Discovery of 3-[(4,5,7-Trifluorobenzothiazol-2-yl)methyl]indole-N-acetic Acid (Lidorestat) and Congeners as Highly Potent and Selective Inhibitors of Aldose Reductase for Treatment of Chronic Diabetic Complications
Van Zandt, Michael C, Jones, Michael L, Gunn, David E, Geraci, Leo S, Jones, J. Howard, Sawicki, Diane R, Sredy, Janet, Jacot, Jorge L, DiCioccio, A. Thomas, Petrova, Tatiana, Mitschler, Andre, Podjarny, Alberto D
Published in Journal of medicinal chemistry (05.05.2005)
Published in Journal of medicinal chemistry (05.05.2005)
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Discovery of [3-(4,5,7-trifluoro-benzothiazol-2-ylmethyl)-pyrrolo[2,3-b] pyridin-1-yl]acetic acids as highly potent and selective inhibitors of aldose reductase for treatment of chronic diabetic complications
VAN ZANDT, Michael C, DOAN, Brian, SAWICKI, Diane R, SREDY, Janet, PODJARNY, Alberto D
Published in Bioorganic & medicinal chemistry letters (01.04.2009)
Published in Bioorganic & medicinal chemistry letters (01.04.2009)
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Novel Benzofuran and Benzothiophene Biphenyls as Inhibitors of Protein Tyrosine Phosphatase 1B with Antihyperglycemic Properties
Malamas, Michael S, Sredy, Janet, Moxham, Christopher, Katz, Alan, Xu, Weixin, McDevitt, Robert, Adebayo, Folake O, Sawicki, Diane R, Seestaller, Laura, Sullivan, Donald, Taylor, Joseph R
Published in Journal of medicinal chemistry (06.04.2000)
Published in Journal of medicinal chemistry (06.04.2000)
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PTP1B Inhibition and Antihyperglycemic Activity in the ob/ob Mouse Model of Novel 11-Arylbenzo[b]naphtho[2,3-d]furans and 11-Arylbenzo[b]naphtho[2,3-d]thiophenes
Wrobel, Jay, Sredy, Janet, Moxham, Christopher, Dietrich, Arlene, Li, Zenan, Sawicki, Diane R, Seestaller, Laura, Wu, Li, Katz, Alan, Sullivan, Donald, Tio, Cesario, Zhang, Zhong-Yin
Published in Journal of medicinal chemistry (26.08.1999)
Published in Journal of medicinal chemistry (26.08.1999)
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Design and synthesis of highly potent and selective (2-arylcarbamoyl-phenoxy)-acetic acid inhibitors of aldose reductase for treatment of chronic diabetic complications
Van Zandt, Michael C., Sibley, Evelyn O., McCann, Erin E., Combs, Kerry J., Flam, Brenda, Sawicki, Diane R., Sabetta, Al, Carrington, Anne, Sredy, Janet, Howard, Eduardo, Mitschler, Andre, Podjarny, Alberto D.
Published in Bioorganic & medicinal chemistry (01.11.2004)
Published in Bioorganic & medicinal chemistry (01.11.2004)
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New Azolidinediones as Inhibitors of Protein Tyrosine Phosphatase 1B with Antihyperglycemic Properties
Malamas, Michael S, Sredy, Janet, Gunawan, Iwan, Mihan, Brenda, Sawicki, Diane R, Seestaller, Laura, Sullivan, Donald, Flam, Brenda R
Published in Journal of medicinal chemistry (09.03.2000)
Published in Journal of medicinal chemistry (09.03.2000)
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Synthesis and PTP1B Inhibition of Novel 4-Aryl-1-Oxa-9-Thiacyclopenta[ b]fluorenes
Wrobel, Jay, Li, Zenan, Sredy, Janet, Sawicki, Diane R, Seestaller, Laura, Sullivan, Donald
Published in Bioorganic & medicinal chemistry letters (17.07.2000)
Published in Bioorganic & medicinal chemistry letters (17.07.2000)
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Discovery of [3-(4,5,7-trifluoro-benzothiazol-2-ylmethyl)-pyrrolo[2,3-b]pyridin -1-yl]ace tic acids as highly potent and selective inhibitors of aldose reductase for treatment of chronic diabetic complications
Van Zandt, Michael C, Doan, Brian, Sawicki, Diane R, Sredy, Janet, Podjarny, Alberto D
Published in Bioorganic & medicinal chemistry letters (01.04.2009)
Published in Bioorganic & medicinal chemistry letters (01.04.2009)
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Triglyceride modulation by acifran analogs: activity towards the niacin high and low affinity G protein-coupled receptors HM74A and HM74
Mahboubi, Keyvan, Witman-Jones, Terri, Adamus, Jean E., Letsinger, Jack T., Whitehouse, Darren, Moorman, Allan R., Sawicki, Diane, Bergenhem, Nils, Ross, Stuart A.
Published in Biochemical and biophysical research communications (10.02.2006)
Published in Biochemical and biophysical research communications (10.02.2006)
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Structural abnormalities do not explain the early functional abnormalities in the peripheral nerves of the streptozotocin diabetic rat
WALKER, DAVID, CARRINGTON, ANNE, CANNAN, SUSAN A., SAWICKI, DIANE, SREDY, JANET, BOULTON, ANDREW J. M., MALIK, RAYAZ A.
Published in Journal of anatomy (01.10.1999)
Published in Journal of anatomy (01.10.1999)
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Insulin resistance is associated with abnormal dephosphorylation of a synthetic phosphopeptide corresponding to the major autophosphorylation sites of the insulin receptor
Sredy, Janet, Sawicki, Diane R., Flam, Brenda R., Sullivan, Donald
Published in Metabolism, clinical and experimental (01.08.1995)
Published in Metabolism, clinical and experimental (01.08.1995)
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Adenosine triphosphatase activity in sciatic nerve tissue of streptozocin-induced diabetic rats with and without high dietary sucrose: effect of aldose reductase inhibitors
Sredy, J, Flam, B R, Sawicki, D R
Published in Proceedings of the Society for Experimental Biology and Medicine (01.06.1991)
Published in Proceedings of the Society for Experimental Biology and Medicine (01.06.1991)
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