Predicting protein targets for drug-like compounds using transcriptomics
Pabon, Nicolas A, Xia, Yan, Estabrooks, Samuel K, Ye, Zhaofeng, Herbrand, Amanda K, Süß, Evelyn, Biondi, Ricardo M, Assimon, Victoria A, Gestwicki, Jason E, Brodsky, Jeffrey L, Camacho, Carlos J, Bar-Joseph, Ziv
Published in PLoS computational biology (01.12.2018)
Published in PLoS computational biology (01.12.2018)
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Bidirectional Allosteric Communication between the ATP-Binding Site and the Regulatory PIF Pocket in PDK1 Protein Kinase
Schulze, Jörg O., Saladino, Giorgio, Busschots, Katrien, Neimanis, Sonja, Süß, Evelyn, Odadzic, Dalibor, Zeuzem, Stefan, Hindie, Valerie, Herbrand, Amanda K., Lisa, María-Natalia, Alzari, Pedro M., Gervasio, Francesco L., Biondi, Ricardo M.
Published in Cell chemical biology (20.10.2016)
Published in Cell chemical biology (20.10.2016)
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Modulation of the substrate specificity of the kinase PDK1 by distinct conformations of the full-length protein
Sacerdoti, Mariana, Gross, Lissy Z F, Riley, Andrew M, Zehnder, Karin, Ghode, Abhijeet, Klinke, Sebastián, Anand, Ganesh Srinivasan, Paris, Kristina, Winkel, Angelika, Herbrand, Amanda K, Godage, H Yasmin, Cozier, Gyles E, Süß, Evelyn, Schulze, Jörg O, Pastor-Flores, Daniel, Bollini, Mariela, Cappellari, María Victoria, Svergun, Dmitri, Gräwert, Melissa A, Aramendia, Pedro F, Leroux, Alejandro E, Potter, Barry V L, Camacho, Carlos J, Biondi, Ricardo M
Published in Science signaling (13.06.2023)
Published in Science signaling (13.06.2023)
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Modulation of the Allosteric Communication between the Polo-Box Domain and the Catalytic Domain in Plk1 by Small Compounds
Raab, Monika, Sanhaji, Mourad, Pietsch, Larissa, Béquignon, Isabelle, Herbrand, Amanda K, Süß, Evelyn, Gande, Santosh L, Caspar, Birgit, Kudlinzki, Denis, Saxena, Krishna, Sreeramulu, Sridhar, Schwalbe, Harald, Strebhardt, Klaus, Biondi, Ricardo M
Published in ACS chemical biology (17.08.2018)
Published in ACS chemical biology (17.08.2018)
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An Allosteric Inhibitor Scaffold Targeting the PIF-Pocket of Atypical Protein Kinase C Isoforms
Arencibia, Jose M, Fröhner, Wolfgang, Krupa, Magdalena, Pastor-Flores, Daniel, Merker, Piotr, Oellerich, Thomas, Neimanis, Sonja, Schmithals, Christian, Köberle, Verena, Süß, Evelyn, Zeuzem, Stefan, Stark, Holger, Piiper, Albrecht, Odadzic, Dalibor, Schulze, Jörg O, Biondi, Ricardo M
Published in ACS chemical biology (17.02.2017)
Published in ACS chemical biology (17.02.2017)
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PIF-Pocket as a Target for C. albicans Pkh Selective Inhibitors
Pastor-Flores, Daniel, Schulze, Jörg O, Bahí, Anna, Giacometti, Romina, Ferrer-Dalmau, Jofre, Passeron, Susana, Engel, Matthias, Süß, Evelyn, Casamayor, Antonio, Biondi, Ricardo M
Published in ACS chemical biology (18.10.2013)
Published in ACS chemical biology (18.10.2013)
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Allosteric Regulation of Protein Kinase PKCζ by the N-Terminal C1 Domain and Small Compounds to the PIF-Pocket
Lopez-Garcia, Laura A., Schulze, Jörg O., Fröhner, Wolfgang, Zhang, Hua, Süß, Evelyn, Weber, Nadja, Navratil, Jeanette, Amon, Sabine, Hindie, Valerie, Zeuzem, Stefan, Jørgensen, Thomas J.D., Alzari, Pedro M., Neimanis, Sonja, Engel, Matthias, Biondi, Ricardo M.
Published in Chemistry & biology (23.11.2011)
Published in Chemistry & biology (23.11.2011)
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