Targeting the MAPK Signaling Pathway in Cancer: Promising Preclinical Activity with the Novel Selective ERK1/2 Inhibitor BVD-523 (Ulixertinib)
Germann, Ursula A, Furey, Brinley F, Markland, William, Hoover, Russell R, Aronov, Alex M, Roix, Jeffrey J, Hale, Michael, Boucher, Diane M, Sorrell, David A, Martinez-Botella, Gabriel, Fitzgibbon, Matthew, Shapiro, Paul, Wick, Michael J, Samadani, Ramin, Meshaw, Kathryn, Groover, Anna, DeCrescenzo, Gary, Namchuk, Mark, Emery, Caroline M, Saha, Saurabh, Welsch, Dean J
Published in Molecular cancer therapeutics (01.11.2017)
Published in Molecular cancer therapeutics (01.11.2017)
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Journal Article
Novel Noncatalytic Substrate-Selective p38α-Specific MAPK Inhibitors with Endothelial-Stabilizing and Anti-Inflammatory Activity
Shah, Nirav G, Tulapurkar, Mohan E, Ramarathnam, Aparna, Brophy, Amanda, Martinez, 3rd, Ramon, Hom, Kellie, Hodges, Theresa, Samadani, Ramin, Singh, Ishwar S, MacKerell, Jr, Alexander D, Shapiro, Paul, Hasday, Jeffrey D
Published in The Journal of immunology (1950) (15.04.2017)
Published in The Journal of immunology (1950) (15.04.2017)
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Journal Article
Importance of Domain Closure for the Autoactivation of ERK2
Barr, Daniel, Oashi, Taiji, Burkhard, Kimberly, Lucius, Sarah, Samadani, Ramin, Zhang, Jun, Shapiro, Paul, MacKerell, Alexander D, van der Vaart, Arjan
Published in Biochemistry (Easton) (20.09.2011)
Published in Biochemistry (Easton) (20.09.2011)
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Journal Article
Exosomal Proteome Profiling: A Potential Multi-Marker Cellular Phenotyping Tool to Characterize Hypoxia-Induced Radiation Resistance in Breast Cancer
Thomas, Stefani N, Liao, Zhongping, Clark, David, Chen, Yangyi, Samadani, Ramin, Mao, Li, Ann, David K, Baulch, Janet E, Shapiro, Paul, Yang, Austin J
Published in Proteomes (01.09.2013)
Published in Proteomes (01.09.2013)
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Journal Article
Book Review
CD73 Inhibitor Oleclumab Plus Osimertinib in Previously Treated Patients With Advanced T790M-Negative EGFR-Mutated NSCLC: A Brief Report
Kim, Dong-Wan, Kim, Sang-We, Camidge, D. Ross, Shu, Catherine A., Marrone, Kristen A., Le, Xiuning, Blakely, Collin M., Park, Keunchil, Chang, Gee-Chen, Patel, Sandip Pravin, Kar, Gozde, Cooper, Zachary A., Samadani, Ramin, Pluta, Michael, Kumar, Rakesh, Ramalingam, Suresh
Published in Journal of thoracic oncology (01.05.2023)
Published in Journal of thoracic oncology (01.05.2023)
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Journal Article
Mechanistic Analysis of an Extracellular Signal-Regulated Kinase 2-Interacting Compound that Inhibits Mutant BRAF-Expressing Melanoma Cells by Inducing Oxidative Stress
Martinez, 3rd, Ramon, Huang, Weiliang, Samadani, Ramin, Mackowiak, Bryan, Centola, Garrick, Chen, Lijia, Conlon, Ivie L, Hom, Kellie, Kane, Maureen A, Fletcher, Steven, Shapiro, Paul
Published in The Journal of pharmacology and experimental therapeutics (01.01.2021)
Published in The Journal of pharmacology and experimental therapeutics (01.01.2021)
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Journal Article
Abstract 3705: Overcoming drug resistance in BRaf mutated melanoma cells
Samadani, Ramin, Zhang, Jun, Mackerell, Alexander, Fletcher, Steven, Shapiro, Paul
Published in Cancer research (Chicago, Ill.) (01.10.2014)
Published in Cancer research (Chicago, Ill.) (01.10.2014)
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Journal Article
Discovery and Clinical Proof-of-Concept of RLY-2608, a First-in-Class Mutant-Selective Allosteric PI3Kα Inhibitor That Decouples Antitumor Activity from Hyperinsulinemia
Varkaris, Andreas, Pazolli, Ermira, Gunaydin, Hakan, Wang, Qi, Pierce, Levi, Boezio, Alessandro A, Bulku, Artemisa, DiPietro, Lucian, Fridrich, Cary, Frost, Adam, Giordanetto, Fabrizio, Hamilton, Erika P, Harris, Katherine, Holliday, Michael, Hunter, Tamieka L, Iskandar, Amanda, Ji, Yongli, Larivée, Alexandre, LaRochelle, Jonathan R, Lescarbeau, André, Llambi, Fabien, Lormil, Brenda, Mader, Mary M, Mar, Brenton G, Martin, Iain, McLean, Thomas H, Michelsen, Klaus, Pechersky, Yakov, Puente-Poushnejad, Erika, Raynor, Kevin, Rogala, Dipali, Samadani, Ramin, Schram, Alison M, Shortsleeves, Kelley, Swaminathan, Sweta, Tajmir, Shahein, Tan, Gege, Tang, Yong, Valverde, Roberto, Wehrenberg, Bryan, Wilbur, Jeremy, Williams, Bret R, Zeng, Hongtao, Zhang, Hanmo, Walters, W Patrick, Wolf, Beni B, Shaw, David E, Bergstrom, Donald A, Watters, James, Fraser, James S, Fortin, Pascal D, Kipp, D Randal
Published in Cancer discovery (08.02.2024)
Published in Cancer discovery (08.02.2024)
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Journal Article
Abstract CT163: CD73 inhibitor oleclumab plus osimertinib for advanced EGFRm NSCLC: First report of a Phase 1b/2 study
Kim, Dong-Wan, Kim, Sang-We, Camidge, D. Ross, Rizvi, Naiyer A., Marrone, Kristen A., Le, Xiuning, Blakely, Collin, Park, Keunchil, Chang, Gee-Chen, Patel, Sandip Pravin, Cooper, Zachary A., Kumar, Rakesh, Samadani, Ramin, McCombs, Rebecca, Pluta, Michael, Wu, Kevin Yufeng, Ramalingam, Suresh
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Published in Cancer research (Chicago, Ill.) (01.07.2021)
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Journal Article
Abstract PO3-20-04: A first-in-human study of the highly selective PI3Kα inhibitor RLY-5836 in patients with advanced breast cancer and other solid tumors
Varkaris, Andreas, Isakoff, Steven, Perez, Cesar A., O'Neil, Bert, Hamilton, Erika, Conlin, Erin, Tan, Gege, Li, Xiaoyan, Timm, Alison, Samadani, Ramin, Puente-Poushnejad, Erika, Kwak, Eunice, Mar, Brenton G., Schram, Alison M.
Published in Cancer research (Chicago, Ill.) (02.05.2024)
Published in Cancer research (Chicago, Ill.) (02.05.2024)
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Journal Article
Small-molecule inhibitors of ERK-mediated immediate early gene expression and proliferation of melanoma cells expressing mutated BRaf
Samadani, Ramin, Zhang, Jun, Brophy, Amanda, Oashi, Taiji, Priyakumar, U Deva, Raman, E Prabhu, St John, Franz J, Jung, Kwan-Young, Fletcher, Steven, Pozharski, Edwin, MacKerell, Jr, Alexander D, Shapiro, Paul
Published in Biochemical journal (01.05.2015)
Published in Biochemical journal (01.05.2015)
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Abstract OT3-22-01: First-in-human global multi-center study of RLY-2608, a pan mutant and isoform selective PI3Kα inhibitor, as a single agent in advanced solid tumor patients and in combination with fulvestrant in patients with advanced breast cancer
Varkaris, Andreas, Hamilton, Erika, Henry, Jason, Spira, Alexander I., Schram, Alison M., McGuinness, Julia E., Tan, Gege, Li, Xiaoyan, Hunter, Tamieka, Samadani, Ramin, Timm, Alison, Karanovic, Djuro, Subbiah, Vivek, Perez, Cesar A.
Published in Cancer research (Chicago, Ill.) (01.03.2023)
Published in Cancer research (Chicago, Ill.) (01.03.2023)
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Abstract PO3-20-03: First-in-human global study of RLY-2608, a pan-mutant and isoform selective PI3Kα inhibitor, as a single agent in patients with advanced solid tumors and in combination with fulvestrant in patients with advanced breast cancer
Varkaris, Andreas, Jhaveri, Komal, Cabanas, Elena Garralda, Sanz, Lucia, Kim, Janice, Perez, Cesar A., Hamilton, Erika, Spira, Alexander I., Wisinski, Kari, Guerrero, Angel, Henry, Jason, Ahnert, Jordi Rodon, Tan, Gege, Li, Xiaoyan, Hummel, Diana, Hunter, Tamieka, Timm, Alison, Samadani, Ramin, Puente-Poushnejad, Erika, Kwak, Eunice, Mar, Brenton G., Schram, Alison M.
Published in Cancer research (Chicago, Ill.) (02.05.2024)
Published in Cancer research (Chicago, Ill.) (02.05.2024)
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Journal Article
Stereo Matching and View Interpolation Based on Image Domain Triangulation : 3D VIDEO REPRESENTATION, COMPRESSION, AND RENDERING
FICKEL, Guilherme Pinto, JUNG, Claudio R, MALZBENDER, Tom, SAMADANI, Ramin, CULBERTSON, Bruce
Published in IEEE transactions on image processing (2013)
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Published in IEEE transactions on image processing (2013)
Journal Article
Structural modifications of (Z)-3-(2-aminoethyl)-5-(4-ethoxybenzylidene)thiazolidine-2,4-dione that improve selectivity for inhibiting the proliferation of melanoma cells containing active ERK signaling
Jung, Kwan-Young, Samadani, Ramin, Chauhan, Jay, Nevels, Kerrick, Yap, Jeremy L, Zhang, Jun, Worlikar, Shilpa, Lanning, Maryanna E, Chen, Lijia, Ensey, Mary, Shukla, Sagar, Salmo, Rosene, Heinzl, Geoffrey, Gordon, Caryn, Dukes, Troy, MacKerell, Jr, Alexander D, Shapiro, Paul, Fletcher, Steven
Published in Organic & biomolecular chemistry (14.06.2013)
Published in Organic & biomolecular chemistry (14.06.2013)
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Journal Article
견고한 심박수 추정
KULIK VICTOR, MARTIN RUSSEL ALLYN, SAMADANI RAMIN, PUIG CARLOS MANUEL
Year of Publication 27.12.2017
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Year of Publication 27.12.2017
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