Immunomodulatory agents lenalidomide and pomalidomide co-stimulate T cells by inducing degradation of T cell repressors Ikaros and Aiolos via modulation of the E3 ubiquitin ligase complex CRL4(CRBN.)
Gandhi, Anita K, Kang, Jian, Havens, Courtney G, Conklin, Thomas, Ning, Yuhong, Wu, Lei, Ito, Takumi, Ando, Hideki, Waldman, Michelle F, Thakurta, Anjan, Klippel, Anke, Handa, Hiroshi, Daniel, Thomas O, Schafer, Peter H, Chopra, Rajesh
Published in British journal of haematology (01.03.2014)
Published in British journal of haematology (01.03.2014)
Get full text
Journal Article
Enhancement of Cytokine Production and AP-1 Transcriptional Activity in T Cells by Thalidomide-Related Immunomodulatory Drugs
Schafer, Peter H, Gandhi, Anita K, Loveland, Michelle A, Chen, Roger S, Man, Hon-Wah, Schnetkamp, Paul P M, Wolbring, Gregor, Govinda, Sowmya, Corral, Laura G, Payvandi, Faribourz, Muller, George W, Stirling, David I
Published in The Journal of pharmacology and experimental therapeutics (01.06.2003)
Published in The Journal of pharmacology and experimental therapeutics (01.06.2003)
Get full text
Journal Article
Phase 2 Trial of Iberdomide in Systemic Lupus Erythematosus
Merrill, Joan T, Werth, Victoria P, Furie, Richard, van Vollenhoven, Ronald, Dörner, Thomas, Petronijevic, Milan, Velasco, Jorge, Majdan, Maria, Irazoque-Palazuelos, Fedra, Weiswasser, Michael, Korish, Shimon, Ye, Ying, Gaudy, Allison, Schafer, Peter H, Liu, Zhaohui, Agafonova, Nataliya, Delev, Nikolay
Published in The New England journal of medicine (17.03.2022)
Published in The New England journal of medicine (17.03.2022)
Get full text
Journal Article
Lenalidomide efficacy in activated B‐cell‐like subtype diffuse large B‐cell lymphoma is dependent upon IRF4 and cereblon expression
Zhang, Ling‐Hua, Kosek, Jolanta, Wang, Maria, Heise, Carla, Schafer, Peter H., Chopra, Rajesh
Published in British journal of haematology (01.02.2013)
Published in British journal of haematology (01.02.2013)
Get full text
Journal Article
Clinical and Proteomic Correlates of Plasma ACE2 (Angiotensin-Converting Enzyme 2) in Human Heart Failure
Chirinos, Julio A, Cohen, Jordana B, Zhao, Lei, Hanff, Thomas, Sweitzer, Nancy, Fang, James, Corrales-Medina, Vicente, Anmar, Ron, Morley, Michael, Zamani, Payman, Bhattacharya, Priyanka, Brandimarto, Jeff, Jia, Yi, Basso, Michael D, Wang, Zhaoqing, Ebert, Christina, Ramirez-Valle, Francisco, Schafer, Peter H, Seiffert, Dietmar, Gordon, David A, Cappola, Thomas
Published in Hypertension (Dallas, Tex. 1979) (01.11.2020)
Published in Hypertension (Dallas, Tex. 1979) (01.11.2020)
Get full text
Journal Article
Circulating biomarker analyses in a longitudinal cohort of patients with IPF
Ebert, Christina, Walsh, Alice M, Sereda, Larisa, Wilson, Carole L, Schafer, Peter H, Fischer, Aryeh, Zhao, Lei, Ramirez-Valle, Francisco, Gordon, David, Schnapp, Lynn M
Published in American journal of physiology. Lung cellular and molecular physiology (01.03.2024)
Published in American journal of physiology. Lung cellular and molecular physiology (01.03.2024)
Get full text
Journal Article
CC-5079: A Small Molecule with MKP1, Antiangiogenic, and Antitumor Activity
Vu, Huan N., M.D, Miller, Walter J., D.O, O'Connor, Sarah A., B.S, He, Mei, M.S, Schafer, Peter H., Ph.D, Payvandi, Faribourz, Ph.D, Muller, George W., Ph.D, Stirling, David I, Libutti, Steven K., M.D
Published in The Journal of surgical research (01.11.2010)
Published in The Journal of surgical research (01.11.2010)
Get full text
Journal Article
Mechanisms Underlying the Clinical Effects of Apremilast for Psoriasis
Pincelli, Carlo, Schafer, Peter H, French, Lars E, Augustin, Matthias, Krueger, James G
Published in Journal of drugs in dermatology (01.08.2018)
Get more information
Published in Journal of drugs in dermatology (01.08.2018)
Journal Article
Biological impact of iberdomide in patients with active systemic lupus erythematosus
Lipsky, Peter E, Vollenhoven, Ronald van, Dörner, Thomas, Werth, Victoria P, Merrill, Joan T, Furie, Richard, Petronijevic, Milan, Velasco Zamora, Benito, Majdan, Maria, Irazoque-Palazuelos, Fedra, Terbrueggen, Robert, Delev, Nikolay, Weiswasser, Michael, Korish, Shimon, Stern, Mark, Hersey, Sarah, Ye, Ying, Gaudy, Allison, Liu, Zhaohui, Gagnon, Robert, Tang, Shaojun, Schafer, Peter H
Published in Annals of the rheumatic diseases (01.08.2022)
Published in Annals of the rheumatic diseases (01.08.2022)
Get full text
Journal Article
Combination therapy targeting the tumor microenvironment is effective in a model of human ocular melanoma
Mangiameli, David P, Blansfield, Joseph A, Kachala, Stephan, Lorang, Dominique, Schafer, Peter H, Muller, George W, Stirling, David I, Libutti, Steven K
Published in Journal of translational medicine (18.07.2007)
Published in Journal of translational medicine (18.07.2007)
Get full text
Journal Article
Pomalidomide in Patients with Interstitial Lung Disease due to Systemic Sclerosis: A Phase II, Multicenter, Randomized, Double-blind, Placebo-controlled, Parallel-group Study
Hsu, Vivien M, Denton, Christopher P, Domsic, Robyn T, Furst, Daniel E, Rischmueller, Maureen, Stanislav, Marina, Steen, Virginia D, Distler, Jörg H W, Korish, Shimon, Cooper, Alyse, Choi, Suktae, Schafer, Peter H, Horan, Gerald, Hough, Douglas R
Published in Journal of rheumatology (01.03.2018)
Published in Journal of rheumatology (01.03.2018)
Get more information
Journal Article
Pomalidomide and Lenalidomide Induce p21WAF-1 Expression in Both Lymphoma and Multiple Myeloma through a LSD1-Mediated Epigenetic Mechanism
ESCOUBET-LOZACH, Laure, LIN, I-Lin, JENSEN-PERGAKES, Kristen, BRADY, Helen A, GANDHI, Anita K, SCHAFER, Peter H, MULLER, George W, WORLAND, Peter J, CHAN, Kyle W. H, VERHELLE, Dominique
Published in Cancer research (Chicago, Ill.) (15.09.2009)
Published in Cancer research (Chicago, Ill.) (15.09.2009)
Get full text
Journal Article
Proteomic Associations of NT-proBNP (N-Terminal Pro-B-Type Natriuretic Peptide) in Heart Failure With Preserved Ejection Fraction
Azzo, Joe David, Dib, Marie-Joe, Zagkos, Loukas, Zhao, Lei, Wang, Zhaoqing, Chang, Ching-Pin, Ebert, Christina, Salman, Oday, Gan, Sushrima, Zamani, Payman, Cohen, Jordana B, van Empel, Vanessa, Richards, A Mark, Javaheri, Ali, Mann, Douglas L, Rietzschel, Ernst R, Schafer, Peter H, Seiffert, Dietmar A, Gill, Dipender, Burgess, Stephen, Ramirez-Valle, Francisco, Gordon, David A, Cappola, Thomas P, Chirinos, Julio A
Published in Circulation. Heart failure (01.02.2024)
Published in Circulation. Heart failure (01.02.2024)
Get full text
Journal Article
Advancing research paradigms and pathophysiological pathways in psoriatic arthritis and ankylosing spondylitis: Proceedings of the 2017 Platform for the Exchange of Expertise and Research (PEER) meeting
Abraham, Sonya, Barton, Anne, Eder, Lihi, Lim, Adrian, McGonagle, Dennis, McHugh, Neil, Pennington, Stephen, Sengupta, Raj, Siebert, Stefan, Bowness, Paul, Schafer, Peter H., Cullen, Eva, FitzGerald, Oliver
Published in Seminars in arthritis and rheumatism (01.06.2019)
Published in Seminars in arthritis and rheumatism (01.06.2019)
Get full text
Journal Article
Conference Proceeding
Efficacy, tolerability, and pharmacodynamics of apremilast in recalcitrant plaque psoriasis: a phase II open-label study
Gottlieb, Alice B, Matheson, Robert T, Menter, Alan, Leonardi, Craig L, Day, Robert M, Hu, Chiachi, Schafer, Peter H, Krueger, James G
Published in Journal of drugs in dermatology (01.08.2013)
Get more information
Published in Journal of drugs in dermatology (01.08.2013)
Journal Article
Apremilast, a novel phosphodiesterase 4 (PDE4) inhibitor, regulates inflammation through multiple cAMP downstream effectors
Perez-Aso, Miguel, Montesinos, M Carmen, Mediero, Aránzazu, Wilder, Tuere, Schafer, Peter H, Cronstein, Bruce
Published in Arthritis research & therapy (15.09.2015)
Published in Arthritis research & therapy (15.09.2015)
Get full text
Journal Article