A condensate-hardening drug blocks RSV replication in vivo
Risso-Ballester, Jennifer, Galloux, Marie, Cao, Jingjing, Le Goffic, Ronan, Hontonnou, Fortune, Jobart-Malfait, Aude, Desquesnes, Aurore, Sake, Svenja M., Haid, Sibylle, Du, Miaomiao, Zhang, Xiumei, Zhang, Huanyun, Wang, Zhaoguo, Rincheval, Vincent, Zhang, Youming, Pietschmann, Thomas, Eléouët, Jean-François, Rameix-Welti, Marie-Anne, Altmeyer, Ralf
Published in Nature (London) (22.07.2021)
Published in Nature (London) (22.07.2021)
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Journal Article
Labyrinthopeptins as virolytic inhibitors of respiratory syncytial virus cell entry
Blockus, Sebastian, Sake, Svenja M., Wetzke, Martin, Grethe, Christina, Graalmann, Theresa, Pils, Marina, Le Goffic, Ronan, Galloux, Marie, Prochnow, Hans, Rox, Katharina, Hüttel, Stephan, Rupcic, Zeljka, Wiegmann, Bettina, Dijkman, Ronald, Rameix-Welti, Marie-Anne, Eléouët, Jean-François, Duprex, W Paul, Thiel, Volker, Hansen, Gesine, Brönstrup, Mark, Haid, Sibylle, Pietschmann, Thomas
Published in Antiviral research (01.05.2020)
Published in Antiviral research (01.05.2020)
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Journal Article
Protecting-Group-Mediated Diastereoselective Synthesis of C4′-Methylated Uridine Analogs and Their Activity against the Human Respiratory Syncytial Virus
Köllmann, Christoph, Sake, Svenja M, Jones, Peter G, Pietschmann, Thomas, Werz, Daniel B
Published in Journal of organic chemistry (20.03.2020)
Published in Journal of organic chemistry (20.03.2020)
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Journal Article
Repurposing screen identifies novel candidates for broad-spectrum coronavirus antivirals and druggable host targets
Haid, Sibylle, Matthaei, Alina, Winkler, Melina, Sake, Svenja M, Gunesch, Antonia P, Milke, Vanessa, Köhler, Natalie M, Rückert, Jessica, Vieyres, Gabrielle, Kühl, David, Nguyen, Tu-Trinh, Göhl, Matthias, Lasswitz, Lisa, Zapatero-Belinchón, Francisco J, Brogden, Graham, Gerold, Gisa, Wiegmann, Bettina, Bilitewski, Ursula, Brown, Richard J P, Brönstrup, Mark, Schulz, Thomas F, Pietschmann, Thomas
Published in Antimicrobial agents and chemotherapy (06.03.2024)
Published in Antimicrobial agents and chemotherapy (06.03.2024)
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Journal Article
Respiratory Syncytial Virus Two-Step Infection Screen Reveals Inhibitors of Early and Late Life Cycle Stages
Sake, Svenja M, Kosch, Christina, Blockus, Sebastian, Haid, Sibylle, Gunesch, Antonia P, Zhang, Xiaoyu, Friesland, Martina, Trummer, Sofie B, Grethe, Christina, Kühnel, Anne, Rückert, Jessica, Duprex, W Paul, Huang, Jiabin, Rameix-Welti, Marie-Anne, Empting, Martin, Fischer, Nicole, Hirsch, Anna K H, Schulz, Thomas F, Pietschmann, Thomas
Published in Antimicrobial agents and chemotherapy (20.12.2022)
Published in Antimicrobial agents and chemotherapy (20.12.2022)
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Journal Article
Drug repurposing screen identifies lonafarnib as respiratory syncytial virus fusion protein inhibitor
Sake, Svenja M., Zhang, Xiaoyu, Rajak, Manoj Kumar, Urbanek-Quaing, Melanie, Carpentier, Arnaud, Gunesch, Antonia P., Grethe, Christina, Matthaei, Alina, Rückert, Jessica, Galloux, Marie, Larcher, Thibaut, Le Goffic, Ronan, Hontonnou, Fortune, Chatterjee, Arnab K., Johnson, Kristen, Morwood, Kaycie, Rox, Katharina, Elgaher, Walid A. M., Huang, Jiabin, Wetzke, Martin, Hansen, Gesine, Fischer, Nicole, Eléouët, Jean-Francois, Rameix-Welti, Marie-Anne, Hirsch, Anna K. H., Herold, Elisabeth, Empting, Martin, Lauber, Chris, Schulz, Thomas F., Krey, Thomas, Haid, Sibylle, Pietschmann, Thomas
Published in Nature communications (08.02.2024)
Published in Nature communications (08.02.2024)
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Journal Article
Drug repurposing screen identifies lonafarnib as respiratory syncytial virus fusion protein inhibitor
Sake, Svenja M, Zhang, Xiaoyu, Rajak, Manoj Kumar, Urbanek-Quaing, Melanie, Carpentier, Arnaud, Gunesch, Antonia P, Grethe, Christina, Matthaei, Alina, Rückert, Jessica, Galloux, Marie, Larcher, Thibaut, Le Goffic, Ronan, Hontonnou, Fortune, Chatterjee, Arnab K, Johnson, Kristen, Morwood, Kaycie, Rox, Katharina, Elgaher, Walid a M, Huang, Jiabin, Wetzke, Martin, Hansen, Gesine, Fischer, Nicole, Éléouët, Jean-François, Rameix-Welti, Marie-Anne, Hirsch, Anna K H, Herold, Elisabeth, Empting, Martin, Lauber, Chris, Schulz, Thomas F, Krey, Thomas, Haid, Sibylle, Pietschmann, Thomas
Published in Nature communications (08.02.2024)
Published in Nature communications (08.02.2024)
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Journal Article
Liver-expressed Cd302 and Cr1l limit hepatitis C virus cross-species transmission to mice
Brown, Richard J P, Tegtmeyer, Birthe, Sheldon, Julie, Khera, Tanvi, Anggakusuma, Todt, Daniel, Vieyres, Gabrielle, Weller, Romy, Joecks, Sebastian, Zhang, Yudi, Sake, Svenja, Bankwitz, Dorothea, Welsch, Kathrin, Ginkel, Corinne, Engelmann, Michael, Gerold, Gisa, Steinmann, Eike, Yuan, Qinggong, Ott, Michael, Vondran, Florian W R, Krey, Thomas, Ströh, Luisa J, Miskey, Csaba, Ivics, Zoltán, Herder, Vanessa, Baumgärtner, Wolfgang, Lauber, Chris, Seifert, Michael, Tarr, Alexander W, McClure, C Patrick, Randall, Glenn, Baktash, Yasmine, Ploss, Alexander, Thi, Viet Loan Dao, Michailidis, Eleftherios, Saeed, Mohsan, Verhoye, Lieven, Meuleman, Philip, Goedecke, Natascha, Wirth, Dagmar, Rice, Charles M, Pietschmann, Thomas
Published in Science advances (01.11.2020)
Published in Science advances (01.11.2020)
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Journal Article
LONAFARNIB FOR USE IN THE TREATMENT OF VIRAL INFECTIONS
HAID, Sibylle, SCHULZ, Thomas, PIETSCHMANN, Thomas, SAKE, Svenja, RÜCKERT, Jessica
Year of Publication 21.03.2024
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Year of Publication 21.03.2024
Patent
LONAFARNIB FOR USE IN THE TREATMENT OF VIRAL INFECTIONS
HAID, Sibylle, SCHULZ, Thomas, PIETSCHMANN, Thomas, SAKE, Svenja, RÜCKERT, Jessica
Year of Publication 29.11.2023
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Year of Publication 29.11.2023
Patent
LONAFARNIB FOR USE IN THE TREATMENT OF VIRAL INFECTIONS
HAID, Sibylle, SCHULZ, Thomas, PIETSCHMANN, Thomas, SAKE, Svenja, RÜCKERT, Jessica
Year of Publication 28.07.2022
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Year of Publication 28.07.2022
Patent
LONAFARNIB FOR USE IN THE TREATMENT OF VIRAL INFECTIONS
HAID, Sibylle, SCHULZ, Thomas, PIETSCHMANN, Thomas, SAKE, Svenja, RÜCKERT, Jessica
Year of Publication 27.07.2022
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Year of Publication 27.07.2022
Patent