Progress towards a public chemogenomic set for protein kinases and a call for contributions
Drewry, David H, Wells, Carrow I, Andrews, David M, Angell, Richard, Al-Ali, Hassan, Axtman, Alison D, Capuzzi, Stephen J, Elkins, Jonathan M, Ettmayer, Peter, Frederiksen, Mathias, Gileadi, Opher, Gray, Nathanael, Hooper, Alice, Knapp, Stefan, Laufer, Stefan, Luecking, Ulrich, Michaelides, Michael, Müller, Susanne, Muratov, Eugene, Denny, R Aldrin, Saikatendu, Kumar S, Treiber, Daniel K, Zuercher, William J, Willson, Timothy M
Published in PloS one (02.08.2017)
Published in PloS one (02.08.2017)
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The Kinase Chemogenomic Set (KCGS): An Open Science Resource for Kinase Vulnerability Identification
Wells, Carrow I, Al-Ali, Hassan, Andrews, David M, Asquith, Christopher R M, Axtman, Alison D, Dikic, Ivan, Ebner, Daniel, Ettmayer, Peter, Fischer, Christian, Frederiksen, Mathias, Futrell, Robert E, Gray, Nathanael S, Hatch, Stephanie B, Knapp, Stefan, Lücking, Ulrich, Michaelides, Michael, Mills, Caitlin E, Müller, Susanne, Owen, Dafydd, Picado, Alfredo, Saikatendu, Kumar S, Schröder, Martin, Stolz, Alexandra, Tellechea, Mariana, Turunen, Brandon J, Vilar, Santiago, Wang, Jinhua, Zuercher, William J, Willson, Timothy M, Drewry, David H
Published in International journal of molecular sciences (08.01.2021)
Published in International journal of molecular sciences (08.01.2021)
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Proteomics Analysis Unravels the Functional Repertoire of Coronavirus Nonstructural Protein 3
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Published in Journal of Virology (01.06.2008)
Published in Journal of Virology (01.06.2008)
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Nuclear Magnetic Resonance Structure of the N-Terminal Domain of Nonstructural Protein 3 from the Severe Acute Respiratory Syndrome Coronavirus
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Published in Journal of Virology (01.11.2007)
Published in Journal of Virology (01.11.2007)
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Discovery of 7‑Oxo-2,4,5,7-tetrahydro‑6H‑pyrazolo[3,4‑c]pyridine Derivatives as Potent, Orally Available, and Brain-Penetrating Receptor Interacting Protein 1 (RIP1) Kinase Inhibitors: Analysis of Structure–Kinetic Relationships
Yoshikawa, Masato, Saitoh, Morihisa, Katoh, Taisuke, Seki, Tomohiro, Bigi, Simone V, Shimizu, Yuji, Ishii, Tsuyoshi, Okai, Takuro, Kuno, Masako, Hattori, Harumi, Watanabe, Etsuro, Saikatendu, Kumar S, Zou, Hua, Nakakariya, Masanori, Tatamiya, Takayuki, Nakada, Yoshihisa, Yogo, Takatoshi
Published in Journal of medicinal chemistry (22.03.2018)
Published in Journal of medicinal chemistry (22.03.2018)
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Journal Article
Discovery of 7-Oxo-2,4,5,7-tetrahydro-6 H-pyrazolo[3,4- c]pyridine Derivatives as Potent, Orally Available, and Brain-Penetrating Receptor Interacting Protein 1 (RIP1) Kinase Inhibitors: Analysis of Structure-Kinetic Relationships
Yoshikawa, Masato, Saitoh, Morihisa, Katoh, Taisuke, Seki, Tomohiro, Bigi, Simone V, Shimizu, Yuji, Ishii, Tsuyoshi, Okai, Takuro, Kuno, Masako, Hattori, Harumi, Watanabe, Etsuro, Saikatendu, Kumar S, Zou, Hua, Nakakariya, Masanori, Tatamiya, Takayuki, Nakada, Yoshihisa, Yogo, Takatoshi
Published in Journal of medicinal chemistry (22.03.2018)
Published in Journal of medicinal chemistry (22.03.2018)
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Exploiting high-energy hydration sites for the discovery of potent peptide aldehyde inhibitors of the SARS-CoV-2 main protease with cellular antiviral activity
Carney, Daniel W., Leffler, Abba E., Bell, Jeffrey A., Chandrasinghe, Asela S., Cheng, Cecilia, Chang, Edcon, Dornford, Adam, Dougan, Douglas R., Frye, Leah L., Grimes, Mary E., Knehans, Tim, Knight, Jennifer L., Komandla, Mallareddy, Lane, Weston, Li, Hubert, Newman, Sophia R., Phimister, Katalin, Saikatendu, Kumar S., Silverstein, Hercules, Vafaei, Shaghayegh
Published in Bioorganic & medicinal chemistry (01.04.2024)
Published in Bioorganic & medicinal chemistry (01.04.2024)
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Functional Proteomic and Structural Insights into Molecular Recognition in the Nitrilase Family Enzymes
Barglow, Katherine T, Saikatendu, Kumar S, Bracey, Michael H, Huey, Ruth, Morris, Garrett M, Olson, Arthur J, Stevens, Raymond C, Cravatt, Benjamin F
Published in Biochemistry (Easton) (23.12.2008)
Published in Biochemistry (Easton) (23.12.2008)
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The Kinase Chemogenomic Set (KCGS): An open science resource for kinase vulnerability identification
Wells, Carrow I, Al-Ali, Hassan, Andrews, David M, Asquith, Christopher Robert Michael, Axtman, Alison D, Chung, Mirra, Dikic, Ivan, Ebner, Daniel, Elkins, Jon, Ettmayer, Peter, Fischer, Christian, Frederiksen, Mathias, Gray, Nathanael S, Hatch, Stephanie B, Knapp, Stefan, Lee, Shudong, Lucking, Ulrich, Michaelides, Michael, Mills, Caitlin E, Muller, Susanne, Owen, Dafydd, Picado, Alfredo, Ramadan, Kristijan, Saikatendu, Kumar S, Schroder, Martin, Stolz, Alexandra, Tellechea, Maria, Treiber, Daniel K, Turunen, Brandon J, Vilar, Santiago, Wang, Jinhua, Zuercher, William, Willson, Timothy M, Drewry, David H
Published in bioRxiv (23.12.2019)
Published in bioRxiv (23.12.2019)
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Paper
Progress Towards a Public Chemogenomic Set for Protein Kinases and a Call for Contributions
Drewry, David H, Wells, Carrow I, Andrews, David M, Angell, Richard, Al-Ali, Hassan, Axtman, Alison D, Capuzzi, Stephen J, Elkins, Jonathan M, Ettmayer, Peter, Frederiksen, Mathias, Gileadi, Opher, Gray, Nathanael, Hooper, Alice, Knapp, Stefan, Laufer, Stefan, Luecking, Ulrich, Muller, Susanne, Muratov, Eugene, R Aldrin Denny, Saikatendu, Kumar S, Treiber, Daniel K, Zuercher, William J, Willson, Timothy M
Published in bioRxiv (31.01.2017)
Published in bioRxiv (31.01.2017)
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