas, Shannon, Evers, Raymond, Mamaril-Fishman, Donna, Geier, Ethan G, Kehler, Jonathan, Kunta, Jeevan, Mezler, Mario, Laplanche, Loic, Pang, Jodie, Rode, Anja, Soars, Matthew G, Unadkat, Jashvant D, van Waterschoot, Robert A B, Yabut, Jocelyn, Schinkel, Alfred H, Scheer, Nico
Published in Drug metabolism and disposition (01.08.2014)
Published in Drug metabolism and disposition (01.08.2014)
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Journal Article
Identification of Dlk1-Dio3 imprinted gene cluster noncoding RNAs as novel candidate biomarkers for liver tumor promotion
Lempiäinen, Harri, Couttet, Philippe, Bolognani, Federico, Müller, Arne, Dubost, Valérie, Luisier, Raphaëlle, Del Rio Espinola, Alberto, Vitry, Veronique, Unterberger, Elif B, Thomson, John P, Treindl, Fridolin, Metzger, Ute, Wrzodek, Clemens, Hahne, Florian, Zollinger, Tulipan, Brasa, Sarah, Kalteis, Magdalena, Marcellin, Magali, Giudicelli, Fanny, Braeuning, Albert, Morawiec, Laurent, Zamurovic, Natasa, Längle, Ulrich, Scheer, Nico, Schübeler, Dirk, Goodman, Jay, Chibout, Salah-Dine, Marlowe, Jennifer, Theil, Diethilde, Heard, David J, Grenet, Olivier, Zell, Andreas, Templin, Markus F, Meehan, Richard R, Wolf, Roland C, Elcombe, Clifford R, Schwarz, Michael, Moulin, Pierre, Terranova, Rémi, Moggs, Jonathan G
Published in Toxicological sciences (01.02.2013)
Published in Toxicological sciences (01.02.2013)
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Journal Article
In Vivo Responses of the Human and Murine Pregnane X Receptor to Dexamethasone in Mice
SCHEER, Nico, ROSS, Jillian, KAPELYUKH, Yury, RODE, Anja, WOLF, C. Roland
Published in Drug metabolism and disposition (01.07.2010)
Published in Drug metabolism and disposition (01.07.2010)
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Journal Article
PXR and CAR: Nuclear Receptors which Play a Pivotal Role in Drug Disposition and Chemical Toxicity
Stanley, Lesley A., Horsburgh, Brian C., Ross, Jillian, Scheer, Nico, Roland Wolf, C.
Published in Drug metabolism reviews (01.01.2006)
Published in Drug metabolism reviews (01.01.2006)
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Journal Article
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