Synthesis and structure-affinity relationship investigations of 5-aminomethyl and 5-carbamoyl analogues of the antipsychotic sertindole. A new class of selective α1 adrenoceptor antagonists
BALLE, Thomas, PERREGAARD, Jens, LARSEN, Anna K, RAMIREZ, Martha Teresa, SØBY, Karina Krøjer, LILJEFORS, Tommy, ANDERSEN, Kim
Published in Bioorganic & medicinal chemistry (01.03.2003)
Published in Bioorganic & medicinal chemistry (01.03.2003)
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Journal Article
Synthesis and Structure−Affinity Relationship Investigations of 5-Heteroaryl-Substituted Analogues of the Antipsychotic Sertindole. A New Class of Highly Selective α1 Adrenoceptor Antagonists
Balle, Thomas, Perregaard, Jens, Ramirez, Martha Teresa, Larsen, Anna Kirstine, Søby, Karina Krøjer, Liljefors, Tommy, Andersen, Kim
Published in Journal of medicinal chemistry (16.01.2003)
Published in Journal of medicinal chemistry (16.01.2003)
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Journal Article
Synthesis and structure-affinity relationship investigations of 5-heteroaryl-substituted analogues of the antipsychotic sertindole. A new class of highly selective alpha(1) adrenoceptor antagonists
Balle, T, Perregaard, J, Ramirez, MT, Larsen, AK, Soby, KK, Liljefors, T, Andersen, K
Published in Journal of medicinal chemistry (16.01.2003)
Published in Journal of medicinal chemistry (16.01.2003)
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Journal Article
α1 Adrenoceptor subtype selectivity
Balle, Thomas, Andersen, Kim, Søby, Karina Krøjer, Liljefors, Tommy
Published in Journal of molecular graphics & modelling (01.06.2003)
Published in Journal of molecular graphics & modelling (01.06.2003)
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Journal Article
Alpha(1) adrenoceptor subtype selectivity. 3D-QSAR models for a new class of alpha(1) adrenoceptor antagonists derived from the novel antipsychotic sertindole
Balle, Thomas, Andersen, Kim, Søby, Karina Krøjer, Liljefors, Tommy
Published in Journal of molecular graphics & modelling (01.06.2003)
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Published in Journal of molecular graphics & modelling (01.06.2003)
Journal Article
α 1 Adrenoceptor subtype selectivity : 3D-QSAR models for a new class of α 1 adrenoceptor antagonists derived from the novel antipsychotic sertindole
Balle, Thomas, Andersen, Kim, Søby, Karina Krøjer, Liljefors, Tommy
Published in Journal of molecular graphics & modelling (2003)
Published in Journal of molecular graphics & modelling (2003)
Get full text
Journal Article
Synthesis and Structure−Affinity Relationship Investigations of 5-Heteroaryl-Substituted Analogues of the Antipsychotic Sertindole. A New Class of Highly Selective α 1 Adrenoceptor Antagonists
Balle, Thomas, Perregaard, Jens, Ramirez, Martha Teresa, Larsen, Anna Kirstine, Søby, Karina Krøjer, Liljefors, Tommy, Andersen, Kim
Published in Journal of medicinal chemistry (01.01.2003)
Published in Journal of medicinal chemistry (01.01.2003)
Get full text
Journal Article
Synthesis and structure-affinity relationship investigations of 5-aminomethyl and 5-carbamoyl analogues of the antipsychotic sertindole. A new class of selective alpha1 adrenoceptor antagonists
Balle, Thomas, Perregaard, Jens, Larsen, Anna K, Ramirez, Martha Teresa, Krøjer Søby, Karina, Liljefors, Tommy, Andersen, Kim
Published in Bioorganic & medicinal chemistry (20.03.2003)
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Published in Bioorganic & medicinal chemistry (20.03.2003)
Journal Article
Synthesis and structure–affinity relationship investigations of 5-aminomethyl and 5-carbamoyl analogues of the antipsychotic sertindole. A new class of selective α 1 adrenoceptor antagonists
Balle, Thomas, Perregaard, Jens, Larsen, Anna K., Ramirez, Martha Teresa, Krøjer Søby, Karina, Liljefors, Tommy, Andersen, Kim
Published in Bioorganic & medicinal chemistry (2003)
Published in Bioorganic & medicinal chemistry (2003)
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Journal Article
ALCOHOL DERIVATIVES AS KV7 POTASSIUM CHANNEL OPENERS FOR USE IN EPILEPSY OR SEIZURES
Wang, Xiaofang, Ivkovic, Jelena, Sams, Anette Graven, Hong, Jian, Bastlund, Jesper Frank, Larsen, Morten Grupe, Rottlãnder, Mario, Chen, Shu Hui, Das, Debasis, Søby, Karina Krøjer
Year of Publication 08.09.2022
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Year of Publication 08.09.2022
Patent
ALCOHOL DERIVATIVES AS KV7 POTASSIUM CHANNEL OPENERS FOR USE IN EPILEPSY OR SEIZURES
SAMS, Anette, Graven, WANG, Xiaofang, CHEN, Shu, Hui, BASTLUND, Jesper, Frank, DAS, Debasis, IVKOVIC, Jelena, HONG, Jian, SØBY, Karina, Krøjer, LARSEN, Morten, Grupe, ROTTLÄNDER, Mario
Year of Publication 08.06.2022
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Year of Publication 08.06.2022
Patent