Development of a Scalable Process for the Synthesis of DNDI-VL-2098: A Potential Preclinical Drug Candidate for the Treatment of Visceral Leishmaniasis
Satam, Vijay S, Pedada, Srinivasa Rao, Kamaraj, Pasumpon, Antao, Nakita, Singh, Apoorva, Hindupur, Rama Mohan, Pati, Hari N, Thompson, Andrew M, Launay, Delphine, Martin, Denis
Published in Organic process research & development (20.01.2017)
Published in Organic process research & development (20.01.2017)
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Synthesis of highly fluorescent coumarinyl chalcones derived from 8-acetyl-1,4-diethyl-1,2,3,4-tetrahydro-7H-pyrano[2,3-g]quinoxalin-7-one and their spectral characteristics
Jagtap, Amit R, Satam, Vijay S, Rajule, Rajkumar N, Kanetkar, Vinod R
Published in Dyes and pigments (01.10.2011)
Published in Dyes and pigments (01.10.2011)
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Correction to “Development of a Scalable Process for the Synthesis of DNDI-VL-2098: A Potential Preclinical Drug Candidate for the Treatment of Visceral Leishmaniasis”
Satam, Vijay S, Pedada, Srinivasa Rao, Kandadai, Srinivas A, Kamaraj, Pasumpon, Antao, Nakita, Singh, Apoorva, Hindupur, Rama Mohan, Pati, Hari N, Thompson, Andrew M, Launay, Delphine, Martin, Denis
Published in Organic process research & development (21.04.2017)
Published in Organic process research & development (21.04.2017)
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Journal Article
An Improved Kilogram-Scale Synthesis of 2‑Bromo-4-nitro‑1H‑imidazole: A Key Building Block of Nitroimidazole Drugs
Pedada, Srinivasa Rao, Satam, Vijay S, Tambade, Pawan J, Kandadai, Srinivas A, Hindupur, Rama Mohan, Pati, Hari N, Launay, Delphine, Martin, Denis
Published in Organic process research & development (20.09.2013)
Published in Organic process research & development (20.09.2013)
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Journal Article
Synthesis, cytotoxicity, and structure–activity insight of NH- and N-methyl-3,5-bis-(arylidenyl)-4-piperidones
Gregory, Matthew, Dandavati, Armaan, Lee, Megan, Tzou, Samuel, Savagian, Mia, Brien, Kimberly A., Satam, Vijay, Patil, Pravin, Lee, Moses
Published in Medicinal chemistry research (01.11.2013)
Published in Medicinal chemistry research (01.11.2013)
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Journal Article
Practical Synthesis of 6‑Amino-1-hydroxy-2,1-benzoxaborolane: A Key Intermediate of DNDI-6148
Khairnar, Pankaj V., Saathoff, John M., Cook, Daniel W., Hochstetler, Samuel R., Pandya, Urvish, Robinson, Stephen J., Satam, Vijay, Donsbach, Kai O., Gupton, B. Frank, Jin, Li-Mei, Shanahan, Charles S.
Published in Organic process research & development (19.04.2024)
Published in Organic process research & development (19.04.2024)
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Effects of N-terminus modified Hx-amides on DNA binding affinity, sequence specificity, cellular uptake, and gene expression
Kiakos, Konstantinos, Satam, Vijay, Patil, Pravin C., Sweers, Jeffrey, Bowerman, Michael, Tzou, Sam, Olsen, Kevin, Lee, Megan, Schaschl, Helmut, Keppler, Bernhard K., Hochhauser, Daniel, Lee, Moses, Hartley, John A., Pett, Luke
Published in Bioorganic & medicinal chemistry letters (01.09.2021)
Published in Bioorganic & medicinal chemistry letters (01.09.2021)
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Journal Article
Nuclear Localization and Gene Expression Modulation by a Fluorescent Sequence-Selective p-Anisyl-benzimidazolecarboxamido Imidazole-Pyrrole Polyamide
Kiakos, Konstantinos, Pett, Luke, Satam, Vijay, Patil, Pravin, Hochhauser, Daniel, Lee, Moses, Hartley, John A.
Published in Chemistry & biology (23.07.2015)
Published in Chemistry & biology (23.07.2015)
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PA-298 Predicting disease effect on the pharmacokinetics (PK) of sustained and immediate release formulations by applying physiologically based pharmacokinetic (PBPK) modelling
Eriksson, Johanna, Sjögren, Eric, Gillon, Jean-Yves, Goyal, Vishal, Satam, Vijay, Robinson, Stephen, Caplain, Henri, Ribeiro, Isabela, Chenel, Marylore
Published in BMJ global health (17.12.2023)
Published in BMJ global health (17.12.2023)
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Journal Article
Abstract 3755: Genome-wide transcriptome analysis reveals the distinct gene expression profiles and specific biological effects of fluorescent polyamides, HxIP and azaHxPI
Pett, Luke, Satam, Vijay, Patil, Pravin, Lee, Moses, Hartley, John A., Kiakos, Konstantinos
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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DNA-binding properties of new fluorescent AzaHx-amides: Methoxy-pyridyl-aza-benzimidazole-pyrrole-imidazole/pyrrole
Liu, Beibei, Pett, Luke, Kiakos, Konstantinos, Patil, Pravin, Satam, Vijay, Hartley, John A., Lee, Moses, Wilson, W.David
Published in Chembiochem : a European journal of chemical biology (15.08.2018)
Published in Chembiochem : a European journal of chemical biology (15.08.2018)
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Bioavailability of a novel sustained‐release pellet formulation of 5‐flucytosine in healthy‐fed participants for use in patients with cryptococcal meningitis
Ibnou Zekri Lassout, Nabila, Goyal, Vishal, Krantz, Edrich, Simon, Francois, Neven, Anouk, Eriksson, Johanna, Saayman, Amaria, Satam, Vijay, Ruffell, Carol, Victor, Sarika, Chenel, Marylore, Celebic, Aljosa, Caplain, Henri, Gillon, Jean‐Yves, Deshmukh, Abhijit, Antarkar, Amit, Sjögren, Eric, Ribeiro, Isabela
Published in Clinical and translational science (01.09.2024)
Published in Clinical and translational science (01.09.2024)
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DNA‐Binding Properties of New Fluorescent AzaHx Amides: Methoxypyridylazabenzimidazolepyrroleimidazole/pyrrole
Liu, Beibei, Pett, Luke, Kiakos, Konstantinos, Patil, Pravin C., Satam, Vijay, Hartley, John A., Lee, Moses, Wilson, W. David
Published in Chembiochem : a European journal of chemical biology (17.09.2018)
Published in Chembiochem : a European journal of chemical biology (17.09.2018)
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Journal Article
A novel class of trans-methylpyrazoline analogs of combretastatins: Synthesis and in-vitro biological testing
Lee, Megan, Brockway, Olivia, Dandavati, Armaan, Tzou, Samuel, Sjoholm, Robert, Satam, Vijay, Westbrook, Cara, Mooberry, Susan L., Zeller, Matthias, Babu, Balaji, Lee, Moses
Published in European journal of medicinal chemistry (01.07.2011)
Published in European journal of medicinal chemistry (01.07.2011)
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