Quantification of mouse pulmonary cancer models by microcomputed tomography imaging
Fushiki, Hiroshi, Kanoh‐Azuma, Tomoko, Katoh, Masahiro, Kawabata, Ken, Jiang, Jian, Tsuchiya, Nozomi, Satow, Akio, Tamai, Yoshitaka, Hayakawa, Yoshihiro
Published in Cancer science (01.08.2009)
Published in Cancer science (01.08.2009)
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Discovery and in vitro and in vivo profiles of 4-fluoro- N-[4-[6-(isopropylamino)pyrimidin-4-yl]-1,3-thiazol-2-yl]- N-methylbenzamide as novel class of an orally active metabotropic glutamate receptor 1 (mGluR1) antagonist
Satoh, Atsushi, Nagatomi, Yasushi, Hirata, Yukari, Ito, Satoru, Suzuki, Gentaroh, Kimura, Toshifumi, Maehara, Shunsuke, Hikichi, Hirohiko, Satow, Akio, Hata, Mikiko, Ohta, Hisashi, Kawamoto, Hiroshi
Published in Bioorganic & medicinal chemistry letters (15.09.2009)
Published in Bioorganic & medicinal chemistry letters (15.09.2009)
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Pharmacological Effects of the Metabotropic Glutamate Receptor 1 Antagonist Compared with Those of the Metabotropic Glutamate Receptor 5 Antagonist and Metabotropic Glutamate Receptor 2/3 Agonist in Rodents: Detailed Investigations with a Selective Allosteric Metabotropic Glutamate Receptor 1 Antagonist, FTIDC [4-[1-(2-Fluoropyridine-3-yl)-5-methyl-1H-1,2,3-triazol-4-yl]-N-isopropyl-N-methyl-3,6-dihydropyridine-1(2H)-carboxamide]
Satow, Akio, Maehara, Shunsuke, Ise, Satoko, Hikichi, Hirohiko, Fukushima, Miyuki, Suzuki, Gentaroh, Kimura, Toshifumi, Tanak, Takeshi, Ito, Satoru, Kawamoto, Hiroshi, Ohta, Hisashi
Published in The Journal of pharmacology and experimental therapeutics (01.08.2008)
Published in The Journal of pharmacology and experimental therapeutics (01.08.2008)
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Discovery and biological profile of isoindolinone derivatives as novel metabotropic glutamate receptor 1 antagonists: A potential treatment for psychotic disorders
Ito, Satoru, Hirata, Yukari, Nagatomi, Yasushi, Satoh, Atsushi, Suzuki, Gentaroh, Kimura, Toshifumi, Satow, Akio, Maehara, Shunsuke, Hikichi, Hirohiko, Hata, Mikiko, Ohta, Hisashi, Kawamoto, Hiroshi
Published in Bioorganic & medicinal chemistry letters (15.09.2009)
Published in Bioorganic & medicinal chemistry letters (15.09.2009)
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Unique Antipsychotic Activities of the Selective Metabotropic Glutamate Receptor 1 Allosteric Antagonist 2-Cyclopropyl-5-[1-(2-fluoro-3-pyridinyl)-5-methyl-1H-1,2,3-triazol-4-yl]-2,3-dihydro-1H-isoindol-1-one
Satow, Akio, Suzuki, Gentaroh, Maehara, Shunsuke, Hikichi, Hirohiko, Murai, Takeshi, Murai, Takashi, Kawagoe-Takaki, Hiroko, Hata, Mikiko, Ito, Satoru, Ozaki, Satoshi, Kawamoto, Hiroshi, Ohta, Hisashi
Published in The Journal of pharmacology and experimental therapeutics (01.07.2009)
Published in The Journal of pharmacology and experimental therapeutics (01.07.2009)
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Antipsychotic effects of N-desmethylclozapine on sensorimotor gating function in rats — Possible involvement of activation of M₁ muscarinic receptors
Maehara, Shunsuke, Satow, Akio, Hikichi, Hirohiko, Ohta, Hisashi
Published in European journal of pharmacology (01.09.2011)
Published in European journal of pharmacology (01.09.2011)
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Pharmacological Characterization of a New, Orally Active and Potent Allosteric Metabotropic Glutamate Receptor 1 Antagonist, 4-[1-(2-Fluoropyridin-3-yl)-5-methyl-1H-1,2,3-triazol-4-yl]-N-isopropyl-N-methyl-3,6-dihydropyridine-1(2H)-carboxamide (FTIDC)
Suzuki, Gentaroh, Kimura, Toshifumi, Satow, Akio, Kaneko, Naoki, Fukuda, Junko, Hikichi, Hirohiko, Sakai, Naoko, Maehara, Shunsuke, Kawagoe-Takaki, Hiroko, Hata, Mikiko, Azuma, Tomoko, Ito, Satoru, Kawamoto, Hiroshi, Ohta, Hisashi
Published in The Journal of pharmacology and experimental therapeutics (01.06.2007)
Published in The Journal of pharmacology and experimental therapeutics (01.06.2007)
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Correlation of Receptor Occupancy of Metabotropic Glutamate Receptor Subtype 1 (mGluR1) in Mouse Brain With In vivo Activity of Allosteric mGluR1 Antagonists
Suzuki, Gentaroh, Kawagoe-Takaki, Hiroko, Inoue, Takao, Kimura, Toshifumi, Hikichi, Hirohiko, Murai, Takashi, Satow, Akio, Hata, Mikiko, Maehara, Shunsuke, Ito, Satoru, Kawamoto, Hiroshi, Ozaki, Satoshi, Ohta, Hisashi
Published in Journal of Pharmacological Sciences (2009)
Published in Journal of Pharmacological Sciences (2009)
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Face-washing behavior induced by the group I metabotropic glutamate receptor agonist (S)-3,5-DHPG in mice is mediated by mGlu1 receptor
HIKICHI, Hirohiko, IWAHORI, Yuki, MURAI, Takeshi, MAEHARA, Shunsuke, SATOW, Akio, OHTA, Hisashi
Published in European journal of pharmacology (31.05.2008)
Published in European journal of pharmacology (31.05.2008)
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Antipsychotic effects of N-desmethylclozapine on sensorimotor gating function in rats — Possible involvement of activation of M 1 muscarinic receptors
Maehara, Shunsuke, Satow, Akio, Hikichi, Hirohiko, Ohta, Hisashi
Published in European journal of pharmacology (30.09.2011)
Published in European journal of pharmacology (30.09.2011)
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Pharmacological effects of metabotropic glutamate receptor ligands on prepulse inhibition in DBA/2J mice
Hikichi, Hirohiko, Nishino, Miho, Fukushima, Miyuki, Satow, Akio, Maehara, Shunsuke, Kawamoto, Hiroshi, Ohta, Hisashi
Published in European journal of pharmacology (10.08.2010)
Published in European journal of pharmacology (10.08.2010)
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Discovery and biological profile of 4-(1-aryltriazol-4-yl)-tetrahydropyridines as an orally active new class of metabotropic glutamate receptor 1 antagonist
Ito, Satoru, Satoh, Atsushi, Nagatomi, Yasushi, Hirata, Yukari, Suzuki, Gentaroh, Kimura, Toshifumi, Satow, Akio, Maehara, Shunsuke, Hikichi, Hirohiko, Hata, Mikiko, Kawamoto, Hiroshi, Ohta, Hisashi
Published in Bioorganic & medicinal chemistry (15.11.2008)
Published in Bioorganic & medicinal chemistry (15.11.2008)
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Antipsychotic effects of N-desmethylclozapine on sensorimotor gating function in rats - Possible involvement of activation of M sub(1 muscarinic receptors)
Maehara, Shunsuke, Satow, Akio, Hikichi, Hirohiko, Ohta, Hisashi
Published in European journal of pharmacology (30.09.2011)
Published in European journal of pharmacology (30.09.2011)
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Pharmacological effects of metabotropic glutamate receptor ligands on prepulse inhibition in DBA/2J mice: Metabotropic Glutamate Receptors and Cognition
HIKICHI, Hirohiko, NISHINO, Miho, FUKUSHIMA, Miyuki, SATOW, Akio, MAEHARA, Shunsuke, KAWAMOTO, Hiroshi, OHTA, Hisashi
Published in European journal of pharmacology (2010)
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Published in European journal of pharmacology (2010)
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Effects of a novel metabotropic glutamate receptor 7 negative allosteric modulator, 6-(4-methoxyphenyl)-5-methyl-3-pyridin-4-ylisoxazonolo[4,5-c]pyridin-4(5H)-one (MMPIP), on the central nervous system in rodents: Metabotropic Glutamate Receptors and Cognition
HIKICHI, Hirohiko, MURAI, Takeshi, OHTA, Hisashi, OKUDA, Shoki, MAEHARA, Shunsuke, SATOW, Akio, ISE, Satoko, NISHINO, Miho, SUZUKI, Gentaroh, TAKEHANA, Hiroshi, HATA, Mikiko
Published in European journal of pharmacology (2010)
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Published in European journal of pharmacology (2010)
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Face-washing behavior induced by the group I metabotropic glutamate receptor agonist ( S)-3,5-DHPG in mice is mediated by mGlu 1 receptor
Hikichi, Hirohiko, Iwahori, Yuki, Murai, Takeshi, Maehara, Shunsuke, Satow, Akio, Ohta, Hisashi
Published in European journal of pharmacology (2008)
Published in European journal of pharmacology (2008)
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Journal Article
Unique Antipsychotic Activities of the Selective Metabotropic Glutamate Receptor 1 Allosteric Antagonist 2-Cyclopropyl-5-[1-(2-fluoro-3-pyridinyl)-5-methyl-1 H -1,2,3-triazol-4-yl]-2,3-dihydro-1 H -isoindol-1-one
Satow, Akio, Suzuki, Gentaroh, Maehara, Shunsuke, Hikichi, Hirohiko, Murai, Takeshi, Murai, Takashi, Kawagoe-Takaki, Hiroko, Hata, Mikiko, Ito, Satoru, Ozaki, Satoshi, Kawamoto, Hiroshi, Ohta, Hisashi
Published in The Journal of pharmacology and experimental therapeutics (01.07.2009)
Published in The Journal of pharmacology and experimental therapeutics (01.07.2009)
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Journal Article
Antipsychotic effects of N-desmethylclozapine on sensorimotor gating function in rats--possible involvement of activation of M(1) muscarinic receptors
Maehara, Shunsuke, Satow, Akio, Hikichi, Hirohiko, Ohta, Hisashi
Published in European journal of pharmacology (30.09.2011)
Published in European journal of pharmacology (30.09.2011)
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