An Aldol-Based Build/Couple/Pair Strategy for the Synthesis of Medium- and Large-Sized Rings: Discovery of Macrocyclic Histone Deacetylase Inhibitors
Marcaurelle, Lisa A, Comer, Eamon, Dandapani, Sivaraman, Duvall, Jeremy R, Gerard, Baudouin, Kesavan, Sarathy, Lee, Maurice D, Liu, Haibo, Lowe, Jason T, Marie, Jean-Charles, Mulrooney, Carol A, Pandya, Bhaumik A, Rowley, Ann, Ryba, Troy D, Suh, Byung-Chul, Wei, Jingqiang, Young, Damian W, Akella, Lakshmi B, Ross, Nathan T, Zhang, Yan-Ling, Fass, Daniel M, Reis, Surya A, Zhao, Wen-Ning, Haggarty, Stephen J, Palmer, Michelle, Foley, Michael A
Published in Journal of the American Chemical Society (01.12.2010)
Published in Journal of the American Chemical Society (01.12.2010)
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Synthesis and Profiling of a Diverse Collection of Azetidine-Based Scaffolds for the Development of CNS-Focused Lead-like Libraries
Lowe, Jason T, Lee, Maurice D, Akella, Lakshmi B, Davoine, Emeline, Donckele, Etienne J, Durak, Landon, Duvall, Jeremy R, Gerard, Baudouin, Holson, Edward B, Joliton, Adrien, Kesavan, Sarathy, Lemercier, Berenice C, Liu, Haibo, Marié, Jean-Charles, Mulrooney, Carol A, Muncipinto, Giovanni, Welzel-O’Shea, Morgan, Panko, Laura M, Rowley, Ann, Suh, Byung-Chul, Thomas, Meryl, Wagner, Florence F, Wei, Jingqiang, Foley, Michael A, Marcaurelle, Lisa A
Published in Journal of organic chemistry (07.09.2012)
Published in Journal of organic chemistry (07.09.2012)
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Enantioselective Synthesis of Linear Polypropionate Arrays Using Anthracene-Tagged Organosilanes
Kesavan, Sarathy, Su, Qibin, Shao, Jian, Porco, John A, Panek, James S
Published in Organic letters (29.09.2005)
Published in Organic letters (29.09.2005)
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Discovery of Novel, Orally Bioavailable Pyrimidine Ether-Based Inhibitors of ELOVL1
Boyd, Michael J, Collier, Philip N, Clark, Michael P, Deng, Hongbo, Kesavan, Sarathy, Ronkin, Steven M, Waal, Nathan, Wang, Jian, Cao, Jingrong, Li, Pan, Come, Jon, Davies, Ioana, Duffy, John P, Cochran, John E, Court, John J, Chandupatla, Kishan, Jackson, Katrina L, Maltais, Francois, O’Dowd, Hardwin, Boucher, Christina, Considine, Tony, Taylor, William P, Gao, Hong, Chakilam, Ananthisrinivas, Engtrakul, Juntyma, Crawford, Dan, Doyle, Elizabeth, Phillips, Jonathan, Kemper, Raymond, Swett, Rebecca, Empfield, James, Bunnage, Mark E, Charifson, Paul S, Magavi, Sanjay Shivayogi
Published in Journal of medicinal chemistry (23.12.2021)
Published in Journal of medicinal chemistry (23.12.2021)
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Application of a Catalytic Asymmetric Povarov Reaction using Chiral Ureas to the Synthesis of a Tetrahydroquinoline Library
Gerard, Baudouin, O’Shea, Morgan Welzel, Donckele, Etienne, Kesavan, Sarathy, Akella, Lakshmi B, Xu, Hao, Jacobsen, Eric N, Marcaurelle, Lisa A
Published in ACS combinatorial science (12.11.2012)
Published in ACS combinatorial science (12.11.2012)
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Accessing Skeletal Diversity Using Catalyst Control: Formation of n and n + 1 Macrocyclic Triazole Rings
Kelly, Ann Rowley, Wei, Jingqiang, Kesavan, Sarathy, Marié, Jean-Charles, Windmon, Nicole, Young, Damian W, Marcaurelle, Lisa A
Published in Organic letters (04.06.2009)
Published in Organic letters (04.06.2009)
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Synthesis of Stereochemically and Skeletally Diverse Fused Ring Systems from Functionalized C‑Glycosides
Gerard, Baudouin, Lee, Maurice D, Dandapani, Sivaraman, Duvall, Jeremy R, Fitzgerald, Mark E, Kesavan, Sarathy, Lowe, Jason T, Marié, Jean-Charles, Pandya, Bhaumik A, Suh, Byung-Chul, O’Shea, Morgan Welzel, Dombrowski, Michael, Hamann, Diane, Lemercier, Berenice, Murillo, Tiffanie, Akella, Lakshmi B, Foley, Michael A, Marcaurelle, Lisa A
Published in Journal of organic chemistry (07.06.2013)
Published in Journal of organic chemistry (07.06.2013)
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Journal Article
Application of a Catalytic Asymmetric Povarov Reaction using Chiral Ureas to the Synthesis of a Tetrahyroquinoline Library
Gerard, Baudouin, O’Shea, Morgan Welzel, Donckele, Etienne, Kesavan, Sarathy, Akella, Lakshmi B., Xu, Hao, Jacobsen, Eric N., Marcaurelle, Lisa A.
Published in ACS combinatorial science (22.10.2012)
Published in ACS combinatorial science (22.10.2012)
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Journal Article
Correction to Application of a Catalytic Asymmetric Povarov Reaction using Chiral Ureas to the Synthesis of a Tetrahydroquinoline Library
Gerard, Baudouin, O’Shea, Morgan Welzel, Donckele, Etienne, Kesavan, Sarathy, Akella, Lakshmi B, Xu, Hao, Jacobsen, Eric N, Marcaurelle, Lisa A
Published in ACS combinatorial science (13.01.2014)
Published in ACS combinatorial science (13.01.2014)
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Toward the Molecular Flashlight: Preparation, Properties, and Photophysics of a Hypericin–luciferin Tethered Molecule
Wen, Jin, Chowdhury, Pramit, Wills, Nick J., Wannemuehler, Yvonne, Park, Jaehun, Kesavan, Sarathy, Carpenter, S., Kraus, G. A., Petrich, J. W.
Published in Photochemistry and photobiology (01.08.2002)
Published in Photochemistry and photobiology (01.08.2002)
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Journal Article
Tumor Cell Toxicity of Hypericin and Related Analogs
Wills, Nick J., Park, Jaehun, Wen, Jin, Kesavan, Sarathy, Kraus, George A., Petrich, Jacob W., Carpenter, Susan
Published in Photochemistry and photobiology (01.08.2001)
Published in Photochemistry and photobiology (01.08.2001)
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Journal Article
Toward the Molecular Flashlight: Preparation, Properties, and Photophysics of a Hypericin-luciferin Tethered Molecule
Wen, Jin, Chowdhury, Pramit, Wills, Nick J., Wannemuehler, Yvonne, Park, Jaehun, Kesavan, Sarathy, Carpenter, S., Kraus, G. A., Petrich, J. W.
Published in Photochemistry and photobiology (01.08.2002)
Published in Photochemistry and photobiology (01.08.2002)
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Journal Article
Tumor Cell Toxicity of Hypericin and Related Analogs
Wills, Nick J., Park, Jaehun, Wen, Jin, Kesavan, Sarathy, Kraus, George A., Petrich, Jacob W., Carpenter, Susan
Published in Photochemistry and photobiology (01.08.2001)
Published in Photochemistry and photobiology (01.08.2001)
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