Search Results - "SANTOSH S KULKARNI" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Fragment-Based Discovery of New Highly Substituted 1H‑Pyrrolo[2,3‑b]- and 3H‑Imidazolo[4,5‑b]‑Pyridines as Focal Adhesion Kinase Inhibitors

Fragment-Based Discovery of New Highly Substituted 1H‑Pyrrolo[2,3‑b]- and 3H‑Imidazolo[4,5‑b]‑Pyridines as Focal Adhesion Kinase Inhibitors

by Heinrich, Timo, Seenisamy, Jeyaprakashnarayanan, Emmanuvel, Lourdusamy, Kulkarni, Santosh S, Bomke, Jörg, Rohdich, Felix, Greiner, Hartmut, Esdar, Christina, Krier, Mireille, Grädler, Ulrich, Musil, Djordje
Published in Journal of medicinal chemistry (14.02.2013)

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Journal Article

Enantioselective Synthesis and Physicochemical Properties of Libraries of 3-Amino- and 3-Amidofluoropiperidines

Enantioselective Synthesis and Physicochemical Properties of Libraries of 3-Amino- and 3-Amidofluoropiperidines

by Orliac, Aurélie, Routier, Julie, Burgat Charvillon, Fabienne, Sauer, Wolfgang H. B., Bombrun, Agnes, Kulkarni, Santosh S., Gomez Pardo, Domingo, Cossy, Janine
Published in Chemistry : a European journal (24.03.2014)

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Journal Article

Inhibition of Human Acetyl- and Butyrylcholinesterase by Novel Carbamates of (−)- and (+)-Tetrahydrofurobenzofuran and Methanobenzodioxepine

Inhibition of Human Acetyl- and Butyrylcholinesterase by Novel Carbamates of (−)- and (+)-Tetrahydrofurobenzofuran and Methanobenzodioxepine

by Luo, Weiming, Yu, Qian-sheng, Kulkarni, Santosh S, Parrish, Damon A, Holloway, Harold W, Tweedie, David, Shafferman, Avigdor, Lahiri, Debomoy K, Brossi, Arnold, Greig, Nigel H
Published in Journal of medicinal chemistry (06.04.2006)

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Journal Article

Recognition of Benztropine by the Dopamine Transporter (DAT) Differs from That of the Classical Dopamine Uptake Inhibitors Cocaine, Methylphenidate, and Mazindol as a Function of a DAT Transmembrane 1 Aspartic Acid Residue

Recognition of Benztropine by the Dopamine Transporter (DAT) Differs from That of the Classical Dopamine Uptake Inhibitors Cocaine, Methylphenidate, and Mazindol as a Function of a DAT Transmembrane 1 Aspartic Acid Residue

by Ukairo, Okechukwu T, Bondi, Corry D, Newman, Amy Hauck, Kulkarni, Santosh S, Kozikowski, Alan P, Pan, Stephen, Surratt, Christopher K
Published in The Journal of pharmacology and experimental therapeutics (01.08.2005)

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Journal Article

Localization of Cocaine Analog [125I]RTI 82 Irreversible Binding to Transmembrane Domain 6 of the Dopamine Transporter

Localization of Cocaine Analog [125I]RTI 82 Irreversible Binding to Transmembrane Domain 6 of the Dopamine Transporter

by Vaughan, Roxanne A., Sakrikar, Dhananjay S., Parnas, M. Laura, Adkins, Steven, Foster, James D., Duval, Romain A., Lever, John R., Kulkarni, Santosh S., Hauck-Newman, Amy
Published in The Journal of biological chemistry (23.03.2007)

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Journal Article

Discovery of heterobicyclic templates for novel metabotropic glutamate receptor subtype 5 antagonists

Discovery of heterobicyclic templates for novel metabotropic glutamate receptor subtype 5 antagonists

by Kulkarni, Santosh S., Newman, Amy Hauck
Published in Bioorganic & medicinal chemistry letters (01.06.2007)

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Journal Article

Three-dimensional quantitative structure activity relationships (3-D-QSAR) of antihyperglycemic agents

Three-dimensional quantitative structure activity relationships (3-D-QSAR) of antihyperglycemic agents

by KULKARNI, S. S, GEDIYA, L. K, KULKARNI, V. M
Published in Bioorganic & medicinal chemistry (01.07.1999)

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Journal Article

Synthesis of CJ-15,208, a novel κ-opioid receptor antagonist

Synthesis of CJ-15,208, a novel κ-opioid receptor antagonist

by Ross, Nicolette C., Kulkarni, Santosh S., McLaughlin, Jay P., Aldrich, Jane V.
Published in Tetrahedron letters (20.09.2010)

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Journal Article

Structure−Activity Relationships Comparing N-(6-Methylpyridin-yl)-Substituted Aryl Amides to 2-Methyl-6-(substituted-arylethynyl)pyridines or 2-Methyl-4-(substituted-arylethynyl)thiazoles as Novel Metabotropic Glutamate Receptor Subtype 5 Antagonists

Structure−Activity Relationships Comparing N-(6-Methylpyridin-yl)-Substituted Aryl Amides to 2-Methyl-6-(substituted-arylethynyl)pyridines or 2-Methyl-4-(substituted-arylethynyl)thiazoles as Novel Metabotropic Glutamate Receptor Subtype 5 Antagonists

by Kulkarni, Santosh S, Zou, Mu-Fa, Cao, Jianjing, Deschamps, Jeffrey R, Rodriguez, Alice L, Conn, P. Jeffrey, Newman, Amy Hauck
Published in Journal of medicinal chemistry (11.06.2009)

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Journal Article

Design and synthesis of novel heterobiaryl amides as metabotropic glutamate receptor subtype 5 antagonists

Design and synthesis of novel heterobiaryl amides as metabotropic glutamate receptor subtype 5 antagonists

by Kulkarni, Santosh S., Newman, Amy Hauck
Published in Bioorganic & medicinal chemistry letters (01.04.2007)

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Journal Article

Unexpected Opioid Activity Profiles of Analogues of the Novel Peptide Kappa Opioid Receptor Ligand CJ-15,208

Unexpected Opioid Activity Profiles of Analogues of the Novel Peptide Kappa Opioid Receptor Ligand CJ-15,208

by Aldrich, Jane V., Kulkarni, Santosh S., Senadheera, Sanjeewa N., Ross, Nicolette C., Reilley, Kate J., Eans, Shainnel O., Ganno, Michelle L., Murray, Thomas F., McLaughlin, Jay P.
Published in ChemMedChem (05.09.2011)

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Journal Article

Synthesis of cyclic tetrapeptide CJ 15,208: a novel kappa opioid receptor antagonist

Synthesis of cyclic tetrapeptide CJ 15,208: a novel kappa opioid receptor antagonist

by Kulkarni, Santosh S, Ross, Nicolette C, McLaughlin, Jay P, Aldrich, Jane V
Published in Advances in experimental medicine and biology (2009)

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Journal Article

Novel Anticholinesterases Based on the Molecular Skeletons of Furobenzofuran and Methanobenzodioxepine

Novel Anticholinesterases Based on the Molecular Skeletons of Furobenzofuran and Methanobenzodioxepine

by Luo, Weiming, Yu, Qian-sheng, Zhan, Ming, Parrish, Damon, Deschamps, Jeffrey R, Kulkarni, Santosh S, Holloway, Harold W, Alley, George M, Lahiri, Debomoy K, Brossi, Arnold, Greig, Nigel H
Published in Journal of medicinal chemistry (24.02.2005)

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Journal Article

Structure−Activity Relationships at Monoamine Transporters for a Series of N-Substituted 3α-(Bis[4-fluorophenyl]methoxy)tropanes: Comparative Molecular Field Analysis, Synthesis, and Pharmacological Evaluation

Structure−Activity Relationships at Monoamine Transporters for a Series of N-Substituted 3α-(Bis[4-fluorophenyl]methoxy)tropanes: Comparative Molecular Field Analysis, Synthesis, and Pharmacological Evaluation

by Kulkarni, Santosh S, Grundt, Peter, Kopajtic, Theresa, Katz, Jonathan L, Newman, Amy Hauck
Published in Journal of medicinal chemistry (17.06.2004)

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Journal Article

GLYCOSIDASE INHIBITOR

GLYCOSIDASE INHIBITOR

by ANNA QUATTROPANI, SANTOSH S KULKARNI, AWADUT GAJENDRA GIRI
Year of Publication 05.12.2019

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Patent

Design and synthesis of noncompetitive metabotropic glutamate receptor subtype 5 antagonists

Design and synthesis of noncompetitive metabotropic glutamate receptor subtype 5 antagonists

by Kulkarni, Santosh S., Nightingale, Barbara, Dersch, Christina M., Rothman, Richard B., Newman, Amy Hauck
Published in Bioorganic & medicinal chemistry letters (01.07.2006)

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Journal Article

Design and synthesis of cyclic arodyn analogues by ring-closing metathesis (RCM) for kappa opioid receptor (KOP) antagonists

Design and synthesis of cyclic arodyn analogues by ring-closing metathesis (RCM) for kappa opioid receptor (KOP) antagonists

by Fang, Wei-Jie, Kulkarni, Santosh S, Murray, Thomas F, Aldrich, Jane V
Published in Advances in experimental medicine and biology (2009)

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Journal Article

Dual Probes for the Dopamine Transporter and σ1 Receptors: Novel Piperazinyl Alkyl-bis(4‘-fluorophenyl)amine Analogues as Potential Cocaine-Abuse Therapeutic Agents

Dual Probes for the Dopamine Transporter and σ1 Receptors: Novel Piperazinyl Alkyl-bis(4‘-fluorophenyl)amine Analogues as Potential Cocaine-Abuse Therapeutic Agents

by Cao, Jianjing, Kulkarni, Santosh S, Husbands, Stephen M, Bowen, Wayne D, Williams, Wanda, Kopajtic, Theresa, Katz, Jonathan L, George, Clifford, Newman, Amy Hauck
Published in Journal of medicinal chemistry (19.06.2003)

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Journal Article

Three-Dimensional Quantitative Structure−Activity Relationships of Mazindol Analogues at the Dopamine Transporter

Three-Dimensional Quantitative Structure−Activity Relationships of Mazindol Analogues at the Dopamine Transporter

by Kulkarni, Santosh S, Newman, Amy Hauck, Houlihan, William J
Published in Journal of medicinal chemistry (12.09.2002)

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Journal Article

Three-Dimensional Quantitative Structure−Activity Relationship of Interleukin 1-β Converting Enzyme Inhibitors: A Comparative Molecular Field Analysis Study

Three-Dimensional Quantitative Structure−Activity Relationship of Interleukin 1-β Converting Enzyme Inhibitors: A Comparative Molecular Field Analysis Study

by Kulkarni, Santosh S, Kulkarni, Vithal M
Published in Journal of medicinal chemistry (11.02.1999)

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Journal Article

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