Assessment of Prognostic Indicators and Survival-Based Impact of Holistic Approach in Oral Cancer Patients: An Observational Study
Kandalkar, Sachin S, Sharma, Manish, Ahirrao, Bhagyashri, Kanna, Abdul Suban A, Sheikh, Tauseef A, Ziauddin, Saudagar M
Published in Curēus (Palo Alto, CA) (19.08.2024)
Published in Curēus (Palo Alto, CA) (19.08.2024)
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Journal Article
Modifications of flexible nonyl chain and nucleobase head group of (+)-erythro-9-(2′s-hydroxy-3′s-nonyl)adenine [(+)-EHNA] as adenosine deaminase inhibitors
Kandalkar, Sachin R., Ramaiah, Parimi Atchuta, Joshi, Manoj, Wavhal, Atul, Waman, Yogesh, Raje, Amol A., Tambe, Ashwini, Ansari, Shariq, De, Siddhartha, Palle, Venkata P., Mookhtiar, Kasim A., Deshpande, Anil M., Barawkar, Dinesh A.
Published in Bioorganic & medicinal chemistry (15.10.2017)
Published in Bioorganic & medicinal chemistry (15.10.2017)
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Journal Article
Discovery of liver-directed glucokinase activator having anti-hyperglycemic effect without hypoglycemia
Deshpande, Anil M., Bhuniya, Debnath, De, Siddhartha, Dave, Bhavesh, Vyavahare, Vinod P., Kurhade, Santosh H., Kandalkar, Sachin R., Naik, Keshav P., Kobal, Balasaheb S., Kaduskar, Rahul D., Basu, Sujay, Jain, Vaibhav, Patil, Pratima, Chaturvedi Joshi, Sandhya, Bhat, Ganesh, Raje, Amol A., Reddy, Satyanarayana, Gundu, Jayasagar, Madgula, Vamsi, Tambe, Suhas, Shitole, Prasad, Umrani, Dhananjay, Chugh, Anita, Palle, Venkata P., Mookhtiar, Kasim A.
Published in European journal of medicinal chemistry (16.06.2017)
Published in European journal of medicinal chemistry (16.06.2017)
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Journal Article
Highly efficient one-pot amination of carboxylate-substituted nitrogen-containing heteroaryl chlorides via Staudinger reaction
Kandalkar, Sachin R., Kaduskar, Rahul D., Ramaiah, Parimi Atchuta, Barawkar, Dinesh A., Bhuniya, Debnath, Deshpande, Anil M.
Published in Tetrahedron letters (30.01.2013)
Published in Tetrahedron letters (30.01.2013)
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Journal Article
Potent and Selective Inhibitors of Long Chain l-2-Hydroxy Acid Oxidase Reduced Blood Pressure in DOCA Salt-Treated Rats
Barawkar, Dinesh A, Meru, Ashwin, Bandyopadhyay, Anish, Banerjee, Abir, Deshpande, Anil M, Athare, Chandrashekhar, Koduru, Chandrasekhar, Khose, Goraksha, Gundu, Jayasagar, Mahajan, Koshu, Patil, Pradeep, Kandalkar, Sachin R, Niranjan, Sanjay, Bhosale, Shubhangi, De, Siddhartha, Mukhopadhyay, Sudit, Chaudhary, Sumit, Koul, Summon, Singh, Umesh, Chugh, Anita, Palle, Venkata P, Mookhtiar, Kasim A, Vacca, Joseph, Chakravarty, Prasun K, Nargund, Ravi P, Wright, Samuel D, Roy, Sophie, Graziano, Michael P, Singh, Sheo B, Cully, Doris, Cai, Tian-Quan
Published in ACS medicinal chemistry letters (08.12.2011)
Published in ACS medicinal chemistry letters (08.12.2011)
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Journal Article
Development of Tunable Mechanism-Based Carbasugar Ligands that Stabilize Glycoside Hydrolases through the Formation of Transient Covalent Intermediates
Bhosale, Sandeep, Kandalkar, Sachin, Gilormini, Pierre-André, Akintola, Oluwafemi, Rowland, Rhianna, Adabala, Pal John Pal, King, Dustin, Deen, Matthew C., Chen, Xi, Davies, Gideon J., Vocadlo, David J., Bennet, Andrew J.
Published in ACS catalysis (20.09.2024)
Published in ACS catalysis (20.09.2024)
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Journal Article
ChemInform Abstract: Highly Efficient One-Pot Amination of Carboxylate-Substituted Nitrogen-Containing Heteroaryl Chlorides via Staudinger Reaction
Kandalkar, Sachin R., Kaduskar, Rahul D., Ramaiah, Parimi Atchuta, Barawkar, Dinesh A., Bhuniya, Debnath, Deshpande, Anil M.
Published in ChemInform (28.05.2013)
Published in ChemInform (28.05.2013)
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Journal Article
RBx-0597, a potent, selective and slow-binding inhibitor of dipeptidyl peptidase-IV for the treatment of type 2 diabetes
Singh, Shuchita, Sethi, Sachin, Khanna, Vivek, Benjamin, Biju, Kant, Rajiv, Sattigeri, Jitendra, Bansal, Vinay S, Bhatnagar, Pradip Kumar, Davis, Joseph Alex
Published in European journal of pharmacology (10.02.2011)
Published in European journal of pharmacology (10.02.2011)
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Journal Article
Discovery of pyrazole carboxylic acids as potent inhibitors of rat long chain l-2-hydroxy acid oxidase
Barawkar, Dinesh A., Bandyopadhyay, Anish, Deshpande, Anil, Koul, Summon, Kandalkar, Sachin, Patil, Pradeep, Khose, Goraksha, Vyas, Samir, Mone, Mahesh, Bhosale, Shubhangi, Singh, Umesh, De, Siddhartha, Meru, Ashwin, Gundu, Jayasagar, Chugh, Anita, Palle, Venkata P., Mookhtiar, Kasim A., Vacca, Joseph P., Chakravarty, Prasun K., Nargund, Ravi P., Wright, Samuel D., Roy, Sophie, Graziano, Michael P., Cully, Doris, Cai, Tian-Quan, Singh, Sheo B.
Published in Bioorganic & medicinal chemistry letters (01.07.2012)
Published in Bioorganic & medicinal chemistry letters (01.07.2012)
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Journal Article
Erratum to “RBx-0597, a potent, selective and slow-binding inhibitor of dipeptidyl peptidase-IV for the treatment of type 2 diabetes” [European Journal of Pharmacology 652 (1–3) (2011) 157–163]
Singh, Shuchita, Roy, Subhasis, Sethi, Sachin, Benjamin, Biju, Sundaram, Sindhuja, Khanna, Vivek, Kandalkar, Sachin R., Pal, Chanchal, Kant, Rajiv, Patra, Ashok Kumar, Rayasam, Geetavani, Mittra, Shivani, Saini, Kulvinder Singh, Paliwal, Jyoti, Chugh, Anita, Ahmed, Shahadat, Sattigeri, Jitendra, Cliff, Ian, Ray, Abhijit, Bansal, Vinay S., Bhatnagar, Pradip Kumar, Davis, Joseph Alex
Published in European journal of pharmacology (01.03.2011)
Published in European journal of pharmacology (01.03.2011)
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Journal Article
Derivados de acetamida como ativadores de glicoquinase, seu processo e aplicações medicinais
KESHAV NAIK, ANIL DESHPANDE, VENKATA POORNAPRAGNACHARYULU PALLE, BHAVESH DAVE, SIDDHARTHA DE, SANTOSH KURHADE, SANDEEP BHAUSAHEB BHOSALE, BALASAHEB KOBAL, GOBIND SING KAPKOTI, KASIM A. MOOKHTIAR, SACHIN KANDALKAR, DEBANATH BHUNIYA
Year of Publication 22.04.2015
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Year of Publication 22.04.2015
Patent
BENZAMIDE COMPOUNDS AS GLUCOKINASE ACTIVATORS AND THEIR PHARMACEUTICAL APPLICATION
DAVE, BHAVESH, NAIK, KESHAV, BHUNIYA, DEBNATH, DESHPANDE, ANIL, PALLE, VENKATA, KANDALKAR, SACHIN
Year of Publication 11.08.2011
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Year of Publication 11.08.2011
Patent
ACETAMIDE DERIVATIVES AS GLUCOKINASE ACTIVATORS, THEIR PROCESS AND MEDICINAL APPLICATIONS
DAVE, BHAVESH, VENKATA, POORNAPRAGNACHARYULU PALLE, NAIK, KESHAV, MOOKHTIAR, KASIM A, KOBAL, BALASAHEB, GOBIND, SING KAPKOTI, DE, SIDDHARTHA, DESHPANDE, ANIL, KURHADE, SANTOSH, KANDALKAR, SACHIN, BHUNIYA, DEBANATH, SANDEEP, BHAUSAHEB BHOSALE
Year of Publication 17.03.2015
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Year of Publication 17.03.2015
Patent
ACETAMIDE DERIVATIVES AS GLUCOKINASE ACTIVATORS, THEIR PROCESS AND MEDICINAL APPLICATIONS
BHOSALE, SANDEEP, BHAUSAHEB, DAVE, BHAVESH, NAIK, KESHAV, MOOKHTIAR, KASIM A, KOBAL, BALASAHEB, PALLE, VENKATA, POORNAPRAGNACHARYULU, DE, SIDDHARTHA, DESHPANDE, ANIL, KURHADE, SANTOSH, KANDALKAR, SACHIN, KAPKOTI, GOBIND, SING, BHUNIYA, DEBANATH
Year of Publication 08.01.2014
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Year of Publication 08.01.2014
Patent