Carbonic anhydrase inhibitors. Interaction of 2-(hydrazinocarbonyl)-3-phenyl-1H-indole-5-sulfonamide with 12 mammalian isoforms : Kinetic and X-ray crystallographic studies
GÜZEL, Ozlen, TEMPERINI, Claudia, INNOCENTI, Alessio, SCOZZAFAVA, Andrea, SALMAN, Aydin, SUPURAN, Claudiu T
Published in Bioorganic & medicinal chemistry (2008)
Published in Bioorganic & medicinal chemistry (2008)
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Journal Article
Carbonic anhydrase inhibitors : Synthesis and inhibition studies against mammalian isoforms I-XV with a series of 2-(hydrazinocarbonyl)-3-substituted-phenyl-1H-indole-5-sulfonamides
GÜZEL, Ozlen, INNOCENTI, Alessio, SCOZZAFAVA, Andrea, SALMAN, Aydin, PARKKILA, Seppo, HILVO, Mika, SUPURAN, Claudiu T
Published in Bioorganic & medicinal chemistry (15.10.2008)
Published in Bioorganic & medicinal chemistry (15.10.2008)
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Journal Article
Carbonic anhydrase inhibitors: Synthesis and inhibition studies against mammalian isoforms I-XV with a series of 2-(hydrazinocarbonyl)-3-substituted-phenyl-1H-indole-5-sulfonamide s
Guezel, Oezlen, Innocenti, Alessio, Scozzafava, Andrea, Salman, Aydin, Parkkila, Seppo, Hilvo, Mika, Supuran, Claudiu T
Published in Bioorganic & medicinal chemistry (01.10.2008)
Published in Bioorganic & medicinal chemistry (01.10.2008)
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Discovery of Low Nanomolar and Subnanomolar Inhibitors of the Mycobacterial β-Carbonic Anhydrases Rv1284 and Rv3273
Güzel, Özlen, Maresca, Alfonso, Scozzafava, Andrea, Salman, Aydın, Balaban, Alexandru T, Supuran, Claudiu T
Published in Journal of medicinal chemistry (09.07.2009)
Published in Journal of medicinal chemistry (09.07.2009)
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Carbonic anhydrase inhibitors. Aromatic/heterocyclic sulfonamides incorporating phenacetyl, pyridylacetyl and thienylacetyl tails act as potent inhibitors of human mitochondrial isoforms VA and VB
Güzel, Özlen, Innocenti, Alessio, Scozzafava, Andrea, Salman, Aydın, Supuran, Claudiu T.
Published in Bioorganic & medicinal chemistry (15.07.2009)
Published in Bioorganic & medicinal chemistry (15.07.2009)
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Carbonic anhydrase inhibitors. Phenacetyl-, pyridylacetyl- and thienylacetyl-substituted aromatic sulfonamides act as potent and selective isoform VII inhibitors
Güzel, Özlen, Innocenti, Alessio, Scozzafava, Andrea, Salman, Aydın, Supuran, Claudiu T.
Published in Bioorganic & medicinal chemistry letters (15.06.2009)
Published in Bioorganic & medicinal chemistry letters (15.06.2009)
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Synthesis and biological evaluation of new 4-thiazolidinone derivatives
Güzel, Özlen, Salman, Ayd n
Published in Journal of enzyme inhibition and medicinal chemistry (01.08.2009)
Published in Journal of enzyme inhibition and medicinal chemistry (01.08.2009)
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Carbonic anhydrase inhibitors. Synthesis of 2,4,6-trimethylpyridinium derivatives of 2-(hydrazinocarbonyl)-3-aryl-1H-indole-5-sulfonamides acting as potent inhibitors of the tumor-associated isoform IX and XII
Güzel, Özlen, Maresca, Alfonso, Scozzafava, Andrea, Salman, Aydın, Balaban, Alexandru T., Supuran, Claudiu T.
Published in Bioorganic & medicinal chemistry letters (01.06.2009)
Published in Bioorganic & medicinal chemistry letters (01.06.2009)
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ChemInform Abstract: Synthesis of New Spiroindolinones Incorporating a Benzothiazole Moiety as Antioxidant Agents
Karali, Nilguen, Guezel, Oezlen, Oezsoy, Nurten, Oezbey, Sueheyla, Salman, Aydin
Published in ChemInform (13.07.2010)
Published in ChemInform (13.07.2010)
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Carbonic anhydrase inhibitors: Synthesis and inhibition studies against mammalian isoforms I–XV with a series of 2-(hydrazinocarbonyl)-3-substituted-phenyl-1 H-indole-5-sulfonamides
Güzel, Özlen, Innocenti, Alessio, Scozzafava, Andrea, Salman, Aydın, Parkkila, Seppo, Hilvo, Mika, Supuran, Claudiu T.
Published in Bioorganic & medicinal chemistry (2008)
Published in Bioorganic & medicinal chemistry (2008)
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Midkine secretion protects Hep3B cells from cadmium induced cellular damage
Yazihan, Nuray, Ataoglu, Haluk, Akcil, Ethem, Yener, Burcu, Salman, Bulent, Aydin, Cengiz
Published in World journal of gastroenterology : WJG (07.01.2008)
Published in World journal of gastroenterology : WJG (07.01.2008)
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