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Ribosomes from an Oxazolidinone-Resistant Mutant Confer Resistance to Eperezolid in a Staphylococcus aureus Cell-Free Transcription-Translation Assay
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Published in Antimicrobial Agents and Chemotherapy (01.04.1998)
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The synthesis and antibacterial activity of 1,3,4-Thiadiazole phenyl oxazolidinone analogues
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Published in Bioorganic & medicinal chemistry letters (01.12.2003)
Published in Bioorganic & medicinal chemistry letters (01.12.2003)
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New Antibacterial tetrahydro-4(2 H)-thiopyran and thiomorpholine S-oxide and S, S-dioxide phenyloxazolidinones
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Published in Bioorganic & medicinal chemistry letters (01.12.2003)
Published in Bioorganic & medicinal chemistry letters (01.12.2003)
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Synthesis and biological evaluation of benzazepine oxazolidinone antibacterials
Johnson, Paul D., Aristoff, Paul A., Zurenko, Gary E., Schaadt, Ronda D., Yagi, Betty H., Ford, Charles W., Hamel, Judith C., Stapert, Douglas, Moerman, Judy K.
Published in Bioorganic & medicinal chemistry letters (01.12.2003)
Published in Bioorganic & medicinal chemistry letters (01.12.2003)
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Carbon–carbon-linked (pyrazolylphenyl)oxazolidinones with antibacterial activity against multiple drug resistant gram-positive and fastidious gram-negative bacteria
Lee, Chi Sing, Allwine, Debra A, Barbachyn, Michael R, Grega, Kevin C, Dolak, Lester A, Ford, Charles W, Jensen, Randy M, Seest, Eric P, Hamel, Judith C, Schaadt, Ronda D, Stapert, Douglas, Yagi, Betty H, Zurenko, Gary E, Genin, Michael J
Published in Bioorganic & medicinal chemistry (01.12.2001)
Published in Bioorganic & medicinal chemistry (01.12.2001)
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Nitrogen−Carbon-Linked (Azolylphenyl)oxazolidinones with Potent Antibacterial Activity Against the Fastidious Gram-Negative Organisms Haemophilus influenzae and Moraxella catarrhalis
Genin, Michael J, Hutchinson, Douglas K, Allwine, Debra A, Hester, Jackson B, Emmert, D. Edward, Garmon, Stuart A, Ford, Charles W, Zurenko, Gary E, Hamel, Judith C, Schaadt, Ronda D, Stapert, Douglas, Yagi, Betty H, Friis, Janice M, Shobe, Eric M, Adams, Wade J
Published in Journal of medicinal chemistry (17.12.1998)
Published in Journal of medicinal chemistry (17.12.1998)
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Substituent Effects on the Antibacterial Activity of Nitrogen−Carbon-Linked (Azolylphenyl)oxazolidinones with Expanded Activity Against the Fastidious Gram-Negative Organisms Haemophilus i nfluenzae and Moraxella c atarrhalis
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Published in Journal of medicinal chemistry (09.03.2000)
Published in Journal of medicinal chemistry (09.03.2000)
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Journal Article
Substituent Effects on the Antibacterial Activity of Nitrogen−Carbon-Linked (Azolylphenyl)oxazolidinones with Expanded Activity Against the Fastidious Gram-Negative Organisms Haemophilus influenzae and Moraxella catarrhalis
GENIN, Michael J., ALLWINE, Debra A., ANDERSON, David J., BARBACHYN, Michael R., EMMERT, D. Edward, GARMON, Stuart A., GRABER, David R., GREGA, Kevin C., HESTER, Jackson B., HUTCHINSON, Douglas K., MORRIS, Joel, REISCHER, Robert J., FORD, Charles W., ZURENKO, Gary E., HAMEL, Judith C., SCHAADT, Ronda D., STAPERT, Douglas, YAGI, Betty H.
Published in Journal of medicinal chemistry (09.03.2000)
Published in Journal of medicinal chemistry (09.03.2000)
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In vitro activities of U-100592 and U-100766, novel oxazolidinone antibacterial agents
ZURENKO, G. E, YAGI, B. H, SCHAADT, R. D, ALLISON, J. W, KILBURN, J. O, GLICKMAN, S. E, HUTCHINSON, D. K, BARBACHYN, M. R, BRICKNER, S. J
Published in Antimicrobial Agents and Chemotherapy (01.04.1996)
Published in Antimicrobial Agents and Chemotherapy (01.04.1996)
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Identification of Phenylisoxazolines as Novel and Viable Antibacterial Agents Active against Gram-Positive Pathogens
Barbachyn, Michael R, Cleek, Gary J, Dolak, Lester A, Garmon, Stuart A, Morris, Joel, Seest, Eric P, Thomas, Richard C, Toops, Dana S, Watt, William, Wishka, Donn G, Ford, Charles W, Zurenko, Gary E, Hamel, Judith C, Schaadt, Ronda D, Stapert, Douglas, Yagi, Betty H, Adams, Wade J, Friis, Janice M, Slatter, J. Gregory, Sams, James P, Oien, Nancee L, Zaya, Matthew J, Wienkers, Larry C, Wynalda, Michael A
Published in Journal of medicinal chemistry (16.01.2003)
Published in Journal of medicinal chemistry (16.01.2003)
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Synthesis and biological evaluation of benzazepine oxazolidinone antibacterials: Antibacterial agents: solutions for the evolving problems of resistance
JOHNSON, Paul D, ARISTOFF, Paul A, ZURENKO, Gary E, SCHAADT, Ronda D, YAGI, Betty H, FORD, Charles W, HAMEL, Judith C, STAPERT, Douglas, MOERMAN, Judy K
Published in Bioorganic & medicinal chemistry letters (2003)
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Published in Bioorganic & medicinal chemistry letters (2003)
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The synthesis and antibacterial activity of 1,3,4-thiadiazole phenyl oxazolidinone analogues: Antibacterial agents: solutions for the evolving problems of resistance
THOMASCO, Lisa M, GADWOOD, Robert C, YAGI, Betty H, WEAVER, Elizabeth A, OCHOADA, Jason M, FORD, Charles W, ZURENKO, Gary E, HAMEL, Judith C, STAPERT, Douglas, MOERMAN, Judy K, SCHAADT, Ronda D
Published in Bioorganic & medicinal chemistry letters (2003)
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Published in Bioorganic & medicinal chemistry letters (2003)
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New antibacterial tetrahydro-4(2H)-thiopyran and thiomorpholine S-oxide and S, S-dioxide phenyloxazolidinones: Antibacterial agents: solutions for the evolving problems of resistance
SINGH, Upinder, RAJU, B, FRIIS, Janice M, COURTNEY, Maria, PALANDRA, Joe, HACKBARTH, Corinne J, LOPEZ, Sara, WU, Charlotte, MORTELL, Kathleen H, TRIAS, Joaquim, ZHENGYU YUAN, PATEL, Dinesh V, LAM, Stuart, GORDEEV, Mikhail F, ZHOU, Joseph, GADWOOD, Robert C, FORD, Charles W, ZURENKO, Gary E, SCHAADT, Ronda D, MORIN, Sara E, ADAMS, Wade J
Published in Bioorganic & medicinal chemistry letters (2003)
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Published in Bioorganic & medicinal chemistry letters (2003)
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Serum inhibitory titers and serum bactericidal titers for human subjects receiving multiple doses of the antibacterial oxazolidinones eperezolid and linezolid
Schaadt, Ronda D., Batts, Donald H., Daley-Yates, Peter T., Pawsey, Steven D., Stalker, Dennis J., Zurenko, Gary E.
Published in Diagnostic microbiology and infectious disease (01.08.1997)
Published in Diagnostic microbiology and infectious disease (01.08.1997)
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U-87947E, a protein quinolone antibacterial agent incorporating a bicyclo[1.1.1]pent-1-yl ( BCP) subunit
Barbachyn, Michael R., Hutchinson, Douglas K., Toops, Dana S., Reid, Raymond J., Zurenko, Gary E., Yagi, Betty H., Schaadt, Ronda D., Allison, John W.
Published in Bioorganic & medicinal chemistry letters (1993)
Published in Bioorganic & medicinal chemistry letters (1993)
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Synthesis and antibacterial activity of new tropone-substituted phenyloxazolidinone antibacterial agents 2. Modification of the phenyl ring — the potentiating effect of fluorine substitution on in vivo activity
Barbachyn, Michael R., Toops, Dana S., Grega, Kevin C., Hendges, Susan K., Ford, Charles W., Zurenko, Gary E., Hamel, Judith C., Schaadt, Jonda D., Stapert, Douglas, Yagi, Betty H., Buysse, Jerry M., Demyan, William F., Kilburn, James O., Glickman, Suzanne E.
Published in Bioorganic & medicinal chemistry letters (07.05.1996)
Published in Bioorganic & medicinal chemistry letters (07.05.1996)
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Journal Article
Synthesis and antibacterial activity of new tropone-substituted phenyloxazolidinone antibacterial agents 1. Identification of leads and importance of the tropone substitution pattern
Barbachyn, Michael R., Toops, Dana S., Ulanowicz, Debra A., Grega, Kevin C., Brickner, Steven J., Ford, Charles W., Zurenko, Gary E., Hamel, Judith C., Schaadt, Ronda D., Stapert, Douglas, Yagi, Betty H., Buysse, Jerry M., Demyan, William F., Kilburn, James O., Glickman, Suzanne E.
Published in Bioorganic & medicinal chemistry letters (07.05.1996)
Published in Bioorganic & medicinal chemistry letters (07.05.1996)
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Journal Article
The bactericidal activity and postantibiotic effect of trospectomycin
Yagi, Betty H., Schaadt, Ronda D., Zurenko, Gary E.
Published in Diagnostic microbiology and infectious disease (01.07.1992)
Published in Diagnostic microbiology and infectious disease (01.07.1992)
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