PROCESS FOR THE PREPARATION OF N-((1R,2S,SR)-5-(TERT-BUTYLAMINO)-2-((S)-3-(7-TERT-BUTYLPYRAZOLO[1,5-A][1,3,5]TRIAZIN-4-YLAMINO)-2-OXOPYRROLIDIN-1-YL)CYCLOHEXYL)ACETAMIDE
Fan, Yu, Gonzalez-Bobes, Francisco, Hickey, Matthew R, Razler, Thomas M, Aytar, Burcu Selin, Green, Rebecca A, Savage, Scott A, Sfouggatakis, Chris, Leahy, David K, Deerberg, Joerg, La Cruz, Thomas E, Borovika, Alina, Zaretsky, Serge, Zheng, Bin, Fenster, Michael David Bengt, Lauser, Kathleen, Eastgate, Martin G, Zhu, Ye, Luo, Helen Y, Domagalski, Nathan R, Chan, Collin, Lee, Hong Geun, Soumeillant, Maxime C. D, Kopp, Nathaniel David, Forest, Robert V
Year of Publication 27.05.2022
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Year of Publication 27.05.2022
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PROCESS FOR THE PREPARATION OF N-((1R,2S,SR)-5-(TERT-BUTYLAMINO)-2-((S)-3-(7-TERT-BUTYLPYRAZOLO[1,5-A][1,3,5]TRIAZIN-4-YLAMINO)-2-OXOPYRROLIDIN-1-YL)CYCLOHEXYL)ACETAMIDE
Fan, Yu, Gonzalez-Bobes, Francisco, Hickey, Matthew R, Razler, Thomas M, Aytar, Burcu Selin, Green, Rebecca A, Savage, Scott A, Sfouggatakis, Chris, Leahy, David K, Deerberg, Joerg, La Cruz, Thomas E, Borovika, Alina, Zaretsky, Serge, Zheng, Bin, Fenster, Michael David Bengt, Lauser, Kathleen, Eastgate, Martin G, Zhu, Ye, Luo, Helen Y, Domagalski, Nathan R, Chan, Collin, Lee, Hong Geun, Soumeillant, Maxime C. D, Kopp, Nathaniel David, Forest, Robert V
Year of Publication 13.05.2022
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Year of Publication 13.05.2022
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Hepatitis C virus inhibitors
Ferreira, Glenn, Mack, Brendan, Domagalski, Nathan R, Hallow, Daniel M, Savage, Scott A, Vemishetti, Purushotham, Qiu, Yuping, Hobson, Lindsay, Rogers, Amanda, Fenster, Michael, Lou, Sha
Year of Publication 03.12.2019
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Year of Publication 03.12.2019
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PROCESS FOR THE PREPARATION OF N-((1R,2S,SR)-5-(TERT-BUTYLAMINO)-2-((S)-3-(7-TERT-BUTYLPYRAZOLO(1,5-A)(1,3,5)TRIAZIN-4-YLAMINO)-2-OXOPYRROLIDIN-1-YL)CYCLOHEXYL)ACETAMIDE
DOMAGALSKI Nathan R, FOREST Robert V, BOROVIKA Alina, FAN Yu, AYTAR Burcu Selin, LAUSER Kathleen, GREEN Rebecca A, FENSTER Michael David Bengt, LEAHY David K, SAVAGE Scott A, ZHU Ye, LA CRUZ Thomas E, LEE Hong Geun, RAZLER Thomas M, HICKEY Matthew R, ZHENG Bin, ZARETSKY Serge, DEERBERG Joerg, CHAN Collin, EASTGATE Martin D, LUO Helen Y, SOUMEILLANT Maxime C.D, GONZALEZ-BOBES Francisco, SFOUGGATAKIS Chris, KOPP Nathaniel David
Year of Publication 29.04.2022
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Year of Publication 29.04.2022
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PROCESS FOR THE PREPARATION OF N-((1R,2S,SR)-5-(TERT-BUTYLAMINO)-2-((S)-3-(7-TERT-BUTYLPYRAZOLO[1,5-A][1,3,5]TRIAZIN-4-YLAMINO)-2-OXOPYRROLIDIN-1-YL)CYCLOHEXYL)ACETAMIDE
BOROVIKA, ALINA, EASTGATE, MARTIN, D, GONZALEZ-BOBES, FRANCISCO, SAVAGE, SCOTT A, DOMAGALSKI, NATHAN, R, ZHU, YE, FOREST, ROBERT, V, SFOUGGATAKIS, CHRIS, CHAN, COLLIN, AYTAR, BURCU, SELIN, LAUSER, KATHLEEN, ZARETSKY, SERGE, ZHENG, BIN, GREEN, REBECCA, A, RAZLER, THOMAS, M, FENSTER, MICHAEL, DAVID, BENGT, FAN, YU, LA CRUZ, THOMAS, E, SOUMEILLANT, MAXIME, C., D, LUO, HELEN, Y, LEAHY, DAVID, K, KOPP, NATHANIEL, DAVID, LEE, HONG, GEUN, HICKEY, MATTHEW, R, DEERBERG, JOERG
Year of Publication 31.03.2022
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Year of Publication 31.03.2022
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PROCESS FOR THE PREPARATION OF N-((1R,2S,SR)-5-(TERT-BUTYLAMINO)-2-((S)-3-(7-TERT-BUTYLPYRAZOLO[1,5-A][1,3,5]TRIAZIN-4-YLAMINO)-2-OXOPYRROLIDIN-1-YL)CYCLOHEXYL)ACETAMIDE
SFOUGGATAKIS, Chris, ZARETSKY, Serge, DOMAGALSKI, Nathan R, EASTGATE, Martin D, RAZLER, Thomas M, LA CRUZ, Thomas E, LAUSER, Kathleen, FENSTER, Michael David Bengt, SOUMEILLANT, Maxime C.D, AYTAR, Burcu Selin, LUO, Helen Y, FAN, Yu, LEE, Hong Geun, LEAHY, David K, KOPP, Nathaniel David, CHAN, Collin, ZHENG, Bin, SAVAGE, Scott A, FOREST, Robert V, GREEN, Rebecca A, HICKEY, Matthew R, DEERBERG, Joerg, GONZALEZ-BOBES, Francisco, BOROVIKA, Alina, ZHU, Ye
Year of Publication 10.03.2022
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Year of Publication 10.03.2022
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FREMGANGSMÅDE TIL FREMSTILLING AF N-((1R,2S,SR)-5-(TERT-BUTYLAMINO)-2-((S)-3-(7- TERT-BUTYLPYRAZOLO[1,5-A][1,3,5]TRIAZIN-4-YLAMINO)-2-OXOPYRROLIDIN-1- YL)CYCLOHEXYL)ACETAMID
SFOUGGATAKIS, Chris, ZARETSKY, Serge, DOMAGALSKI, Nathan R, EASTGATE, Martin D, RAZLER, Thomas M, LA CRUZ, Thomas E, LAUSER, Kathleen, FENSTER, Michael David Bengt, SOUMEILLANT, Maxime C.D, AYTAR, Burcu Selin, LUO, Helen Y, FAN, Yu, LEE, Hong Geun, LEAHY, David K, KOPP, Nathaniel David, CHAN, Collin, ZHENG, Bin, SAVAGE, Scott A, FOREST, Robert V, GREEN, Rebecca A, HICKEY, Matthew R, DEERBERG, Joerg, GONZALEZ-BOBES, Francisco, BOROVIKA, Alina, ZHU, Ye
Year of Publication 07.03.2022
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Year of Publication 07.03.2022
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PROCESS FOR THE PREPARATION OF N-((1R,2S,SR)-5-(TERT-BUTYLAMINO)-2-((S)-3-(7-TERT-BUTYLPYRAZOLO[1,5-A][1,3,5]TRIAZIN-4-YLAMINO)-2-OXOPYRROLIDIN-1-YL)CYCLOHEXYL)ACETAMIDE
BOROVIKA, ALINA, AYTAR, BURCU SELIN, GONZALEZ-BOBES, FRANCISCO, SAVAGE, SCOTT A, GREEN, REBECCA A, ZHU, YE, HICKEY, MATTHEW R, KOPP, NATHANIEL DAVID, SFOUGGATAKIS, CHRIS, CHAN, COLLIN, LAUSER, KATHLEEN, FOREST, ROBERT V, LEE, HONG GEUN, ZARETSKY, SERGE, ZHENG, BIN, LUO, HELEN Y, LA CRUZ, THOMAS E, SOUMEILLANT, MAXIME C.D, FAN, YU, EASTGATE, MARTIN D, RAZLER, THOMAS M, LEAHY, DAVID K, DOMAGALSKI, NATHAN R, FENSTER, MICHAEL DAVID BENGT, DEERBERG, JOERG
Year of Publication 07.03.2022
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Year of Publication 07.03.2022
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Process for the preparation of N-((1R,2S,5R)-5-(tert-butylamino)-2-((S)-3-(7-tert-butylpyrazolo[1,5-a][1,3,5]triazin-4-ylamino)-2-oxopyrroldin-1-yl)cyclohexyl)acetamide
Fan, Yu, Eastgate, Martin D, Gonzalez-Bobes, Francisco, Hickey, Matthew R, Razler, Thomas M, Aytar, Burcu Selin, Green, Rebecca A, Savage, Scott A, Sfouggatakis, Chris, Leahy, David K, Deerberg, Joerg, La Cruz, Thomas E, Borovika, Alina, Zaretsky, Serge, Zheng, Bin, Fenster, Michael David Bengt, Lauser, Kathleen, Zhu, Ye, Luo, Helen Y, Domagalski, Nathan R, Chan, Collin, Lee, Hong Geun, Soumeillant, Maxime C. D, Kopp, Nathaniel David, Forest, Robert V
Year of Publication 22.02.2022
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Year of Publication 22.02.2022
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PROCESS FOR THE PREPARATION OF N-((1R,2S,SR)-5-(TERT-BUTYLAMINO)-2-((S)-3-(7-TERT-BUTYLPYRAZOLO[1,5-A][1,3,5]TRIAZIN-4-YLAMINO)-2-OXOPYRROLIDIN-1-YL)CYCLOHEXYL)ACETAMIDE
SFOUGGATAKIS, Chris, ZARETSKY, Serge, DOMAGALSKI, Nathan R, EASTGATE, Martin D, RAZLER, Thomas M, LA CRUZ, Thomas E, LAUSER, Kathleen, FENSTER, Michael David Bengt, SOUMEILLANT, Maxime C.D, AYTAR, Burcu Selin, LUO, Helen Y, FAN, Yu, LEE, Hong Geun, LEAHY, David K, KOPP, Nathaniel David, CHAN, Collin, ZHENG, Bin, SAVAGE, Scott A, FOREST, Robert V, GREEN, Rebecca A, HICKEY, Matthew R, DEERBERG, Joerg, GONZALEZ-BOBES, Francisco, BOROVIKA, Alina, ZHU, Ye
Year of Publication 01.12.2021
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Year of Publication 01.12.2021
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HEPATITIS C VIRUS INHIBITORS
SAVAGE, Scott A, FENSTER, Michael, ROGERS, Amanda, LOU, Sha, HOBSON, Lindsay, QIU, Yuping, HALLOW, Daniel M, VEMISHETTI, Purushotham, FERREIRA, Glenn, DOMAGALSKI, Nathan R, MACK, Brendan
Year of Publication 07.06.2018
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Year of Publication 07.06.2018
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Methods of producing an HIV maturation inhibitor
Ortiz, Adrian, Nye, Jeffrey A, Kiau, Susanne, Savage, Scott A, Ho, Jeanne, Soumeillant, Maxime, Eastgate, Martin D, Benkovics, Tamas, Strotman, Neil A, Haley, Matthew W, Xu, Zhongmin, Tan, Yichen
Year of Publication 05.03.2019
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Year of Publication 05.03.2019
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PROCESS FOR THE PREPARATION OF N-((1R,2S,5R)-5-(TERT-BUTYLAMINO)-2-((S)-3-(7-TERT-BUTYLPYRAZOLO[1,5-A][1,3,5]TRIAZIN-4-YLAMINO)-2-OXOPYRROLIDIN-1-YL)CYCLOHEXYL)ACETAMIDE
Fan, Yu, Eastgate, Martin D, Gonzalez-Bobes, Francisco, Hickey, Matthew R, Razler, Thomas M, Soumeillant, Maxime C.D, Aytar, Burcu Selin, Green, Rebecca A, Savage, Scott A, Sfouggatakis, Chris, Leahy, David K, Deerberg, Joerg, La Cruz, Thomas E, Borovika, Alina, Zaretsky, Serge, Zheng, Bin, Fenster, Michael David Bengt, Lauser, Kathleen, Zhu, Ye, Luo, Helen Y, Domagalski, Nathan R, Chan, Collin, Lee, Hong Geun, Kopp, Nathaniel David, Forest, Robert V
Year of Publication 16.07.2020
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Year of Publication 16.07.2020
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PROCESS FOR THE PREPARATION OF N-((1R,2S,5R)-5-(TERT
SFOUGGATAKIS, Chris, ZARETSKY, Serge, DOMAGALSKI, Nathan R, EASTGATE, Martin D, RAZLER, Thomas M, LA CRUZ, Thomas E, LAUSER, Kathleen, FENSTER, Michael David Bengt, SOUMEILLANT, Maxime C.D, AYTAR, Burcu Selin, LUO, Helen Y, FAN, Yu, LEE, Hong Geun, LEAHY, David K, KOPP, Nathaniel David, CHAN, Collin, ZHENG, Bin, SAVAGE, Scott A, FOREST, Robert V, GREEN, Rebecca A, HICKEY, Matthew R, DEERBERG, Joerg, GONZALEZ-BOBES, Francisco, BOROVIKA, Alina, ZHU, Ye
Year of Publication 27.05.2020
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Year of Publication 27.05.2020
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Process for the preparation of N-((1R,2S,5R)-5-(tert,-butylamino)-2- ((S)-3-(7-tert-butylpyrazolo[l,5-a][1,3,5]triazin-4-ylamino)-2- oxopyrrolidin- 1 -yl)c yclohexyl) acetamide
SFOUGGATAKIS, Chris, ZARETSKY, Serge, DOMAGALSKI, Nathan R, EASTGATE, Martin D, RAZLER, Thomas M, LA CRUZ, Thomas E, LAUSER, Kathleen, FENSTER, Michael David Bengt, SOUMEILLANT, Maxime C.D, AYTAR, Burcu Selin, LUO, Helen Y, FAN, Yu, LEE, Hong Geun, LEAHY, David K, KOPP, Nathaniel David, CHAN, Collin, ZHENG, Bin, SAVAGE, Scott A, FOREST, Robert V, GREEN, Rebecca A, HICKEY, Matthew R, DEERBERG, Joerg, GONZALEZ-BOBES, Francisco, BOROVIKA, Alina, ZHU, Ye
Year of Publication 02.04.2020
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Year of Publication 02.04.2020
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Process for the preparation of n-((1r,2s,5r)-5-(tert-butylamino)-2-((s)-3-(7-tert-butylpyrazolo[1,5-a][1,3,5]triazin-4-ylamino)-2-oxopyrrolidin-1-yl)cyclohexyl)acetamide
DOMAGALSKI Nathan R, FOREST Robert V, FAN Yu, BOROVIKA Alina, AYTAR Burcu Selin, LAUSER Kathleen, GREEN Rebecca A, FENSTER Michael David Bengt, LEAHY David K, SAVAGE Scott A, ZHU Ye, LA CRUZ Thomas E, LEE Hong Geun, RAZLER Thomas M, HICKEY Matthew R, ZHENG Bin, ZARETSKY Serge, DEERBERG Joerg, CHAN Collin, EASTGATE Martin D, LUO Helen Y, SOUMEILLANT Maxime C.D, GONZALEZ-BOBES Francisco, SFOUGGATAKIS Chris, KOPP Nathaniel David
Year of Publication 31.03.2020
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Year of Publication 31.03.2020
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Process for the preparation of N-((lR,2S,5R)-5-(7¾'i?7,-butylamino)-2- ((s)-3-(7-7e ?7,-butylpyrazolo[l,5-a][l,3,5]triazin-4-ylamino)-2- oxopyrrolidin- 1 -yl)c yclohexyl) acetamide
SFOUGGATAKIS, Chris, ZARETSKY, Serge, DOMAGALSKI, Nathan R, EASTGATE, Martin D, RAZLER, Thomas M, LA CRUZ, Thomas E, LAUSER, Kathleen, FENSTER, Michael David Bengt, SOUMEILLANT, Maxime C.D, AYTAR, Burcu Selin, LUO, Helen Y, FAN, Yu, LEE, Hong Geun, LEAHY, David K, KOPP, Nathaniel David, CHAN, Collin, ZHENG, Bin, SAVAGE, Scott A, FOREST, Robert V, GREEN, Rebecca A, HICKEY, Matthew R, DEERBERG, Joerg, GONZALEZ-BOBES, Francisco, BOROVIKA, Alina, ZHU, Ye
Year of Publication 05.03.2020
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Year of Publication 05.03.2020
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PROCESS FOR THE PREPARATION OF N-((1R,2S,5R)-5-(TERT-BUTYLAMINO)-2-((S)-3-(7-TERT-BUTYLPYRAZOLO[1,5-A][1,3,5]TRIAZIN-4-YLAMINO)-2-OXOPYRROLIDIN-1-YL)CYCLOHEXYL)ACETAMIDE
SFOUGGATAKIS, Chris, ZARETSKY, Serge, DOMAGALSKI, Nathan R, EASTGATE, Martin D, RAZLER, Thomas M, LA CRUZ, Thomas E, LAUSER, Kathleen, FENSTER, Michael David Bengt, SOUMEILLANT, Maxime C.D, AYTAR, Burcu Selin, LUO, Helen Y, FAN, Yu, LEE, Hong Geun, LEAHY, David K, KOPP, Nathaniel David, CHAN, Collin, ZHENG, Bin, SAVAGE, Scott A, FOREST, Robert V, GREEN, Rebecca A, HICKEY, Matthew R, DEERBERG, Joerg, GONZALEZ-BOBES, Francisco, BOROVIKA, Alina, ZHU, Ye
Year of Publication 27.02.2020
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Year of Publication 27.02.2020
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Methods of producing an HIV maturation inhibitor
Ortiz, Adrian, Nye, Jeffrey A, Kiau, Susanne, Savage, Scott A, Ho, Jeanne, Soumeillant, Maxime, Eastgate, Martin D, Benkovics, Tamas, Strotman, Neil A, Haley, Matthew W, Xu, Zhongmin, Tan, Yichen
Year of Publication 26.07.2018
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Year of Publication 26.07.2018
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HEPATITIS C VIRUS INHIBITORS
SAVAGE, Scott A, FENSTER, Michael, ROGERS, Amanda, LOU, Sha, HOBSON, Lindsay, QIU, Yuping, HALLOW, Daniel M, VEMISHETTI, Purushotham, FERREIRA, Glenn, DOMAGALSKI, Nathan R, MACK, Brendan
Year of Publication 03.05.2017
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Year of Publication 03.05.2017
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