Highly Selective Inhibitors of Dipeptidyl Peptidase 9 (DPP9) Derived from the Clinically Used DPP4-Inhibitor Vildagliptin
Benramdane, Siham, De Loose, Joni, Filippi, Nicolò, Espadinha, Margarida, Beyens, Olivier, Rymenant, Yentl Van, Dirkx, Laura, Bozdag, Murat, Feijens, Pim-Bart, Augustyns, Koen, Caljon, Guy, De Winter, Hans, De Meester, Ingrid, Van der Veken, Pieter
Published in Journal of medicinal chemistry (28.09.2023)
Published in Journal of medicinal chemistry (28.09.2023)
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Journal Article
Vildagliptin‐Derived Dipeptidyl Peptidase 9 (DPP9) Inhibitors: Identification of a DPP8/9‐Specific Lead
Benramdane, Siham, De Loose, Joni, Beyens, Olivier, Van Rymenant, Yentl, Vliegen, Gwendolyn, Augustyns, Koen, De Winter, Hans, De Meester, Ingrid, Van der Veken, Pieter
Published in ChemMedChem (03.08.2022)
Published in ChemMedChem (03.08.2022)
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Journal Article
Novel Generation of FAP Inhibitor-Based Homodimers for Improved Application in Radiotheranostics
Martin, Marcel, Ballal, Sanjana, Yadav, Madhav Prasad, Bal, Chandrasekhar, Van Rymenant, Yentl, De Loose, Joni, Verhulst, Emile, De Meester, Ingrid, Van Der Veken, Pieter, Roesch, Frank
Published in Cancers (21.03.2023)
Published in Cancers (21.03.2023)
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Journal Article
In Vitro Evaluation of the Squaramide-Conjugated Fibroblast Activation Protein Inhibitor-Based Agents AAZTA5.SA.FAPi and DOTA.SA.FAPi
Moon, Euy Sung, Van Rymenant, Yentl, Battan, Sandeep, De Loose, Joni, Bracke, An, Van der Veken, Pieter, De Meester, Ingrid, Rösch, Frank
Published in Molecules (Basel, Switzerland) (08.06.2021)
Published in Molecules (Basel, Switzerland) (08.06.2021)
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Journal Article
In Vitro and In Situ Activity-Based Labeling of Fibroblast Activation Protein with UAMC1110-Derived Probes
Van Rymenant, Yentl, Tanc, Muhammet, Van Elzen, Roos, Bracke, An, De Wever, Olivier, Augustyns, Koen, Lambeir, Anne-Marie, Kockx, Mark, De Meester, Ingrid, Van Der Veken, Pieter
Published in Frontiers in chemistry (14.04.2021)
Published in Frontiers in chemistry (14.04.2021)
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Journal Article
Synthesis and evaluation of a fluorinated PET imaging probe targeting fibroblast activation protein (FAP)
Filippi, Nicolò, Van Rymenant, Yentl, Cianni, Lorenzo, Stroobants, Sigrid, De Meester, Ingrid, Van der Veken, Pieter, Elvas, Filipe
Published in Nuclear medicine and biology (01.11.2023)
Published in Nuclear medicine and biology (01.11.2023)
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Journal Article
Druglike, 18 F-labeled PET Tracers Targeting Fibroblast Activation Protein
Tanc, Muhammet, Filippi, Nicolò, Van Rymenant, Yentl, Grintsevich, Sergei, Pintelon, Isabel, Verschuuren, Marlies, De Loose, Joni, Verhulst, Emile, Moon, Euy Sung, Cianni, Lorenzo, Stroobants, Sigrid, Augustyns, Koen, Roesch, Frank, De Meester, Ingrid, Elvas, Filipe, Van der Veken, Pieter
Published in Journal of medicinal chemistry (09.05.2024)
Published in Journal of medicinal chemistry (09.05.2024)
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Journal Article
Active site-directed probes targeting dipeptidyl peptidases 8 and 9
Espadinha, Margarida, De Loose, Joni, Corthaut, Sam, Thys, Sofie, Van Rymenant, Yentl, Verhulst, Emile, Benramdane, Siham, Filippi, Nicolò, Augustyns, Koen, Van Wielendaele, Pieter, Pintelon, Isabel, De Meester, Ingrid, Van der Veken, Pieter
Published in European journal of medicinal chemistry (15.04.2024)
Published in European journal of medicinal chemistry (15.04.2024)
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Journal Article
Druglike, 18F‑labeled PET Tracers Targeting Fibroblast Activation Protein
Tanc, Muhammet, Filippi, Nicolò, Van Rymenant, Yentl, Grintsevich, Sergei, Pintelon, Isabel, Verschuuren, Marlies, De Loose, Joni, Verhulst, Emile, Moon, Euy Sung, Cianni, Lorenzo, Stroobants, Sigrid, Augustyns, Koen, Roesch, Frank, De Meester, Ingrid, Elvas, Filipe, Van der Veken, Pieter
Published in Journal of medicinal chemistry (09.05.2024)
Published in Journal of medicinal chemistry (09.05.2024)
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Next generation fibroblast activation protein (FAP) targeting PET tracers - The tetrazine ligation allows an easy and convenient way to 18F-labeled (4-quinolinoyl)glycyl-2-cyanopyrrolidines
Poulie, Christian B.M., Shalgunov, Vladimir, Elvas, Filipe, Van Rymenant, Yentl, Moon, Euy-Sung, Battisti, Umberto Maria, De Loose, Joni, De Meester, Ingrid, Rösch, Frank, Van Der Veken, Pieter, Herth, Matthias M.
Published in European journal of medicinal chemistry (15.12.2023)
Published in European journal of medicinal chemistry (15.12.2023)
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Journal Article
Fibroblast Activation Protein (FAP) targeting homodimeric FAP inhibitor radiotheranostics: a step to improve tumor uptake and retention time
Moon, Euy Sung, Ballal, Sanjana, Yadav, Madhav Prasad, Bal, Chandrasekhar, Van Rymenant, Yentl, Stephan, Sarah, Bracke, An, Van der Veken, Pieter, De Meester, Ingrid, Roesch, Frank
Published in American journal of nuclear medicine and molecular imaging (01.01.2021)
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Published in American journal of nuclear medicine and molecular imaging (01.01.2021)
Journal Article
Intercellular interaction between FAP+ fibroblasts and CD150+ inflammatory monocytes mediates fibrostenosis in Crohn's disease
Ke, Bo-Jun, Abdurahiman, Saeed, Biscu, Francesca, Zanella, Gaia, Dragoni, Gabriele, Santhosh, Sneha, De Simone, Veronica, Zouzaf, Anissa, van Baarle, Lies, Stakenborg, Michelle, Bosáková, Veronika, Van Rymenant, Yentl, Verhulst, Emile, Verstockt, Sare, Klein, Elliott, Bislenghi, Gabriele, Wolthuis, Albert, Frič, Jan, Breynaert, Christine, D'Hoore, Andre, Van der Veken, Pieter, De Meester, Ingrid, Lovisa, Sara, Hawinkels, Lukas Jac, Verstockt, Bram, De Hertogh, Gert, Vermeire, Séverine, Matteoli, Gianluca
Published in The Journal of clinical investigation (23.07.2024)
Published in The Journal of clinical investigation (23.07.2024)
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Journal Article
SP-012 - Fluorinated PET imaging probes targeting fibroblast activation protein: radiolabeling and preclinical evaluation
Elvas, Filipe, Tanc, Muhammet, Van Rymenant, Yentl, Beroske, Lucas, De Lombaerde, Stef, Augustyns, Koen, Staelens, Steven, Stroobants, Sigrid, De Meester, Ingrid, Van der Veken, Pieter
Published in Nuclear medicine and biology (01.05.2021)
Published in Nuclear medicine and biology (01.05.2021)
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Journal Article
Fluorinated PET imaging probes targeting fibroblast activation protein: radiolabeling and preclinical evaluation
Elvas, Filipe, Tanc, Muhammet, Van Rymenant, Yentl, Beroske, Lucas, De Lombaerde, Stef, Augustyns, Koen, Staelens, Steven, Stroobants, Sigrid, De Meester, Ingrid, Van der Veken, Pieter
Published in Nuclear medicine and biology (01.05.2021)
Published in Nuclear medicine and biology (01.05.2021)
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Journal Article
INHIBITORS OF FIBROBLAST ACTIVATION PROTEIN
AUGUSTYNS, Koen, TANÇ, Muhammet, VAN RYMENANT, Yentl, DE MEESTER, Ingrid, ELVAS, Filipe, GRINTSEVICH, Sergei, STROOBANTS, Sigrid, CIANNI, Lorenzo, BEROSKE, Lucas, FILIPPI, Nicolò, VAN DER VEKEN, Pieter
Year of Publication 07.12.2023
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Year of Publication 07.12.2023
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