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Synthesis and structure–activity studies of novel benzocycloheptanone oxazolidinone antibacterial agents
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In Vitro and In Vivo Activities of Syn2190, a Novel β-Lactamase Inhibitor
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Boys, Mark L., Bian, Feng, Kramer, James B., Chio, Christopher L., Ren, Xiao-Dan, Chen, Huifen, Barrett, Stephen D., Sexton, Karen E., Iula, Donna M., Filzen, Gary F., Nguyen, Maria N., Angell, Paul, Downs, Victoria L., Wang, Zhi, Raheja, Neil, Ellsworth, Edmund L., Fakhoury, Stephen, Bratton, Larry D., Keller, Paul R., Gowan, Richard, Drummond, Elena M., Maiti, Samarendra N., Hena, Mostofa A., Lu, Leroy, McConnell, Patrick, Knafels, John D., Thanabal, Venkataraman, Sun, Fang, Alessi, Diane, McCarthy, Ann, Zhang, Erli, Finzel, Barry C., Patel, Sneha, Ciotti, Susan M., Eisma, Rone, Payne, N.A., Gilbertsen, Richard B., Kostlan, Catherine R., Pocalyko, David J., Lala, Deepak S.
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Discovery of 6-ethyl-2,4-diaminopyrimidine-based small molecule renin inhibitors
Holsworth, Daniel D., Jalaie, Mehran, Belliotti, Thomas, Cai, Cuiman, Collard, Wendy, Ferreira, Suzie, Powell, Noel A., Stier, Michael, Zhang, Erli, McConnell, Pat, Mochalkin, Igor, Ryan, Michael J., Bryant, John, Li, Tingsheng, Kasani, Aparna, Subedi, Rajendra, Maiti, Samarendra N., Edmunds, Jeremy J.
Published in Bioorganic & medicinal chemistry letters (01.07.2007)
Published in Bioorganic & medicinal chemistry letters (01.07.2007)
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Synthesis and SAR of novel conformationally-restricted oxazolidinones possessing Gram-positive and fastidious Gram-negative antibacterial activity. Part 1: Substituted pyrazoles
Boyer, Frederick E., Vara Prasad, J.V.N., Choy, Allison L., Chupak, Louis, Dermyer, Michael R., Ding, Qizhu, Huband, Michael D., Jiao, Wenhua, Kaneko, Takushi, Khlebnikov, Vladimir, Kim, Ji-Young, Lall, Manjinder S., Maiti, Samarendra N., Romero, Karina, Wu, Xiujuan
Published in Bioorganic & medicinal chemistry letters (15.08.2007)
Published in Bioorganic & medicinal chemistry letters (15.08.2007)
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Design, synthesis, and pharmacological evaluation of phenoxy pyridyl derivatives as dual norepinephrine reuptake inhibitors and 5-HT1A partial agonists
DOUNAY, Amy B, BARTA, Nancy S, MAITI, Samarendra N, ORTWINE, Daniel F, PROBERT, Al, STRATMAN, Nancy C, SUBEDI, Rajendra, WHISMAN, Tammy, WENJIAN XU, ZOSKI, Kim, CAMPBELL, Brian M, COLEMAN, Corey, COLLANTES, Elizabeth M, DENNY, Lynne, DUTTA, Satavisha, GRAY, David L, DONGFENG HOU, IYER, Rathna
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
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Synthesis of fluorinated 1,8-naphthyridinone derivatives
Repine, Joseph T., Johnson, Douglas S., Stuk, Timothy, White, Andrew D., Stier, Michael A., Li, Tingsheng, Yang, Zhixiang, Maiti, Samarendra N.
Published in Tetrahedron letters (12.11.2007)
Published in Tetrahedron letters (12.11.2007)
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(1 R ,2 S )-4-(2-Cyano-cyclohexyl-oxy)-2-trifluoromethyl-benzonitrile, a potent androgen receptor antagonist for stimulating hair growth and reducing sebum production
Hu, Lain-Yen, Du, Daniel, Hoffman, Jennifer, Smith, Yvonne, Fedij, Victor, Kostlan, Catherine, Johnson, Theodore R., Huang, Yun, Kesten, Steve, Harter, William, Yue, Wen Song, Li, Jie Jack, Barvian, Nicole, Mitchell, Lorna, Lei, Huangshu John, Lefker, Bruce, Carroll, Mathew, Dettling, Danielle, Krieger-Burke, Teresa, Samas, Brian, Yalamanchili, Radhika, Lapham, Kimberly, Pocalyko, David, Sliskovic, Drago, Ciotti, Susan, Stoller, Brenda, Hena, Mostofa A., Ding, Qizhu, Maiti, Samarendra N., Stier, Michael, Welgus, Howard
Published in Bioorganic & medicinal chemistry letters (01.11.2007)
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The discovery of glycine and related amino acid-based factor Xa inhibitors
Kohrt, Jeffrey T., Filipski, Kevin J., Cody, Wayne L., Bigge, Christopher F., La, Frances, Welch, Kathleen, Dahring, Tawny, Bryant, John W., Leonard, Daniele, Bolton, Gary, Narasimhan, Lakshmi, Zhang, Erli, Peterson, J. Thomas, Haarer, Staci, Sahasrabudhe, Vaishali, Janiczek, Nancy, Desiraju, Shrilakshmi, Hena, Mostofa, Fiakpui, Charles, Saraswat, Neerja, Sharma, Raman, Sun, Shaoyi, Maiti, Samarendra N., Leadley, Robert, Edmunds, Jeremy J.
Published in Bioorganic & medicinal chemistry (01.07.2006)
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Synthesis and biological evaluation of penam sulfones as inhibitors of β-lactamases
Phillips, Oludotun A., Reddy, Andhe V.N., Setti, Eduardo L., Spevak, Paul, Czajkowski, David P., Atwal, Herninder, Salama, Sameeh, Micetich, Ronald G., Maiti, Samarendra N.
Published in Bioorganic & medicinal chemistry (15.04.2005)
Published in Bioorganic & medicinal chemistry (15.04.2005)
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Synthesis of 4-(R)-Naphthalene-2-yloxy-1-(1-Phenyl-(S)-Ethyl)-Pyrrolidin-3-(R)-ol and 4-(S)-Naphthalen-2-yloxy-1-(1-Phenyl-(S)-Ethyl)-Pyrrolidin-3-(S)-ol: Versatile Chiral Intermediates for Synthesis
Holsworth, Daniel D., Stier, Michael, Wang, Wei, Edmunds, Jeremy J., Li, Tingsheng, Maiti, Samarendra N.
Published in Synthetic communications (31.12.2004)
Published in Synthetic communications (31.12.2004)
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Synthesis and .beta.-lactamase inhibitory properties of 2.beta.-[(1,2,3-triazol-1-yl)methyl]-2.alpha.-methylpenam-3.alpha.-carboxylic acid 1,1-dioxide and related triazolyl derivatives
Micetich, Ronald G, Maiti, Samarendra N, Spevak, Paul, Hall, Tse W, Yamabe, Shigeru, Ishida, Naobumi, Tanaka, Motoaki, Yamazaki, Tomio, Nakai, Akira, Ogawa, Kazuo
Published in Journal of medicinal chemistry (01.08.1987)
Published in Journal of medicinal chemistry (01.08.1987)
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Synthesis and .BETA.-lactamase inhibitory activity of 6-((1-heteroarylthioethyl-1,2,3-triazol4-yl)methylene)-penam sulfones
IM, CHAEUK, MAITI, SAMARENDRA N., MICETICH, RONALD G., DANESHXALAB, MOHSEN, ATCHISON, KEVIN, PHILLIPS, OLUDOTUN A., KUNUGITA, CHIEKO
Published in Journal of antibiotics (1994)
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Studies on penam sulfones III. Synthesis and β-lactamase inhibitory activity of sodium (6R)-6-(α-hydroxybenzyl)-2β-methoxyiminomethyl-2α-methylpenam-3α-carboxylate 1,1-dioxide and sodium 2β-acyl-2α-methylpenam-3α-carboxylate 1,1-dioxide
Czajkowski, David P, Reddy, Andhe V.N, Setti, Eduardo L, Phillips, Oludotun A, Micetich, Ronald G, Kunugita, Chieko, Maiti, Samarendra N
Published in Bioorganic & medicinal chemistry letters (1997)
Published in Bioorganic & medicinal chemistry letters (1997)
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A versatile copper-catalyzed coupling reaction of pyridin-2(1 H)-ones with aryl halides
Filipski, Kevin J., Kohrt, Jeffrey T., Casimiro-Garcia, Agustin, Van Huis, Chad A., Dudley, Danette A., Cody, Wayne L., Bigge, Christopher F., Desiraju, Shrilakshmi, Sun, Shaoyi, Maiti, Samarendra N., Jaber, Mohamad R., Edmunds, Jeremy J.
Published in Tetrahedron letters (30.10.2006)
Published in Tetrahedron letters (30.10.2006)
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Studies on Penam Sulfones. II. Synthesis and .BETA.-Lactamase Inhibitory Activity of 2.BETA.-Carboxamide Penicillanic Acid Sulfones
REDDY, NARENDER A. V., SETTI, EDUARDO L., PHILLIPS, OLUDOTUN A., CZAJKOWSKI, DAVID P., ATWAL, HARNINDER, ATCHISON, KEVIN, MICETICH, RONALD G., MAITI, SAMARENDRA N., KUNUGITA, CHIEKO, HYODO, AKIO
Published in Journal of antibiotics (1997)
Published in Journal of antibiotics (1997)
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