Novel dual LSD1/HDAC6 inhibitor for the treatment of cancer
Gajendran, Chandru, Tantry, Subramanyam Janardhan, M, Naveen Sadhu, Mohammed, Zainuddin, Dewang, Purushottam, Hallur, Mahanandeesha, Nair, Sreekala, Vaithilingam, Krishnakumar, Nagayya, Basavaprabhu, Rajagopal, Sridharan, Sivanandhan, Dhanalakshmi
Published in PloS one (03.01.2023)
Published in PloS one (03.01.2023)
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Journal Article
Novel dual LSD1/HDAC6 inhibitors for the treatment of multiple myeloma
Naveen Sadhu, M, Sivanandhan, Dhanalakshmi, Gajendran, Chandru, Tantry, Subramanyam, Dewang, Purushottam, Murugan, Kannan, Chickamunivenkatappa, Srinatha, Zainuddin, Mohd, Nair, Sreekala, Vaithilingam, Krishnakumar, Rajagopal, Sridharan
Published in Bioorganic & medicinal chemistry letters (15.02.2021)
Published in Bioorganic & medicinal chemistry letters (15.02.2021)
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Journal Article
Alleviation of arthritis through prevention of neutrophil extracellular traps by an orally available inhibitor of protein arginine deiminase 4
Gajendran, Chandru, Fukui, Shoichi, Sadhu, Naveen M, Zainuddin, Mohammed, Rajagopal, Sridharan, Gosu, Ramachandraiah, Gutch, Sarah, Fukui, Saeko, Sheehy, Casey E, Chu, Long, Vishwakarma, Santosh, Jeyaraj, D A, Hallur, Gurulingappa, Wagner, Denisa D, Sivanandhan, Dhanalakshmi
Published in Scientific reports (23.02.2023)
Published in Scientific reports (23.02.2023)
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Journal Article
A Novel Selective Inhibitor JBI-589 Targets PAD4-Mediated Neutrophil Migration to Suppress Tumor Progression
Deng, Hui, Lin, Cindy, Garcia-Gerique, Laura, Fu, Shuyu, Cruz, Zachary, Bonner, Erin E, Rosenwasser, Matthew, Rajagopal, Sridharan, Sadhu, M Naveen, Gajendran, Chandru, Zainuddin, Mohd, Gosu, Ramachandraiah, Sivanandhan, Dhanalakshmi, Shelef, Miriam A, Nam, Brian, Vogl, Dan T, Gabrilovich, Dmitry I, Nefedova, Yulia
Published in Cancer research (Chicago, Ill.) (04.10.2022)
Published in Cancer research (Chicago, Ill.) (04.10.2022)
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Journal Article
PD1/PD-L1 억제제로서의 화합물 및 이의 방법
MOHD ZAINUDDIN, SADHU NAVEEN, SIVANANDHAN DHANALAKSHMI, RAJAGOPAL SRIDHARAN
Year of Publication 31.01.2024
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Year of Publication 31.01.2024
Patent
Abstract 1128: Selective, novel, small molecule PRMT5 inhibitors for treatment of cancer
Sivanandhan, Dhanalakshmi, Rajagopal, Sridharan, M, Naveen Sadhu, Gajendran, Chandru, Vadivelu, Saravanan, Tamizharasan, Natarajan, Swamy, Indu N., Viswakarma, Santhosh, Siddiqui, Amir, wahid, Saif, Zainuddin, Mohammed, G, Rudresh, Daram, Prashanthi, Gosu, Ramchandraiah, Tiagaraj, Dinesh, Garapaty, Shivani, Nair, Sreekala, Kapoor, Namratha
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Published in Cancer research (Chicago, Ill.) (01.07.2021)
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Journal Article
Abstract 1630: Novel, small molecule inhibitors of PD-L1/PD-1 interaction
Sivanandhan, Dhanalakshmi, Rajagopal, Sridharan, M, Naveen Sadhu, Gajendran, Chandru, venkateshappa, Chandregowda, Reddy, Muralidhar, Kishore, Pendyala Satya, Deshpande, Pratima, kannan, Sundarajan, Sahareen, Tabassum, Viswakarma, Santhosh, Siddiqui, Amir, Zainuddin, Mohammed, G, Rudresh, Daram, Prashanthi, Gosu, Ramchandraiah, Devi, Rashmi Rekha
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Published in Cancer research (Chicago, Ill.) (01.07.2021)
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Journal Article
Novel, small molecule inhibitors of PD-1/PD-L1 pathway
Rastelli, Luca, Rajagopal, Sridharan, Gajendran, Chandru, Sadhu, Naveen M., Mohd, Zainuddin, Gosu, Ramachandraiah, Friedmann-Morvinski, Dinorah, Kandan, Saravanan, Birudukota, Swarnakumari, S, Srinivasan, V, Krishnakumar, Wahid, Saif, Siddiqui, Amir, Viswakarma, Santosh, Narayan, Ashwini, G, Rudresh, Mullurwar, Sadanand R., Sher, Divsha, Mansur, Shahar, Sivanandhan, Dhanalakshmi
Published in Journal of clinical oncology (01.06.2022)
Published in Journal of clinical oncology (01.06.2022)
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Journal Article
Abstract B029: LSD1-HDAC6 dual inhibitor JBI-802 is an epigenetic modulating agent with a novel mechanism of action that target MYC amplification in multiple neuroendocrine tumor types
Sivanandhan, Dhanalakshmi, Rajagopal, Sridharan, Gajendran, Chandru, Sadhu, Naveen, Zainuddin, Mohd, Gosu, Ramachandraiah, Rastelli, Luca
Published in Cancer research (Chicago, Ill.) (01.12.2022)
Published in Cancer research (Chicago, Ill.) (01.12.2022)
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Journal Article
1386 Novel gut-restricted small molecule inhibitor of PD-L1 for targeting GI cancers
Sivanandhan, Dhanalakshmi, Sridharan Rajagopal, Gajendran, Chandru, Naveen, Sadhu M, Zainuddin, Mohammed, Ramachandraiah Gosu, Rastelli, Luca
Published in Journal for immunotherapy of cancer (01.11.2022)
Published in Journal for immunotherapy of cancer (01.11.2022)
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Journal Article
Abstract 6269: JBI-778, a novel brain-penetrant small molecule PRMT5 inhibitor for treatment of cancer
Sivanandhan, Dhanalakshmi, Gajendran, Chandru, M, Naveen Sadhu, Mohammed, Zainuddin, Gosu, Ramachandraiah, Sher, Divsha, Mansur, Shahar, Friedmann-Morvinski, Dinorah, Rajagopal, Sridharan, Rastelli, Luca
Published in Cancer research (Chicago, Ill.) (04.04.2023)
Published in Cancer research (Chicago, Ill.) (04.04.2023)
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Journal Article
Abstract 2646: Novel, isoform selective PAD4 inhibitors for the treatment of cancer
Sivanandhan, Dhanalakshmi, Rajagopal, Sridharan, G, Chandru, Zainuddin, Mohd, Sadhu, Naveen, Gosu, Ramachandraiah, Rastelli, Luca, Siddiqui, Amir, Singh, Sharad, G, Rudresh, Mullurwar, Sadanand, Kandan, Saravanan, Vishwakarma, Santosh, Hallur, Gurulingappa, Trivedi, Ravi, A, Jeyaraj D
Published in Cancer research (Chicago, Ill.) (15.06.2022)
Published in Cancer research (Chicago, Ill.) (15.06.2022)
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Journal Article
DUAL LSD1/HDAC INHIBITORS
GAJENDRAN, Chandru, SIVANANDHAN, Dhanalakshmi, RASTELLI, Luca, SADHU, Naveen, SRIDHARAN, Rajagopal
Year of Publication 15.08.2024
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Year of Publication 15.08.2024
Patent
COMPOUNDS AS PD1/PD-L1 INHIBITORS AND METHODS THEREOF
SIVANANDHAN, Dhanalakshmi, SADHU, Naveen, MOHD, Zainuddin, RAJAGOPAL, Sridharan
Year of Publication 25.07.2024
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Year of Publication 25.07.2024
Patent
COMPOUNDS AS PD1/PD-L1 INHIBITORS AND METHODS THEREOF
SIVANANDHAN, Dhanalakshmi, SADHU, Naveen, MOHD, Zainuddin, RAJAGOPAL, Sridharan
Year of Publication 28.02.2024
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Year of Publication 28.02.2024
Patent
Compounds as pd1/pd-l1 inhibitors and methods thereof
SIVANANDHAN Dhanalakshmi, MOHD Zainuddin, RAJAGOPAL Sridharan, SADHU Naveen
Year of Publication 01.12.2023
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Year of Publication 01.12.2023
Patent
COMPOUNDS AS PD1/PD-L1 INHIBITORS AND METHODS THEREOF
SIVANANDHAN, Dhanalakshmi, SADHU, Naveen, MOHD, Zainuddin, RAJAGOPAL, Sridharan
Year of Publication 19.10.2023
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Year of Publication 19.10.2023
Patent
DUAL LSD1/HDAC INHIBITORS
GAJENDRAN, Chandru, SIVANANDHAN, Dhanalakshmi, RASTELLI, Luca, SADHU, Naveen, SRIDHARAN, Rajagopal
Year of Publication 14.09.2023
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Year of Publication 14.09.2023
Patent
COMPOUNDS AS PD1/PD-L1 INHIBITORS AND METHODS THEREOF
SIVANANDHAN, Dhanalakshmi, SADHU, Naveen, MOHD, Zainuddin, RAJAGOPAL, Sridharan
Year of Publication 27.10.2022
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Year of Publication 27.10.2022
Patent
COMPOUNDS AS PD1/PD-L1 INHIBITORS AND METHODS THEREOF
MOHD, ZAINUDDIN, SIVANANDHAN, DHANALAKSHMI, RAJAGOPAL, SRIDHARAN, SADHU, NAVEEN
Year of Publication 27.10.2022
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Year of Publication 27.10.2022
Patent