Optimization of Alkylidene Hydrazide Based Human Glucagon Receptor Antagonists. Discovery of the Highly Potent and Orally Available 3-Cyano-4-hydroxybenzoic Acid [1-(2,3,5,6-Tetramethylbenzyl)-1H-indol-4-ylmethylene]hydrazide
Madsen, Peter, Ling, Anthony, Plewe, Michael, Sams, Christian K, Knudsen, Lotte B, Sidelmann, Ulla G, Ynddal, Lars, Brand, Christian L, Andersen, Birgitte, Murphy, Douglas, Teng, Min, Truesdale, Larry, Kiel, Dan, May, John, Kuki, Atsuo, Shi, Shenghua, Johnson, Michael D, Teston, Kimberly Ann, Feng, Jun, Lakis, James, Anderes, Kenna, Gregor, Vlad, Lau, Jesper
Published in Journal of medicinal chemistry (19.12.2002)
Published in Journal of medicinal chemistry (19.12.2002)
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Human glucagon receptor antagonists based on alkylidene hydrazides
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Published in Bioorganic & medicinal chemistry letters (25.02.2002)
Published in Bioorganic & medicinal chemistry letters (25.02.2002)
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Novel Glucagon Receptor Antagonists with Improved Selectivity over the Glucose-Dependent Insulinotropic Polypeptide Receptor
Kodra, János T, Jørgensen, Anker Steen, Andersen, Birgitte, Behrens, Carsten, Brand, Christian Lehn, Christensen, Inger Thøger, Guldbrandt, Mette, Jeppesen, Claus Bekker, Knudsen, Lotte B, Madsen, Peter, Nishimura, Erica, Sams, Christian, Sidelmann, Ulla G, Pedersen, Raymon A, Lynn, Francis C, Lau, Jesper
Published in Journal of medicinal chemistry (11.09.2008)
Published in Journal of medicinal chemistry (11.09.2008)
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New β-Alanine Derivatives Are Orally Available Glucagon Receptor Antagonists
Lau, Jesper, Behrens, Carsten, Sidelmann, Ulla G, Knudsen, Lotte B, Lundt, Behrend, Sams, Christian, Ynddal, Lars, Brand, Christian L, Pridal, Lone, Ling, Anthony, Kiel, Dan, Plewe, Michael, Shi, Shengua, Madsen, Peter
Published in Journal of medicinal chemistry (11.01.2007)
Published in Journal of medicinal chemistry (11.01.2007)
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Coordination chemistry of transition metal complexes of a novel pentadentate ligand
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Published in Inorganica Chimica Acta (18.06.2001)
Published in Inorganica Chimica Acta (18.06.2001)
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Year of Publication 18.07.2023
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Year of Publication 18.07.2023
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Year of Publication 11.05.2021
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Year of Publication 28.03.2022
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Year of Publication 28.02.2022
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Year of Publication 15.11.2021
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Year of Publication 25.10.2021
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Year of Publication 25.02.2020
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Year of Publication 11.08.2021
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